메뉴 건너뛰기




Volumn 21, Issue 5, 1999, Pages 507-513

Effects of chronic administration of glucocorticoid on midazolam pharmacokinetics in humans

Author keywords

CYP3A4; Drug interaction; Induction; UDP glucuronosyltransferase

Indexed keywords

GLUCOCORTICOID; GLUCURONOSYLTRANSFERASE; MIDAZOLAM;

EID: 0032836340     PISSN: 01634356     EISSN: None     Source Type: Journal    
DOI: 10.1097/00007691-199910000-00003     Document Type: Article
Times cited : (22)

References (31)
  • 1
    • 0028237729 scopus 로고
    • Interindividual variations in human liver cytochrome P-450 enzymes involved in the oxidation of drugs, carcinogens and toxic chemicals: Studies with liver microsomes of 30 Japanese and 30 Caucasians
    • Shimada T, Yamazaki H, Mimura M, et al. Interindividual variations in human liver cytochrome P-450 enzymes involved in the oxidation of drugs, carcinogens and toxic chemicals: studies with liver microsomes of 30 Japanese and 30 Caucasians. J. Pharmacol Exp Ther 1994;270:414-23.
    • (1994) J. Pharmacol Exp Ther , vol.270 , pp. 414-423
    • Shimada, T.1    Yamazaki, H.2    Mimura, M.3
  • 2
    • 0028054999 scopus 로고
    • Extrahepatic metabolism of drug in humans
    • Krishna DR, Klotz U. Extrahepatic metabolism of drug in humans. Clin Pharmacokinet 1994;26:144-60.
    • (1994) Clin Pharmacokinet , vol.26 , pp. 144-160
    • Krishna, D.R.1    Klotz, U.2
  • 3
    • 0029738490 scopus 로고    scopus 로고
    • First-pass metabolism of midazolam by the human intestine
    • Paine MF, Shen DD, Kunze KL, et al. First-pass metabolism of midazolam by the human intestine. Clin Pharmacol Ther 1996;60: 14-24.
    • (1996) Clin Pharmacol Ther , vol.60 , pp. 14-24
    • Paine, M.F.1    Shen, D.D.2    Kunze, K.L.3
  • 4
    • 0030015297 scopus 로고    scopus 로고
    • Oral first-pass elimination of midazolam involves both gastrointestinal and hepatic CYP3A-mediated metabolism
    • Thummel KE, O'Shea D, Paine MF, et al. Oral first-pass elimination of midazolam involves both gastrointestinal and hepatic CYP3A-mediated metabolism. Clin Pharmacol Ther 1996;59: 491-502.
    • (1996) Clin Pharmacol Ther , vol.59 , pp. 491-502
    • Thummel, K.E.1    O'Shea, D.2    Paine, M.F.3
  • 6
    • 0026629650 scopus 로고
    • Pharmacokinetics of midazolem administered by continuous intravenous infusion to intensive care patients
    • Malacrida R, Fritz ME, Suter PM, Crevoisier C. Pharmacokinetics of midazolem administered by continuous intravenous infusion to intensive care patients. Crit Care Med 1992;20:1123-6.
    • (1992) Crit Care Med , vol.20 , pp. 1123-1126
    • Malacrida, R.1    Fritz, M.E.2    Suter, P.M.3    Crevoisier, C.4
  • 8
    • 0024373348 scopus 로고
    • Oxidation of midazolam and triazolam by human liver cytochrome P-450IIIA4
    • Kronbach T, Mathys D, Umeno M, et al. Oxidation of midazolam and triazolam by human liver cytochrome P-450IIIA4. Mol Pharmacol 1989;36:89-96.
    • (1989) Mol Pharmacol , vol.36 , pp. 89-96
    • Kronbach, T.1    Mathys, D.2    Umeno, M.3
  • 9
    • 0025999285 scopus 로고
    • In vitro forecasting of drugs which may interfere with the biotransformation of midazolam
    • Gascon MP, Dayer P. In vitro forecasting of drugs which may interfere with the biotransformation of midazolam. Eur J Clin Pharmacol 1991;41:573-8.
    • (1991) Eur J Clin Pharmacol , vol.41 , pp. 573-578
    • Gascon, M.P.1    Dayer, P.2
  • 10
    • 0028361593 scopus 로고
    • Inhibition of human CYP3A catalyzed l'-hydroxy midazolam formation by ketoconazole, nifedipine, erythromycin, cimetidine and nizatidine
    • Wrighton SA, Ring BJ. Inhibition of human CYP3A catalyzed l'-hydroxy midazolam formation by ketoconazole, nifedipine, erythromycin, cimetidine and nizatidine. Pharm Res 1994;11: 921-4.
    • (1994) Pharm Res , vol.11 , pp. 921-924
    • Wrighton, S.A.1    Ring, B.J.2
  • 11
    • 0028126571 scopus 로고
    • Midazolam is metabolized by at least three different cytochrome P450 enzymes
    • Wandel C, Böcker R, Böhrer H, et al. Midazolam is metabolized by at least three different cytochrome P450 enzymes. Br J Anaesth 1994;73:658-61.
    • (1994) Br J Anaesth , vol.73 , pp. 658-661
    • Wandel, C.1    Böcker, R.2    Böhrer, H.3
  • 12
    • 0027985506 scopus 로고
    • Use of midazolam as a human cytochrome P450-3A probe: II. Characterization of interand intraindividual hepatic CYP3A variability after liver transplantation
    • Thummel KE, Shen DD, Podoll TD, et al. Use of midazolam as a human cytochrome P450-3A probe: II. Characterization of interand intraindividual hepatic CYP3A variability after liver transplantation. J Pharmacol Exp Ther 1994;271:557-66.
    • (1994) J Pharmacol Exp Ther , vol.271 , pp. 557-566
    • Thummel, K.E.1    Shen, D.D.2    Podoll, T.D.3
  • 13
    • 0028114619 scopus 로고
    • Use of midazolam as a human cytochrome P4503A probe: I. In vitro-in vivo correlations in liver transplant patients
    • Thummel KE, Shen DD, Podoll TD, et al. Use of midazolam as a human cytochrome P4503A probe: I. In vitro-in vivo correlations in liver transplant patients. J Pharmacol Exp Ther 1994;271:549-56.
    • (1994) J Pharmacol Exp Ther , vol.271 , pp. 549-556
    • Thummel, K.E.1    Shen, D.D.2    Podoll, T.D.3
  • 14
    • 0028357256 scopus 로고
    • Midazolam should be avoided in patients receiving the systemic antimycotics ketoconazole or itraconazole
    • Olkkola KT, Backman JT, Neuvonen PJ. Midazolam should be avoided in patients receiving the systemic antimycotics ketoconazole or itraconazole. Clin Pharmacol Ther 1994;55:481-5.
    • (1994) Clin Pharmacol Ther , vol.55 , pp. 481-485
    • Olkkola, K.T.1    Backman, J.T.2    Neuvonen, P.J.3
  • 15
    • 0029664974 scopus 로고    scopus 로고
    • The effect of systemic antimycotics, itraconazole and fluconazole, on the pharmacokinetics and pharmcodynamics of intravenous and oral midazolam
    • Olkkola KT, Ahonen J, Neuvonen PJ. The effect of systemic antimycotics, itraconazole and fluconazole, on the pharmacokinetics and pharmcodynamics of intravenous and oral midazolam. Anesth Analg 1996;82:511-6.
    • (1996) Anesth Analg , vol.82 , pp. 511-516
    • Olkkola, K.T.1    Ahonen, J.2    Neuvonen, P.J.3
  • 16
    • 0027477751 scopus 로고
    • A potentially hazardous interaction between erythromycin and midazolam
    • Olkkola KT, Aranko K, Luurila H, et al. A potentially hazardous interaction between erythromycin and midazolam. Clin Pharmacol Ther 1993;53:298-305.
    • (1993) Clin Pharmacol Ther , vol.53 , pp. 298-305
    • Olkkola, K.T.1    Aranko, K.2    Luurila, H.3
  • 17
    • 0030030330 scopus 로고    scopus 로고
    • Concentration and effects of oral midazolam are greatly reduced in patients treated with carbamazepine or phenytoin
    • Backman JT, Olkkola KT, Ojala M, et al. Concentration and effects of oral midazolam are greatly reduced in patients treated with carbamazepine or phenytoin. Epilepsia 1996;37:253-7.
    • (1996) Epilepsia , vol.37 , pp. 253-257
    • Backman, J.T.1    Olkkola, K.T.2    Ojala, M.3
  • 18
    • 0030068752 scopus 로고    scopus 로고
    • Rifampin drastically reduces plasma concentrations and effects of oral midazolam
    • Backman JT, Olkkola KT, Neuvonen PJ. Rifampin drastically reduces plasma concentrations and effects of oral midazolam. Clin Phamacol Ther 1996;59:7-13.
    • (1996) Clin Phamacol Ther , vol.59 , pp. 7-13
    • Backman, J.T.1    Olkkola, K.T.2    Neuvonen, P.J.3
  • 19
    • 0041301863 scopus 로고
    • Identification of an inducible form of cytochrome P-450 in human liver
    • Watkins PB, Wrighton SA, Maurel P, et al. Identification of an inducible form of cytochrome P-450 in human liver. Proc Natl Acad Sci USA 1985;82:6310-4.
    • (1985) Proc Natl Acad Sci USA , vol.82 , pp. 6310-6314
    • Watkins, P.B.1    Wrighton, S.A.2    Maurel, P.3
  • 20
    • 0024556650 scopus 로고
    • Erythromycin breath test as an assay of glucocorticoid-inducible liver cytochrome P-450
    • Watkins PB, Murray SA, Winkelman LG, et al. Erythromycin breath test as an assay of glucocorticoid-inducible liver cytochrome P-450. J Clin Invest 1989;83:688-97.
    • (1989) J Clin Invest , vol.83 , pp. 688-697
    • Watkins, P.B.1    Murray, S.A.2    Winkelman, L.G.3
  • 21
    • 0027050416 scopus 로고
    • Effect of corticosteroids on the expression of cytochromes P450 and on cyclosporin A oxidase in primary cultures of human hepatocytes
    • Pichard L, Fabre I, Daujat M, et al. Effect of corticosteroids on the expression of cytochromes P450 and on cyclosporin A oxidase in primary cultures of human hepatocytes. Mol Pharmacol 1992;41: 1047-55.
    • (1992) Mol Pharmacol , vol.41 , pp. 1047-1055
    • Pichard, L.1    Fabre, I.2    Daujat, M.3
  • 22
    • 0022421630 scopus 로고
    • Determination of midazolam (Versed®) and its metabolites in plasma by high-performance liquid chromatography
    • Puglisi CV, Pao J, Ferrara FJ, deSilva JAF. Determination of midazolam (Versed®) and its metabolites in plasma by high-performance liquid chromatography. J Chromatogr 1985;344:199-209.
    • (1985) J Chromatogr , vol.344 , pp. 199-209
    • Puglisi, C.V.1    Pao, J.2    Ferrara, F.J.3    DeSilva, J.A.F.4
  • 24
    • 0021192084 scopus 로고
    • Effects of age, gender, and obesity on midazolam kinetics
    • Greenblatt DJ, Abernethy DR, Locniskar A, et al. Effects of age, gender, and obesity on midazolam kinetics. Anesthesioloqy 1984; 61:27-35.
    • (1984) Anesthesioloqy , vol.61 , pp. 27-35
    • Greenblatt, D.J.1    Abernethy, D.R.2    Locniskar, A.3
  • 25
    • 0022973593 scopus 로고
    • p in primary monolayer cultures of adult rat hepatocytes and in human liver
    • p in primary monolayer cultures of adult rat hepatocytes and in human liver. J Biol Chem 1986;261:8270-5.
    • (1986) J Biol Chem , vol.261 , pp. 8270-8275
    • Schuetz, E.G.1    Hazelton, G.A.2    Hall, J.3
  • 26
    • 0027160090 scopus 로고
    • Differential effects of human recombinant interleukin-1β and dexamethasone on hepatic drug-metabolizing enzymes in male and female rats
    • Ferrari L, Herber R, Batt A-M, Siest G. Differential effects of human recombinant interleukin-1β and dexamethasone on hepatic drug-metabolizing enzymes in male and female rats. Biochem Pharmacol 1993;45:2269-77.
    • (1993) Biochem Pharmacol , vol.45 , pp. 2269-2277
    • Ferrari, L.1    Herber, R.2    Batt, A.-M.3    Siest, G.4
  • 27
    • 0021963088 scopus 로고
    • Dexamethasone increase UDP-glucuronyltransferase activity towards bilirubin, oestradial and testosterone in foetal liver from rhesus monkey during late gestation
    • Leakey JEA, Althaus ZR, Bailey JR, Slikker WJr. Dexamethasone increase UDP-glucuronyltransferase activity towards bilirubin, oestradial and testosterone in foetal liver from rhesus monkey during late gestation. Biochem J 1985;225:183-8.
    • (1985) Biochem J , vol.225 , pp. 183-188
    • Leakey, J.E.A.1    Althaus, Z.R.2    Bailey, J.R.3    Slikker W., Jr.4
  • 28
    • 0027264759 scopus 로고
    • The effects of inducing agents on cytochrome P450 and UDP-glucuronyltransferase activities in human HepG2 hepatoma cells
    • Doostdar H, Grant MH, Melvin WT, Wolf CR. The effects of inducing agents on cytochrome P450 and UDP-glucuronyltransferase activities in human HepG2 hepatoma cells. Biochem Pharmacol 1993;46:629-35.
    • (1993) Biochem Pharmacol , vol.46 , pp. 629-635
    • Doostdar, H.1    Grant, M.H.2    Melvin, W.T.3    Wolf, C.R.4
  • 30
    • 0029972195 scopus 로고    scopus 로고
    • The nifedipinerifampin interaction. Evidence for induction of gut wall metabolism
    • Holtbecker N, Fromm MF, Kroemer HK, et al. The nifedipinerifampin interaction. Evidence for induction of gut wall metabolism. Drug Metab Dispos 1996;24:1121-3.
    • (1996) Drug Metab Dispos , vol.24 , pp. 1121-1123
    • Holtbecker, N.1    Fromm, M.F.2    Kroemer, H.K.3
  • 31
    • 0026464616 scopus 로고
    • Identification of rifampin-inducible P450IIIA4 (CYP3A4) in human small bowel enterocytes
    • Kolars JC, Schmiedlin-Ren P, Schetz JD, Fang C, Watkins PB. Identification of rifampin-inducible P450IIIA4 (CYP3A4) in human small bowel enterocytes. J Clin Invest 1992;90:1871-8.
    • (1992) J Clin Invest , vol.90 , pp. 1871-1878
    • Kolars, J.C.1    Schmiedlin-Ren, P.2    Schetz, J.D.3    Fang, C.4    Watkins, P.B.5


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.