-
1
-
-
0009644628
-
Some quantitative uses of drug antagonists
-
Arunlakshana O, Schild HO (1959) Some quantitative uses of drug antagonists. Br J Pharmacol 14: 48-58
-
(1959)
Br J Pharmacol
, vol.14
, pp. 48-58
-
-
Arunlakshana, O.1
Schild, H.O.2
-
2
-
-
0024308134
-
Drug discrimination in pentylenetetrazole-trained baboons: Generalization to buspirone and beta-CCE but not lorazepam or pentobarbital
-
Ator NA, Cook JM, Griffiths RR (1989) Drug discrimination in pentylenetetrazole-trained baboons: Generalization to buspirone and beta-CCE but not lorazepam or pentobarbital. Drug Dev Res 16:257-267
-
(1989)
Drug Dev Res
, vol.16
, pp. 257-267
-
-
Ator, N.A.1
Cook, J.M.2
Griffiths, R.R.3
-
3
-
-
0028358846
-
Discriminative-stimulus effects of azaspirodecanedione anxiolytics in baboons trained to discriminate β-carboline-3-carboxylic acid ethyl ester or pentylenetetrazole
-
Ator NA, Cook JM, Allen MS, Griffiths RR (1994) Discriminative-stimulus effects of azaspirodecanedione anxiolytics in baboons trained to discriminate β-carboline-3-carboxylic acid ethyl ester or pentylenetetrazole. Behav Pharmacol 5:176-188
-
(1994)
Behav Pharmacol
, vol.5
, pp. 176-188
-
-
Ator, N.A.1
Cook, J.M.2
Allen, M.S.3
Griffiths, R.R.4
-
4
-
-
0019996866
-
Interaction of convulsive ligands with benzodiazepine receptors
-
Braestrup C, Schmiechen R, Neef G, Nielsen M, Petersen EN (1982) Interaction of convulsive ligands with benzodiazepine receptors. Science 216:1241-1243
-
(1982)
Science
, vol.216
, pp. 1241-1243
-
-
Braestrup, C.1
Schmiechen, R.2
Neef, G.3
Nielsen, M.4
Petersen, E.N.5
-
5
-
-
0023709743
-
Intrinsic activity and the discriminative effects of drugs
-
Colpaert FC, Balster RL (eds) Transduction mechanisms of drug stimuli Springer, Berlin Heidelberg New York
-
Colpaert FC (1988) Intrinsic activity and the discriminative effects of drugs. In: Colpaert FC, Balster RL (eds) Transduction mechanisms of drug stimuli (Psychopharmacology series 4). Springer, Berlin Heidelberg New York, pp 154-160
-
(1988)
Psychopharmacology Series
, vol.4
, pp. 154-160
-
-
Colpaert, F.C.1
-
6
-
-
0019513358
-
Ethyl β-carboline carboxylate lowers seizure threshold and antagonizes flurazepam-induced sedation in rats
-
Cowen PJ, Green AR, Martin IL, Nutt DJ (1981) Ethyl β-carboline carboxylate lowers seizure threshold and antagonizes flurazepam-induced sedation in rats. Nature 290:54-55
-
(1981)
Nature
, vol.290
, pp. 54-55
-
-
Cowen, P.J.1
Green, A.R.2
Martin, I.L.3
Nutt, D.J.4
-
7
-
-
0026564355
-
Discriminative stimulus properties of RU 33965, a benzodiazepine receptor weak partial inverse agonist
-
Gardner CR, Budhram P, Parker FL (1992) Discriminative stimulus properties of RU 33965, a benzodiazepine receptor weak partial inverse agonist. Pharmacol Biochem Behav 43:583-588
-
(1992)
Pharmacol Biochem Behav
, vol.43
, pp. 583-588
-
-
Gardner, C.R.1
Budhram, P.2
Parker, F.L.3
-
8
-
-
0028224691
-
Discriminative stimulus properties of the benzodiazepine receptor inverse agonist methyl-6,7-dimethoxy-4-ethyl-β-carboline-3-carboxylate (DMCM)
-
Kirby LG, Rowan GA, Smith RL, Lucki I (1994) Discriminative stimulus properties of the benzodiazepine receptor inverse agonist methyl-6,7-dimethoxy-4-ethyl-β-carboline-3-carboxylate (DMCM). Psychopharmacology 113:351-360
-
(1994)
Psychopharmacology
, vol.113
, pp. 351-360
-
-
Kirby, L.G.1
Rowan, G.A.2
Smith, R.L.3
Lucki, I.4
-
9
-
-
0022981542
-
β-carbolines selectively antagonize the cholecystokinin action in isolated guinea-pig gallbladder muscle
-
Kubota K, Itonaga M (1986) β-carbolines selectively antagonize the cholecystokinin action in isolated guinea-pig gallbladder muscle. Jpn J Pharmacol 42:501-506
-
(1986)
Jpn J Pharmacol
, vol.42
, pp. 501-506
-
-
Kubota, K.1
Itonaga, M.2
-
11
-
-
0024156974
-
Discriminative stimulus control by the anxiogenic beta-carboline FG 7142: Generalization to a physiological stressor
-
Leidenheimer NJ, Schechter MD (1988) Discriminative stimulus control by the anxiogenic beta-carboline FG 7142: generalization to a physiological stressor. Pharmacol Biochem Behav 30:351-355
-
(1988)
Pharmacol Biochem Behav
, vol.30
, pp. 351-355
-
-
Leidenheimer, N.J.1
Schechter, M.D.2
-
12
-
-
0025960045
-
Inverse agonist properties of the FG 7142 discriminative stimulus
-
Leidenheimer NJ, Schechter MD (1991a) Inverse agonist properties of the FG 7142 discriminative stimulus. Pharmacol Biochem Behav 38:99-104
-
(1991)
Pharmacol Biochem Behav
, vol.38
, pp. 99-104
-
-
Leidenheimer, N.J.1
Schechter, M.D.2
-
13
-
-
0026029680
-
Inverse agonist properties of the THBC discriminative stimulus: Asymmetrical generalization with FG 7142
-
Leidenheimer NJ, Schechter MD (1991b) Inverse agonist properties of the THBC discriminative stimulus: asymmetrical generalization with FG 7142. Pharmacol Biochem Behav 38:519-525
-
(1991)
Pharmacol Biochem Behav
, vol.38
, pp. 519-525
-
-
Leidenheimer, N.J.1
Schechter, M.D.2
-
14
-
-
0026706137
-
Evidence for a noradrenergic involvement in mediating the FG 7142 discriminative stimulus
-
Leidenheimer NJ, Schechter MD (1992) Evidence for a noradrenergic involvement in mediating the FG 7142 discriminative stimulus. Pharmacol Biochem Behav 43:77-83
-
(1992)
Pharmacol Biochem Behav
, vol.43
, pp. 77-83
-
-
Leidenheimer, N.J.1
Schechter, M.D.2
-
15
-
-
0027712759
-
Molecular biology of gamma-aminobutyric acid type A/benzodiazepine receptors
-
Stephens DN (ed). Springer, Berlin Heidelberg New York
-
Lüddens H (1993) Molecular biology of gamma-aminobutyric acid type A/benzodiazepine receptors. In: Stephens DN (ed) Anxiolytic β-carbolines, from molecular biology to the clinic. Springer, Berlin Heidelberg New York, pp 16-28
-
(1993)
Anxiolytic β-carbolines, from Molecular Biology to the Clinic
, pp. 16-28
-
-
Lüddens, H.1
-
16
-
-
0029043192
-
Psychopharmacology of benzodiazepines - An update
-
Malizia AL, Nutt DJ (1995) Psychopharmacology of benzodiazepines - an update. Human Psychopharmacol 10:S1-S14
-
(1995)
Human Psychopharmacol
, vol.10
-
-
Malizia, A.L.1
Nutt, D.J.2
-
17
-
-
0022006620
-
Discriminative stimulus properties of methyl 6,7-dimethoxy-4-ethyl-β-carboline-3-carboxylate (DMCM), an inverse agonist at benzodiazepine receptors
-
Nielsen EB, Jepsen SV, Nielsen M, Braestrup C (1985) Discriminative stimulus properties of methyl 6,7-dimethoxy-4-ethyl-β-carboline-3-carboxylate (DMCM), an inverse agonist at benzodiazepine receptors. Life Sci 36:15-23
-
(1985)
Life Sci
, vol.36
, pp. 15-23
-
-
Nielsen, E.B.1
Jepsen, S.V.2
Nielsen, M.3
Braestrup, C.4
-
18
-
-
0021050981
-
DMCM: A potent convulsive benzodiazepine receptor ligand
-
Petersen EN (1983) DMCM: a potent convulsive benzodiazepine receptor ligand. Eur J Pharmacol 94:117-124
-
(1983)
Eur J Pharmacol
, vol.94
, pp. 117-124
-
-
Petersen, E.N.1
-
19
-
-
0021159954
-
Proconflict effect of benzodiazepine receptor inverse agonists and other inhibitors of GABA function
-
Petersen EN, Jensen LH (1984) Proconflict effect of benzodiazepine receptor inverse agonists and other inhibitors of GABA function. Eur J Pharmacol 103:91-97
-
(1984)
Eur J Pharmacol
, vol.103
, pp. 91-97
-
-
Petersen, E.N.1
Jensen, L.H.2
-
22
-
-
0028893945
-
Drug discrimination analysis of midazolam under a three-lever procedure I. Dose-dependent differences in generalization and antagonism
-
Sannerud CA, Ator NA (1995a) Drug discrimination analysis of midazolam under a three-lever procedure I. Dose-dependent differences in generalization and antagonism. J Pharmacol Exp Ther 272:100-111
-
(1995)
J Pharmacol Exp Ther
, vol.272
, pp. 100-111
-
-
Sannerud, C.A.1
Ator, N.A.2
-
23
-
-
0028784279
-
Drug discrimination analysis of midazolam under a three-lever procedure II. Differential effects of benzodiazepine receptor agonists
-
Sannerud CA, Ator NA (1995b) Drug discrimination analysis of midazolam under a three-lever procedure II. Differential effects of benzodiazepine receptor agonists. J Pharmacol Exp Ther 275:183-193
-
(1995)
J Pharmacol Exp Ther
, vol.275
, pp. 183-193
-
-
Sannerud, C.A.1
Ator, N.A.2
-
24
-
-
4243300297
-
β-Carboline-3-carboxylic acid ethyl ester: A lead for new psychotropic drugs
-
Stephens DN (ed). Springer, Berlin Heidelberg New York
-
Schmiechen R, Seidelmann D, Huth A (1993) β-Carboline-3-carboxylic acid ethyl ester: a lead for new psychotropic drugs. In: Stephens DN (ed) Anxiolytic β-carbolines, from molecular biology to the clinic. Springer, Berlin Heidelberg New York, pp 29-49
-
(1993)
Anxiolytic β-carbolines, from Molecular Biology to the Clinic
, pp. 29-49
-
-
Schmiechen, R.1
Seidelmann, D.2
Huth, A.3
-
25
-
-
0023687683
-
β-carbolines as antagonists of the discriminative stimulus effects of diazepam in rats
-
Shannon HE, Hagen TJ, Guzman F, Cook JA (1988) β-carbolines as antagonists of the discriminative stimulus effects of diazepam in rats. J Pharmacol Exp Ther 246:275-281
-
(1988)
J Pharmacol Exp Ther
, vol.246
, pp. 275-281
-
-
Shannon, H.E.1
Hagen, T.J.2
Guzman, F.3
Cook, J.A.4
-
26
-
-
0029417325
-
A receptor inverse agonists modulate γ-aminobutyric acid via the loreclezole binding site as well as the benzodiazepine site
-
A receptor inverse agonists modulate γ-aminobutyric acid via the loreclezole binding site as well as the benzodiazepine site. Mol Pharmacol 48:965-969
-
(1995)
Mol Pharmacol
, vol.48
, pp. 965-969
-
-
Stevenson, A.1
Wingrove, P.B.2
Whiting, P.J.3
Wafford, K.A.4
-
27
-
-
0022617301
-
Discriminative and aversive properties of β-carboline-carboxylic acid ethyl ester, a benzodiazepine receptor inverse agonist, in rhesus monkeys
-
Takada K, Winger G, Cook JM, Larscheid P, Woods JH (1986) Discriminative and aversive properties of β-carboline-carboxylic acid ethyl ester, a benzodiazepine receptor inverse agonist, in rhesus monkeys. Life Sci 38:1049-1056
-
(1986)
Life Sci
, vol.38
, pp. 1049-1056
-
-
Takada, K.1
Winger, G.2
Cook, J.M.3
Larscheid, P.4
Woods, J.H.5
-
28
-
-
0018655874
-
2 and receptor differentiation: A statistical analysis of competitive antagonism
-
2 and receptor differentiation: a statistical analysis of competitive antagonism. Life Sci 25:637-654
-
(1979)
Life Sci
, vol.25
, pp. 637-654
-
-
Tallarida, R.J.1
Cowan, A.2
Adler, M.W.3
-
29
-
-
0015896090
-
Determination of pharmacological constants: Use of narcotic antagonists to characterize analgesic receptors
-
Braude MS, Harris LS, May EL, Smith JP, Villarreal JE (eds). Advances in biochemical psychopharmacology. Raven Press, New York
-
Takemori AE (1974) Determination of pharmacological constants: use of narcotic antagonists to characterize analgesic receptors. In: Braude MS, Harris LS, May EL, Smith JP, Villarreal JE (eds) Narcotic antagonists, vol 8. Advances in biochemical psychopharmacology. Raven Press, New York, pp 335-344
-
(1974)
Narcotic Antagonists
, vol.8
, pp. 335-344
-
-
Takemori, A.E.1
-
30
-
-
0030936493
-
Role of the NMDA receptor complex in DMCM-induced seizure in mice
-
Tsuda M, Suzuki T, Misawa M (1997) Role of the NMDA receptor complex in DMCM-induced seizure in mice. Neuroreport 8:603-606
-
(1997)
Neuroreport
, vol.8
, pp. 603-606
-
-
Tsuda, M.1
Suzuki, T.2
Misawa, M.3
-
31
-
-
0029786719
-
Functional characterization of human γ-aminobutyric acidA receptors containing the a4 subunit
-
Wafford KA, Thompson SA, Thomas D, Sikela J, Wilcox AS, Whiting PJ (1996) Functional characterization of human γ-aminobutyric acidA receptors containing the a4 subunit. Mol Pharmacol 50:670-678
-
(1996)
Mol Pharmacol
, vol.50
, pp. 670-678
-
-
Wafford, K.A.1
Thompson, S.A.2
Thomas, D.3
Sikela, J.4
Wilcox, A.S.5
Whiting, P.J.6
-
33
-
-
0026769789
-
Discriminative stimulus effects of morphine: Effects of training dose on agonist and antagonist effects of mu opioids
-
Young AM, Masaki MA, Geula C (1992) Discriminative stimulus effects of morphine: effects of training dose on agonist and antagonist effects of mu opioids. J Pharmacol Exp Ther 261: 246-257
-
(1992)
J Pharmacol Exp Ther
, vol.261
, pp. 246-257
-
-
Young, A.M.1
Masaki, M.A.2
Geula, C.3
|