Pharmacological characterization of a GluR6 kainate receptor in cultured hippocampal neurons

European Journal of Pharmacology

Volumn 378, Issue 3, 1999, Pages 331-337

  Bleakman, David ^a   Ogden, Ann Marie ^a   Ornstein, Paul L ^a   Hoo, Ken ^b  

^a ELI LILLY AND COMPANY   (United States)

^b NPS Pharmaceutical Inc   (United States)

Author keywords

(RS) 2 amino 3 (3 hydroxy 5 tert butyl 4 isoxazolyl) propionic acid (ATPA); GluR5 antagonist; Quinoxalinedione

Indexed keywords

1 (4 AMINOPHENYL) 3,4 DIHYDRO 4 METHYL 3 METHYLCARBAMOYL 7,8 METHYLENEDIOXY 5H 2,3 BENZODIAZEPINE; 2 AMINO 3 (3 HYDROXY 5 TERT BUTYL 4 ISOOXAZOLYL) PROPIONIC ACID; 4 [3 (2 NAPHTHYL)ALLYL]GLUTAMIC ACID; 6 (4 CARBOXYBENZYL) 1,2,3,4,4A,5,6,7,8,8A DECAHYDRO 3 ISOQUINOLINECARBOXYLIC ACID; AMPA RECEPTOR; AMPA RECEPTOR ANTAGONIST; BENZODIAZEPINE DERIVATIVE; DECAHYDRO 6 [2 (1H TETRAZOL 5 YL)ETHYL] 3 ISOQUINOLINECARBOXYLIC ACID; DIZOCILPINE; GLUTAMATE RECEPTOR; ION CHANNEL; KAINIC ACID RECEPTOR; QUINOXALINE DERIVATIVE; UNCLASSIFIED DRUG;

ANIMAL EXPERIMENT; ANIMAL TISSUE; ARTICLE; BRAIN DEVELOPMENT; ELECTROPHYSIOLOGY; HIPPOCAMPUS; LIGAND BINDING; MEMBRANE CURRENT; NEWBORN; NONHUMAN; PRIORITY JOURNAL; RAT;

ALPHA-AMINO-3-HYDROXY-5-METHYL-4-ISOXAZOLEPROPIONIC ACID; ANIMALS; BINDING, COMPETITIVE; CELL LINE; DOSE-RESPONSE RELATIONSHIP, DRUG; EXCITATORY AMINO ACID AGONISTS; EXCITATORY AMINO ACID ANTAGONISTS; GENE EXPRESSION; GLUTAMATES; HIPPOCAMPUS; HUMANS; ISOQUINOLINES; KAINIC ACID; MEMBRANE POTENTIALS; NEURONS; PATCH-CLAMP TECHNIQUES; QUINOXALINES; RADIOLIGAND ASSAY; RECEPTORS, AMPA; RECEPTORS, KAINIC ACID; RECOMBINANT FUSION PROTEINS; TETRAZOLES;

EID: 0032801717     PISSN: 00142999     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0014-2999(99)00478-1     Document Type: Article

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