Cross-resistance with dieldrin of a novel tricyclic dinitrile GABA receptor antagonist

British Journal of Pharmacology

Volumn 127, Issue 6, 1999, Pages 1305-1307

  Matsuda, Kazuhiko ^b   Hosie, Alastair M ^a   Holyoke Jr , Caleb W ^c   Rauh, James J ^c   Sattelle, David B ^a  

^a UNIVERSITY OF CAMBRIDGE   (United Kingdom)

^b KINKI UNIVERSITY   (Japan)

^c DUPONT COMPANY   (United States)

Author keywords

Drosophila melanogaster; GABA gated Cl channel; KN244 (a tricyclic dinitrile); RDL (resistant to dieldrin) subunit

Indexed keywords

4 AMINOBUTYRIC ACID; 4 AMINOBUTYRIC ACID RECEPTOR BLOCKING AGENT; 4,4 BIS(TRIFLUOROMETHYL)TRICYCLO[4,2,1,0 2,5]NON 7 ENE 3,3 DICARBONITRILE; CHLORIDE CHANNEL; DIELDRIN; UNCLASSIFIED DRUG;

ANIMAL CELL; ARTICLE; CONTROLLED STUDY; CROSS RESISTANCE; DROSOPHILA MELANOGASTER; NONHUMAN; OOCYTE; PRIORITY JOURNAL; XENOPUS;

ANIMALS; BICYCLO COMPOUNDS; CHLORIDE CHANNELS; DIELDRIN; DOSE-RESPONSE RELATIONSHIP, DRUG; DROSOPHILA MELANOGASTER; GABA ANTAGONISTS; GAMMA-AMINOBUTYRIC ACID; INSECTICIDE RESISTANCE; INSECTICIDES; MEMBRANE POTENTIALS; NITRILES; OOCYTES; RECEPTORS, GABA; XENOPUS;

EID: 0032794352     PISSN: 00071188     EISSN: None     Source Type: Journal    
DOI: 10.1038/sj.bjp.0702663     Document Type: Article

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