메뉴 건너뛰기




Volumn 51, Issue 4-5, 1999, Pages 363-368

Stability and perfusion studies of desmopressin (dDAVP) and prodrugs in the rat jejunum

Author keywords

DDAVP; Desmopressin; Prodrugs; Rat perfusion; Stability; Vasopressin analogue

Indexed keywords

DESMOPRESSIN; ESTERASE; PRODRUG;

EID: 0032765844     PISSN: 09402993     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0940-2993(99)80023-2     Document Type: Conference Paper
Times cited : (3)

References (17)
  • 1
    • 0343193275 scopus 로고
    • Serum esterases (1). Two types of esterases (A and B) hydrolysing p-nitrophenylacetate, proprionate and buryrate, and a method of their determination
    • ALDRIDGE WN: Serum esterases (1). Two types of esterases (A and B) hydrolysing p-nitrophenylacetate, proprionate and buryrate, and a method of their determination. Biochemical Journal 1953; 53: 110-117.
    • (1953) Biochemical Journal , vol.53 , pp. 110-117
    • Aldridge, W.N.1
  • 2
    • 0032507740 scopus 로고    scopus 로고
    • Drug absorption of prodrug esters using the Caco-2 model: Evaluation of ester hydrolysis and transepithelial transport
    • AUGUSTIJNS P, ANNAERT P, HEYLEN P, et al.: Drug absorption of prodrug esters using the Caco-2 model: evaluation of ester hydrolysis and transepithelial transport. Int J Pharm Sci 1998; 166: 45-53.
    • (1998) Int J Pharm Sci , vol.166 , pp. 45-53
    • Augustijns, P.1    Annaert, P.2    Heylen, P.3
  • 3
    • 0026500650 scopus 로고
    • Means to enhance penetration. Prodrugs as a means to improve the delivery of peptide drugs
    • BUNDGAARD H: Means to enhance penetration. Prodrugs as a means to improve the delivery of peptide drugs. Adv Drug Del Rev 1992; 8: 1-38.
    • (1992) Adv Drug Del Rev , vol.8 , pp. 1-38
    • Bundgaard, H.1
  • 4
    • 0029855969 scopus 로고    scopus 로고
    • Comparison between permeability coefficients in rat and human jejunum
    • FAGERHOLM U, JOHANSSON M, LENNERNÄS H: Comparison between permeability coefficients in rat and human jejunum. Pharm Res 1996; 13: 1336-1342.
    • (1996) Pharm Res , vol.13 , pp. 1336-1342
    • Fagerholm, U.1    Johansson, M.2    Lennernäs, H.3
  • 5
    • 0027396128 scopus 로고
    • Pharmacokinetics of 1-deamino-8-D-arginine vasopressin after various routes of administration in healthy volunteers
    • FJELLESTAD-PAULSEN A, HÖGLUND P, LUNDIN S, et al.: Pharmacokinetics of 1-deamino-8-D-arginine vasopressin after various routes of administration in healthy volunteers. Clin Endocrinol 1993; 38: 177-182.
    • (1993) Clin Endocrinol , vol.38 , pp. 177-182
    • Fjellestad-Paulsen, A.1    Höglund, P.2    Lundin, S.3
  • 6
    • 0031126947 scopus 로고    scopus 로고
    • Prodrug strategies to enhance the intestinal absorption of peptides
    • GANGWAR S, PAULETTI GM, WANG B, et al.: Prodrug strategies to enhance the intestinal absorption of peptides. Drug Disc Today 1997; 2: 148-155.
    • (1997) Drug Disc Today , vol.2 , pp. 148-155
    • Gangwar, S.1    Pauletti, G.M.2    Wang, B.3
  • 7
    • 0027472110 scopus 로고
    • Prodrugs of peptides. 18. Synthesis and evaluation of various esters of desmopressin (dDAVP)
    • KAHNS AH, BUUR A, BUNDGAARD H: Prodrugs of peptides. 18. Synthesis and evaluation of various esters of Desmopressin (dDAVP). Pharm Res 1993; 10: 68-74.
    • (1993) Pharm Res , vol.10 , pp. 68-74
    • Kahns, A.H.1    Buur, A.2    Bundgaard, H.3
  • 8
    • 0029063811 scopus 로고
    • Glycosylated peptide hormones: Pharmacological properties and conformational studies of analogues of [1-Desamino, 8-D-arginine]-vasopressin
    • KIHLBERG J, AHMAN J, WALSE B, et al.: Glycosylated peptide hormones: Pharmacological properties and conformational studies of analogues of [1-Desamino, 8-D-arginine]-vasopressin. J Med Chem 1995; 38: 161-169.
    • (1995) J Med Chem , vol.38 , pp. 161-169
    • Kihlberg, J.1    Ahman, J.2    Walse, B.3
  • 9
    • 0031422606 scopus 로고    scopus 로고
    • Rat jejunal permeability and metabolism of μ-selective tetrapeptides in gastrointestinal fluids from humans and rats
    • KRONDAHL E, ORZECHOVSKI A, EKSTROM G, et al.: Rat jejunal permeability and metabolism of μ-selective tetrapeptides in gastrointestinal fluids from humans and rats. Pharm Res 1997; 12: 1780-1785.
    • (1997) Pharm Res , vol.12 , pp. 1780-1785
    • Krondahl, E.1    Orzechovski, A.2    Ekstrom, G.3
  • 10
    • 0030818767 scopus 로고    scopus 로고
    • Enhancing effects of monohexanoin and two other medium-chain glyceride vehicles on intestinal absorption of Desmopressin (dDAVP)
    • LUNDIN PDP, BOJRUP M, LJUSBERG-WAHREN H, et al.: Enhancing effects of monohexanoin and two other medium-chain glyceride vehicles on intestinal absorption of Desmopressin (dDAVP). J Pharmacol Exp Thera 1997; 282: 585-590.
    • (1997) J Pharmacol Exp Thera , vol.282 , pp. 585-590
    • Lundin, P.D.P.1    Bojrup, M.2    Ljusberg-Wahren, H.3
  • 11
    • 0025224640 scopus 로고
    • Absorption of a vasopressin analogue, 1-deamino-8-D-arginine (dDAVP) in a human intestinal epithelial cell line, Caco-2
    • LUNDIN S, ARTHURSSON P: Absorption of a vasopressin analogue, 1-deamino-8-D-arginine (dDAVP) in a human intestinal epithelial cell line, Caco-2. Int J Pharm 1990; 64: 181-186.
    • (1990) Int J Pharm , vol.64 , pp. 181-186
    • Lundin, S.1    Arthursson, P.2
  • 13
    • 0023223086 scopus 로고
    • Prodrugs as drug delivery systems.68. Chemical and plasma catalyzed hydrolysis of various esters of benzoic acid: A reference system for designing prodrug esters of carboxylic acid agents
    • NIELSEN NM, BUNDGAARD H: Prodrugs as drug delivery systems.68. Chemical and plasma catalyzed hydrolysis of various esters of benzoic acid: a reference system for designing prodrug esters of carboxylic acid agents. Int J Pharm Sci 1987; 39: 75-85.
    • (1987) Int J Pharm Sci , vol.39 , pp. 75-85
    • Nielsen, N.M.1    Bundgaard, H.2
  • 14
    • 0343026460 scopus 로고    scopus 로고
    • Prodrugs of peptides and peptidomimetics for improved formulation and delivery
    • OLIYAI R: Prodrugs of peptides and peptidomimetics for improved formulation and delivery. Adv Drug Del Rev 1996; 19: 275-286.
    • (1996) Adv Drug Del Rev , vol.19 , pp. 275-286
    • Oliyai, R.1
  • 15
    • 0027406209 scopus 로고
    • Prodrugs of peptides and proteins for improved formulation and delivery
    • OLIYAI R, STELLA VJ: Prodrugs of peptides and proteins for improved formulation and delivery. Ann Rev Pharmacol Toxicol 1993; 32: 521-544.
    • (1993) Ann Rev Pharmacol Toxicol , vol.32 , pp. 521-544
    • Oliyai, R.1    Stella, V.J.2
  • 16
    • 0025066218 scopus 로고
    • Basic pharmacology of desmopressin. A review
    • VILHARDT H: Basic pharmacology of Desmopressin. A review. Drug Invest 1990; 2: 2-8.
    • (1990) Drug Invest , vol.2 , pp. 2-8
    • Vilhardt, H.1
  • 17
    • 0022877317 scopus 로고
    • Biological effect and plasma concentrations of dDAVP after intranasal and peroral administration to humans
    • VILHARDT H, LUNDIN S: Biological effect and plasma concentrations of dDAVP after intranasal and peroral administration to humans. Gen Pharmacol 1986; 17: 481-483.
    • (1986) Gen Pharmacol , vol.17 , pp. 481-483
    • Vilhardt, H.1    Lundin, S.2


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.