메뉴 건너뛰기




Volumn 58, Issue 4, 1999, Pages 675-680

Exemestane

Author keywords

[No Author keywords available]

Indexed keywords

AROMATASE; ESTRADIOL; ESTRONE; ESTRONE SULFATE; EXEMESTANE; FORMESTANE; MEGESTROL; TAMOXIFEN;

EID: 0032757904     PISSN: 00126667     EISSN: None     Source Type: Journal    
DOI: 10.2165/00003495-199958040-00007     Document Type: Review
Times cited : (27)

References (24)
  • 2
    • 0025648483 scopus 로고
    • 4-Aminoandrostenedione derivatives: A novel class of irreversible aromatase inhibitors. Comparison with FCE-24304 and 4-hydroxyandrostenedione
    • Nov 20
    • 2. di-Salle E, Giudici D. Ornati G, et al. 4-Aminoandrostenedione derivatives: a novel class of irreversible aromatase inhibitors. Comparison with FCE-24304 and 4-hydroxyandrostenedione, J Steroid Biochem Mol Biol 1990 Nov 20; 37: 369-74
    • (1990) J Steroid Biochem Mol Biol , vol.37 , pp. 369-374
    • Di-Salle, E.1    Giudici, D.2    Ornati, G.3
  • 3
    • 0023751351 scopus 로고
    • 6-Methylenandrosta-1,4-diene-3,17-dione (FCE 24304): A new irreversible aromatase inhibitor
    • 3. Giudici D, Ornati G, Briatico G, et al. 6-Methylenandrosta-1,4-diene-3,17-dione (FCE 24304): a new irreversible aromatase inhibitor. J Steroid Biochem 1988; 30: 391-4
    • (1988) J Steroid Biochem , vol.30 , pp. 391-394
    • Giudici, D.1    Ornati, G.2    Briatico, G.3
  • 5
    • 0024351630 scopus 로고
    • Effect of the irreversible aromatase FCE 24304 on DMBA-induced mammary tumors in ovariectomized rats treated with testosterone
    • 5. Zaccheo T, di-Salle E. Effect of the irreversible aromatase FCE 24304 on DMBA-induced mammary tumors in ovariectomized rats treated with testosterone. Cancer Chemother Pharmacol 1989: 25: 95-8
    • (1989) Cancer Chemother Pharmacol , vol.25 , pp. 95-98
    • Zaccheo, T.1    Di-Salle, E.2
  • 6
    • 0026446844 scopus 로고
    • Phase I and endocrine study of exemestane (FCE 24304), a new aromatase inhibitor, in postmenopausal women
    • 6. Evans TR, di-Salle E, Ornati G, et al. Phase I and endocrine study of exemestane (FCE 24304), a new aromatase inhibitor, in postmenopausal women. Cancer Res 1992; 52: 5933-9
    • (1992) Cancer Res , vol.52 , pp. 5933-5939
    • Evans, T.R.1    Di-Salle, E.2    Ornati, G.3
  • 7
    • 0031663593 scopus 로고    scopus 로고
    • In vivo inhibition of aromatization by exemestane, a novel irreversible aromatase inhibitor, in postmenopausal breast cancer patients
    • Sep
    • 7. Geisler J, King N, Anker G. et al. In vivo inhibition of aromatization by exemestane, a novel irreversible aromatase inhibitor, in postmenopausal breast cancer patients. Clin Cancer Res 1998 Sep; 4: 2089-93
    • (1998) Clin Cancer Res , vol.4 , pp. 2089-2093
    • Geisler, J.1    King, N.2    Anker, G.3
  • 8
    • 0030748661 scopus 로고    scopus 로고
    • Endocrine and clinical effects of exemestane (PNU 155971), a novel steroidal aromatase inhibitor, in postmenopausal breast cancer patients: A phase I study
    • Jul
    • 8. Johannessen DC, Engan T, di-Salle E, et al. Endocrine and clinical effects of exemestane (PNU 155971), a novel steroidal aromatase inhibitor, in postmenopausal breast cancer patients: a phase I study. Clin Cancer Res 1997 Jul; 3: 1101-8
    • (1997) Clin Cancer Res , vol.3 , pp. 1101-1108
    • Johannessen, D.C.1    Engan, T.2    Di-Salle, E.3
  • 9
    • 15444348553 scopus 로고    scopus 로고
    • Safety, activity and estrogen inhibition by exemestane in postmenopausal women with advanced breast cancer: A phase I study
    • Sep
    • 9. Paridaens R, Thomas J, Wildiers J, et al. Safety, activity and estrogen inhibition by exemestane in postmenopausal women with advanced breast cancer: a phase I study. Anticancer Drugs 1998 Sep; 9: 675-83
    • (1998) Anticancer Drugs , vol.9 , pp. 675-683
    • Paridaens, R.1    Thomas, J.2    Wildiers, J.3
  • 10
    • 0002339213 scopus 로고
    • Excretion balance and absorption of 14C-exemestane in animals and humans
    • abstract no. 73
    • 10. Castelli MG, Cocchiara G, Zurlo MG, et al. Excretion balance and absorption of 14C-exemestane in animals and humans [abstract no. 73]. J Endocrinol Invest 1994; 17 (3 Suppl. I): 76
    • (1994) J Endocrinol Invest , vol.17 , Issue.3 SUPPL. I , pp. 76
    • Castelli, M.G.1    Cocchiara, G.2    Zurlo, M.G.3
  • 11
    • 0009518209 scopus 로고
    • Relative bioavailability and pharmacokinetics of two different formulations of exemestane, a new aromatase inhibitor
    • abstract no. 76
    • 11. Poggesi I, Allievi C, Strolin Benedetti M, et al. Relative bioavailability and pharmacokinetics of two different formulations of exemestane, a new aromatase inhibitor [abstract no. 76]. J Endocrinol Invest 1994; 17 (3 Suppl. I): 79
    • (1994) J Endocrinol Invest , vol.17 , Issue.3 SUPPL. I , pp. 79
    • Poggesi, I.1    Allievi, C.2    Strolin Benedetti, M.3
  • 12
    • 4243233187 scopus 로고
    • Pharmacokinetics of repeated low-doses of exemestane (1, 2.5, 5 and 10mg) in postmenopausal healthy volunteers
    • abstract no. 952
    • 12. Persiani S, Poggesi I, Cicioni P, et al. Pharmacokinetics of repeated low-doses of exemestane (1, 2.5, 5 and 10mg) in postmenopausal healthy volunteers. [abstract no. 952]. Eur J Cancer 1995; 31 Suppl. 5: s198
    • (1995) Eur J Cancer , Issue.SUPPL. 5
    • Persiani, S.1    Poggesi, I.2    Cicioni, P.3
  • 13
    • 0003213592 scopus 로고    scopus 로고
    • Effect of food and formulation on the pharmacokinetics (PK) and pharmacodynamics (PD) of a single oral dose ol exemestane (Aromasin™, EXE)
    • abstract no. 741
    • 13. Poggesi I, Jannuzzo MG, di-Salle E, et al. Effect of food and formulation on the pharmacokinetics (PK) and pharmacodynamics (PD) of a single oral dose ol exemestane (Aromasin™, EXE) [abstract no. 741]. Proc Am Soc Clin Oncol 1999; 18: 193a
    • (1999) Proc Am Soc Clin Oncol , vol.18
    • Poggesi, I.1    Jannuzzo, M.G.2    Di-Salle, E.3
  • 14
    • 0002786764 scopus 로고
    • Urinary metabolism of exemestane, a new aromatase inhibitor, in rat, dog, monkey and human volunteers
    • abstract no. 75
    • 14. Cocchiara G, Allievi C, Berardi A, et al. Urinary metabolism of exemestane, a new aromatase inhibitor, in rat, dog, monkey and human volunteers [abstract no. 75]. J Endocrinol Invest 1994; 17 (3 Suppl. I): 78
    • (1994) J Endocrinol Invest , vol.17 , Issue.3 SUPPL. I , pp. 78
    • Cocchiara, G.1    Allievi, C.2    Berardi, A.3
  • 15
    • 0345596372 scopus 로고    scopus 로고
    • Third-line hormonal treatment with exemestane in postmenopausal patients with advanced breast cancer progressing on aminoglutethimide: A phase II multicentre multinational study
    • Oct
    • 15. Thürlimann B, Paridaens R, Serin D, et al. Third-line hormonal treatment with exemestane in postmenopausal patients with advanced breast cancer progressing on aminoglutethimide: a phase II multicentre multinational study. Eur J Cancer A 1997 Oct; 33: 1767-73
    • (1997) Eur J Cancer A , vol.33 , pp. 1767-1773
    • Thürlimann, B.1    Paridaens, R.2    Serin, D.3
  • 16
    • 0000340799 scopus 로고    scopus 로고
    • A phase II confirmatory study of antitumour efficacy and safety of exemestane as third-line hormonal treatment of postmenopausal patients with metastatic breast cancer refractory to tamoxifen and megace™
    • abstract no. 439
    • 16. Jones S, Chang A, Lusch C, et al. A phase II confirmatory study of antitumour efficacy and safety of exemestane as third-line hormonal treatment of postmenopausal patients with metastatic breast cancer refractory to tamoxifen and megace™ [abstract no. 439]. Breast Cancer Res Treat 1998; 50 (3): 305
    • (1998) Breast Cancer Res Treat , vol.50 , Issue.3 , pp. 305
    • Jones, S.1    Chang, A.2    Lusch, C.3
  • 17
    • 0000736263 scopus 로고    scopus 로고
    • A phase II study of exemestane in metastatic breast cancer patients failing nonsteroidal aromatase inhibitors
    • abstract no. 435
    • 17. Lonning PE, Bajetta E, Murray R, et al. A phase II study of exemestane in metastatic breast cancer patients failing nonsteroidal aromatase inhibitors [abstract no. 435]. Breast Cancer Res Treat 1998; 50 (3): 304
    • (1998) Breast Cancer Res Treat , vol.50 , Issue.3 , pp. 304
    • Lonning, P.E.1    Bajetta, E.2    Murray, R.3
  • 18
    • 0002649677 scopus 로고    scopus 로고
    • A phase II study of antitumor efficacy and safety of exemestane as third-line hormonal treatment of postmenopausal patients with metastatic breast cancer refractory to tamoxifen and Megace™
    • abstract no. 64p
    • 18. Jones S, Vogel C, Fehrenbacher L, et al. A phase II study of antitumor efficacy and safety of exemestane as third-line hormonal treatment of postmenopausal patients with metastatic breast cancer refractory to tamoxifen and Megace™ [abstract no. 64p]. Ann Oncol 1998; 9 Suppl. 4: 13
    • (1998) Ann Oncol , vol.9 , Issue.SUPPL. 4 , pp. 13
    • Jones, S.1    Vogel, C.2    Fehrenbacher, L.3
  • 19
    • 0001986053 scopus 로고    scopus 로고
    • Activity of exemestane, an irreversible, oral, aromatase inhibitor in metastatic postmenopausal breast cancer patients failing tamoxifen
    • abstract no. 408 Sep
    • 19. Kvinnsland S, Anker G, Dirix LY, et al. Activity of exemestane, an irreversible, oral, aromatase inhibitor in metastatic postmenopausal breast cancer patients failing tamoxifen [abstract no. 408]. Eur J Cancer 1998 Sep; 34 Suppl. 5: s91
    • (1998) Eur J Cancer , vol.34 , Issue.SUPPL. 5
    • Kvinnsland, S.1    Anker, G.2    Dirix, L.Y.3
  • 20
    • 0000340799 scopus 로고    scopus 로고
    • A phase II study of antitumour efficacy and safety of exemestane as a second-line hormonal treatment of postmenopausal patients with metastatic breast cancer refractory to tamoxifen
    • Dec 12-15; San Antonio, Texas
    • 20. Jones S, Belt R, Cooper B, et al. A phase II study of antitumour efficacy and safety of exemestane as a second-line hormonal treatment of postmenopausal patients with metastatic breast cancer refractory to tamoxifen [abstract]. 21st Breast Cancer Symposium; 1998 Dec 12-15; San Antonio, Texas
    • (1998) 21st Breast Cancer Symposium
    • Jones, S.1    Belt, R.2    Cooper, B.3
  • 21
    • 0000628683 scopus 로고    scopus 로고
    • Survival advantage of exemestane EXE, Aromasin® over megestrol acetate in postmenopausal women with advanced breast cancer refractory to tamoxifen: Results of a phase III randomised double-blind study
    • abstract no. 412
    • 21. Kaufmann M, Bajetta E, Dirix LY, et al. Survival advantage of exemestane (EXE, Aromasin® over megestrol acetate in postmenopausal women with advanced breast cancer refractory to tamoxifen: results of a phase III randomised double-blind study [abstract no. 412]. Proc Am Soc Clin Oncol 1999; 18: 109a
    • (1999) Proc Am Soc Clin Oncol , vol.18
    • Kaufmann, M.1    Bajetta, E.2    Dirix, L.Y.3
  • 22
    • 4243881832 scopus 로고    scopus 로고
    • Aromasin™ versus Megace™: Improved outcomes
    • Jun Milan
    • 22. Kaufmann M, Aromasin™ versus Megace™: improved outcomes [abstract]. In: Proceedings of 1st Milan Breast Cancer Conference; 1999 Jun 16; Milan: 6-7
    • (1999) Proceedings of 1st Milan Breast Cancer Conference , vol.16 , pp. 6-7
    • Kaufmann, M.1
  • 23
    • 0009485589 scopus 로고    scopus 로고
    • Hormonal therapy in breast cancer and predominant visceral disease: Effectiveness of the new oral aromatase inactivator, Aromasin™ (Exemestane), in advanced breast cancer patients having progressed on antiestrogens
    • Sep 12-16: Vienna
    • 23. Tedeschi M, Kvinnsland S, Jones SE, et al. Hormonal therapy in breast cancer and predominant visceral disease: effectiveness of the new oral aromatase inactivator, Aromasin™ (Exemestane), in advanced breast cancer patients having progressed on antiestrogens [abstract]. In: Proceedings of European Cancer Conference: 1999 Sep 12-16: Vienna
    • (1999) Proceedings of European Cancer Conference
    • Tedeschi, M.1    Kvinnsland, S.2    Jones, S.E.3


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.