Stereoselective reduction via lithium borotritide: Synthesis of 3H-labeled 2-hydroxy-N-[(5-hydroxy-[5-3H]-1,3,3-trimethylcyclohexyl)methyl]-5 -methylbenzamide

Journal of Labelled Compounds and Radiopharmaceuticals

Volumn 42, Issue 11, 1999, Pages 1061-1068

  Dischino, Douglas D ^a   Meanwell, Nicholas A ^a   Morimoto, Hiromi ^b   Pearce, Bradley C ^a   Than, Chit ^b   Torri, Albert F ^a   Williams, Philip G ^b   Yu, Kuo Long ^a  

^a BRISTOL MYERS SQUIBB   (United States)

^b LAWRENCE BERKELEY NATIONAL LABORATORY   (United States)

Author keywords

Influenza; LiBT4; Stereoselective reduction

Indexed keywords

LITHIUM; LITHIUM COMPOUNDS; REDUCTION; STEREOSELECTIVITY;

CYCLOHEXYL; HIGH SPECIFIC ACTIVITIES; INFLUENZA; LIBT4; METHYLBENZAMIDE; NORMAL PHASE HPLC; STEREO-SELECTIVE; STEREOSELECTIVE REDUCTION; TRIMETHYL;

KETONES;

2 HYDROXY N [(5 HYDROXY 1,3,3 TRIMETHYLCYCLOHEXYL)METHY] 5 METHYLBENZAMIDE H 3; ALCOHOL; BENZAMIDE DERIVATIVE; KETONE; LITHIUM BOROTRITIDE; LITHIUM DERIVATIVE; UNCLASSIFIED DRUG;

ARTICLE; HIGH PERFORMANCE LIQUID CHROMATOGRAPHY; PURIFICATION; STEREOCHEMISTRY; SYNTHESIS;

EID: 0032754753     PISSN: 03624803     EISSN: None     Source Type: Journal    
DOI: 10.1002/(SICI)1099-1344(199911)42:11<1061::AID-JLCR261>3.0.CO;2-N     Document Type: Article

References (8)

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