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Volumn 128, Issue 3, 1999, Pages 760-766

Direct block of native and cloned (Kir2.1) inward rectifier K+ channels by chloroethylclonidine

Author keywords

CEC; Chloroethylclonidine; Imidazolidine; Imidazoline; Inward rectifier; IRK1; Kir; Polyamine; Potassium channel; Skeletal muscle

Indexed keywords

ADRENALIN; ASPARAGINE; ASPARTIC ACID; CHLOROETHYLCLONIDINE; CLONIDINE; NORADRENALIN; POTASSIUM CHANNEL; POTASSIUM ION; PRAZOSIN; RAUWOLSCINE;

EID: 0032744920     PISSN: 00071188     EISSN: None     Source Type: Journal    
DOI: 10.1038/sj.bjp.0702819     Document Type: Article
Times cited : (31)

References (28)
  • 3
    • 0022361070 scopus 로고
    • The isolated stomach preparation of the mouse: A physiological unit for pharmacological analysis
    • BLACK, J.W. & SHANKLEY, N.P. (1985). The isolated stomach preparation of the mouse: a physiological unit for pharmacological analysis. Br. J. Pharmacol., 86, 571-579.
    • (1985) Br. J. Pharmacol. , vol.86 , pp. 571-579
    • Black, J.W.1    Shankley, N.P.2
  • 7
    • 0027317417 scopus 로고
    • Human alpha(2)-adrenergic receptor subtype distribution - Widespread and subtype-selective expression of alpha(2) C10, alpha(2) C4, and alpha(2) C2 messenger-RNA in multiple tissues
    • EASON, M.G. & LIGGETT, S.B. (1993). Human alpha(2)-adrenergic receptor subtype distribution - widespread and subtype-selective expression of alpha(2) C10, alpha(2) C4, and alpha(2) C2 messenger-RNA in multiple tissues. Mol. Pharmacol., 44, 70-75.
    • (1993) Mol. Pharmacol. , vol.44 , pp. 70-75
    • Eason, M.G.1    Liggett, S.B.2
  • 10
    • 0029614872 scopus 로고
    • Chloroethylclonidine increases the incidence of lethal arrhythmias during coronary occlusion in anesthetized dogs
    • GELLER, J.C., CUA, M., PRIETO, L., GUO, S.D., DANILO JR, P. & ROSEN, M.R. (1995). Chloroethylclonidine increases the incidence of lethal arrhythmias during coronary occlusion in anesthetized dogs. E. J. Pharmacol., 294, 423-428.
    • (1995) E. J. Pharmacol. , vol.294 , pp. 423-428
    • Geller, J.C.1    Cua, M.2    Prieto, L.3    Guo, S.D.4    Danilo P., Jr.5    Rosen, M.R.6
  • 12
    • 0001390390 scopus 로고
    • Les constantes electriques de la membrane du muscle
    • KATZ, B. (1949). Les constantes electriques de la membrane du muscle. Archives des science physiologiques, 3, 285-299.
    • (1949) Archives des Science Physiologiques , vol.3 , pp. 285-299
    • Katz, B.1
  • 13
    • 0025816211 scopus 로고
    • Direct prediction of dissociation constants (pKa's) of clonidine-like imidazolines, 2-substituted imidazoles, and 1-methyl-2-substituted-imidazoles from 3D structures using a comparative molecular field analysis (CoMFA) approach
    • KIM, K.H. & MARTIN, Y.C. (1991). Direct prediction of dissociation constants (pKa's) of clonidine-like imidazolines, 2-substituted imidazoles, and 1-methyl-2-substituted-imidazoles from 3D structures using a comparative molecular field analysis (CoMFA) approach. J. Med. Chem., 34, 2056-2060.
    • (1991) J. Med. Chem. , vol.34 , pp. 2056-2060
    • Kim, K.H.1    Martin, Y.C.2
  • 14
    • 0019393868 scopus 로고
    • Inward rectification in frog skeletal muscle fibres and its dependence on membrane potential and external potassium
    • LEECH, C.A. & STANFIELD, P.R. (1981). Inward rectification in frog skeletal muscle fibres and its dependence on membrane potential and external potassium. J. Physiol., 319, 295-309.
    • (1981) J. Physiol. , vol.319 , pp. 295-309
    • Leech, C.A.1    Stanfield, P.R.2
  • 15
    • 0027984375 scopus 로고
    • Potassium channel block by cytoplasmic polyamines as the mechanism of intrinsic rectification
    • LOPATIN, A.N., MAKHINA, E.N. & NICHOLS, C.G. (1994). Potassium channel block by cytoplasmic polyamines as the mechanism of intrinsic rectification. Nature, 372, 366-369.
    • (1994) Nature , vol.372 , pp. 366-369
    • Lopatin, A.N.1    Makhina, E.N.2    Nichols, C.G.3
  • 16
    • 0028004411 scopus 로고
    • Interactions of chloroethylclonidine with rauwolscine-and prazosin-sensitive adrenoceptors in dog saphenous vein
    • LOW, A.M., BOWDISH, T.R., PRASHAD, T.R. & GASPAR, V. (1994). Interactions of chloroethylclonidine with rauwolscine-and prazosin-sensitive adrenoceptors in dog saphenous vein. Br. J. Pharmacol., 113, 1263-1268.
    • (1994) Br. J. Pharmacol. , vol.113 , pp. 1263-1268
    • Low, A.M.1    Bowdish, T.R.2    Prashad, T.R.3    Gaspar, V.4
  • 18
    • 0025085847 scopus 로고
    • Autoradiographic delineation of skeletal-muscle alpha-1-adrenergic receptor distribution
    • MARTIN, W.H., TOLLEY, T.K. & SAFFITZ, J.E. (1990). Autoradiographic delineation of skeletal-muscle alpha-1-adrenergic receptor distribution. Am. J. Physiol., 259, H1402-H1408.
    • (1990) Am. J. Physiol. , vol.259
    • Martin, W.H.1    Tolley, T.K.2    Saffitz, J.E.3
  • 20
    • 0027220063 scopus 로고
    • A sarcolemmal vesicle preparation from rat isolated skeletal muscle suitable for patch-clamp experiments
    • McKILLEN, H.-C. (1993). A sarcolemmal vesicle preparation from rat isolated skeletal muscle suitable for patch-clamp experiments. J. Physiol., 467, p. 242Pp
    • (1993) J. Physiol. , vol.467
    • McKillen, H.-C.1
  • 21
    • 0017169696 scopus 로고
    • Clonidine and related analogues. Quantitative correlations
    • ROUOT, B., LECLERC, G. & WERMUTH, C.G. (1976). Clonidine and related analogues. Quantitative correlations. J. Med. Chem., 19, 1049-1054.
    • (1976) J. Med. Chem. , vol.19 , pp. 1049-1054
    • Rouot, B.1    Leclerc, G.2    Wermuth, C.G.3
  • 22
    • 4243881813 scopus 로고    scopus 로고
    • Block of cardiac inward rectifier potassium current by chloroethylclonidine
    • STADNICKA, A., KWOK, W.M., REHMERT, G.C. & BOSNJAK, Z.J. (1997). Block of cardiac inward rectifier potassium current by chloroethylclonidine. Biophys. J., 72, A251.
    • (1997) Biophys. J. , vol.72
    • Stadnicka, A.1    Kwok, W.M.2    Rehmert, G.C.3    Bosnjak, Z.J.4
  • 24
    • 0018073033 scopus 로고
    • Dissociation constants of clonidine and structurally related imidazolidines
    • TIMMERMANS, P.B. & VAN ZWIETEN, P.A. (1978). Dissociation constants of clonidine and structurally related imidazolidines. Arzneimittel-Forschung., 28, 1676-1681.
    • (1978) Arzneimittel-Forschung. , vol.28 , pp. 1676-1681
    • Timmermans, P.B.1    Van Zwieten, P.A.2
  • 25
    • 0030660324 scopus 로고    scopus 로고
    • Chloroethylclonidine and alpha-adrenoceptor agonist interaction in blood vessels following heart failure
    • TRAN, Y.L. & FORSTER, C. (1997). Chloroethylclonidine and alpha-adrenoceptor agonist interaction in blood vessels following heart failure. Eur. J. Pharmacol., 336, 177-185.
    • (1997) Eur. J. Pharmacol. , vol.336 , pp. 177-185
    • Tran, Y.L.1    Forster, C.2
  • 26
    • 0026330785 scopus 로고
    • Reduction of cardiac outward currents by alpha-1 adrenoceptor stimulation: A subtype-specific effect?
    • WANG, X.L., WETTWER, E. GROSS, G. & RAVENS, U. (1991). Reduction of cardiac outward currents by alpha-1 adrenoceptor stimulation: a subtype-specific effect? J. Pharmacol. Exp. Ther., 259, 783-788.
    • (1991) J. Pharmacol. Exp. Ther. , vol.259 , pp. 783-788
    • Wang, X.L.1    Wettwer, E.2    Gross, G.3    Ravens, U.4
  • 27
    • 0015879604 scopus 로고
    • Ionic blockage of sodium channels in nerve
    • WOODHULL, A.M. (1973). Ionic blockage of sodium channels in nerve. J. Gen. Physiol., 61, 687-708.
    • (1973) J. Gen. Physiol. , vol.61 , pp. 687-708
    • Woodhull, A.M.1


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.