Small molecule antagonists of the bradykinin B1 receptor

Immunopharmacology

Volumn 43, Issue 2-3, 1999, Pages 169-177

  Horlick, Robert A ^a   Ohlmeyer, Michael H ^a   Stroke, Ilana L ^a   Strohl, Barbara ^a   Pan, Gonghua ^a   Schilling, Adriane E ^a   Paradkar, Vidyadhar ^a   Quintero, Jorge G ^a   You, Ming ^a   Riviello, Christopher ^a   Thorn, Megan B ^a   Damaj, Bassam ^a   Fitzpatrick, V Danial ^a   Dolle, Roland E ^a   Webb, Maria L ^a   Baldwin, John J ^a   Sigal, Nolan H ^a  

^a PHARMACOPEIA INC   (United States)

Author keywords

Chemical libraries; Combinatorial chemistry; GPCR; High throughput screening; Receptor binding; Receptor signaling

Indexed keywords

BRADYKININ B1 RECEPTOR; BRADYKININ B1 RECEPTOR ANTAGONIST; KALLIDIN[1-9]; PHOSPHATIDYLINOSITOL; PS 020990; UNCLASSIFIED DRUG;

CALCIUM MOBILIZATION; CONFERENCE PAPER; DRUG ACTIVITY; DRUG POTENCY; DRUG RECEPTOR BINDING; DRUG SCREENING; HUMAN; HUMAN CELL; LUNG FIBROBLAST; NEUROTRANSMISSION; PHOSPHOINOSITIDE METABOLISM; PRIORITY JOURNAL; SIGNAL TRANSDUCTION; STRUCTURE ACTIVITY RELATION;

BRADYKININ; CELL LINE; HUMANS; PEPTIDE LIBRARY; RECEPTOR, BRADYKININ B1; RECEPTORS, BRADYKININ; SIGNAL TRANSDUCTION; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 0032705731     PISSN: 01623109     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0162-3109(99)00130-7     Document Type: Conference Paper

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