-
3
-
-
0028901757
-
125I]iodophenyl)tropane-2β-carboxylic acid isopropyl ester
-
125I]iodophenyl)tropane-2β-carboxylic acid isopropyl ester. Mol Pharmacol 47:779-786.
-
(1995)
Mol Pharmacol
, vol.47
, pp. 779-786
-
-
Boja, J.W.1
Cadet, J.L.2
Kopajtic, T.A.3
Lever, J.4
Seltzman, H.H.5
Wyrick, C.D.6
Lewin, A.H.7
Abraham, P.8
Carroll, F.I.9
-
4
-
-
0025108546
-
New, potent cocaine analogs: Ligand binding and transport studies in rat striatum
-
Boja JW, Carroll FI, Rahman MA, Philip A, Lewin AH and Kuhar MJ (1990) New, potent cocaine analogs: Ligand binding and transport studies in rat striatum. Eur J Pharmacol 184:329-332.
-
(1990)
Eur J Pharmacol
, vol.184
, pp. 329-332
-
-
Boja, J.W.1
Carroll, F.I.2
Rahman, M.A.3
Philip, A.4
Lewin, A.H.5
Kuhar, M.J.6
-
6
-
-
0026460367
-
Selective dopamine transporter inhibition by cocaine analogs
-
Boja JW, McNeill RM, Lewin AH, Abraham P, Carroll FI and Kuhar MJ (1992b) Selective dopamine transporter inhibition by cocaine analogs. NeuroReport 3:984-986.
-
(1992)
NeuroReport
, vol.3
, pp. 984-986
-
-
Boja, J.W.1
McNeill, R.M.2
Lewin, A.H.3
Abraham, P.4
Carroll, F.I.5
Kuhar, M.J.6
-
7
-
-
0026802919
-
125I]RTI-55 to dopamine and serotonin transporters in rat brain
-
125I]RTI-55 to dopamine and serotonin transporters in rat brain. Synapse 12:27-36.
-
(1992)
Synapse
, vol.12
, pp. 27-36
-
-
Boja, J.W.1
Mitchell, W.M.2
Patel, A.3
Kopajtic, T.A.4
Carroll, F.I.5
Lewin, A.H.6
Abraham, P.7
Kuhar, M.J.8
-
8
-
-
0025924967
-
125I]RTI-55: A potent ligand for dopamine transporters
-
125I]RTI-55: A potent ligand for dopamine transporters. Eur J Pharmacol 194:133-134.
-
(1991)
Eur J Pharmacol
, vol.194
, pp. 133-134
-
-
Boja, J.W.1
Patel, A.2
Carroll, F.I.3
Rahman, M.A.4
Philip, A.5
Lewin, A.H.6
Kopajtic, T.A.7
Kuhar, M.J.8
-
10
-
-
0017184389
-
A rapid and sensitive method for the quantitation of microgram quantities of protein utilizing the principle of protein-dye binding
-
Bradford MM (1976) A rapid and sensitive method for the quantitation of microgram quantities of protein utilizing the principle of protein-dye binding. Anal Biochem 72:248-254.
-
(1976)
Anal Biochem
, vol.72
, pp. 248-254
-
-
Bradford, M.M.1
-
12
-
-
0032917977
-
Time course of changes in striatal dopamine transporters and D2 receptors with specific iodinated markers in a rat model of Parkinson's disease
-
Chalon S, Emond P, Bodard S, Vilar MP, Thiercelin C, Besnard JC and Guilloteau D (1999) Time course of changes in striatal dopamine transporters and D2 receptors with specific iodinated markers in a rat model of Parkinson's disease. Synapse 31:134-139.
-
(1999)
Synapse
, vol.31
, pp. 134-139
-
-
Chalon, S.1
Emond, P.2
Bodard, S.3
Vilar, M.P.4
Thiercelin, C.5
Besnard, J.C.6
Guilloteau, D.7
-
13
-
-
0015861774
-
i) and the concentration of inhibitor which causes 50 per cent inhibition (150) of an enzymatic reaction
-
i) and the concentration of inhibitor which causes 50 per cent inhibition (150) of an enzymatic reaction. Biochem Pharmacol 22:3099-3108.
-
(1973)
Biochem Pharmacol
, vol.22
, pp. 3099-3108
-
-
Cheng, Y.C.1
Prussoff, W.H.2
-
14
-
-
0028936065
-
The dopamine transporter: Immunochemical characterization and localization in brain
-
Ciliax BJ, Heilman C, Demchyshyn LL, Pristupa ZB, Ince E, Hersch SM, Niznick HB and Levey AI (1995) The dopamine transporter: Immunochemical characterization and localization in brain. J Neurosci 15:1714-1723.
-
(1995)
J Neurosci
, vol.15
, pp. 1714-1723
-
-
Ciliax, B.J.1
Heilman, C.2
Demchyshyn, L.L.3
Pristupa, Z.B.4
Ince, E.5
Hersch, S.M.6
Niznick, H.B.7
Levey, A.I.8
-
16
-
-
14444270841
-
Synthesis and ligand binding of nortropane derivatives: N-substituted 2β-carbomethoxy-3β-(4′-iodophenyl) nortropane and N-(3-iodoprop-2E-enyl)-2β-carbomethoxy-3β-(3′,4′- disubstituted phenyl)nortropane: New high-affinity and selective compounds for the dopamine transporter
-
Emond P, Garreau L, Chalon S, Boazi M, Caillet M, Bricard J, Frangin Y, Mauclaire L, Besnard J-C and Guilloteau D (1997) Synthesis and ligand binding of nortropane derivatives: N-Substituted 2β-carbomethoxy-3β-(4′-iodophenyl) nortropane and N-(3-iodoprop-2E-enyl)-2β-carbomethoxy-3β-(3′,4′- disubstituted phenyl)nortropane: New high-affinity and selective compounds for the dopamine transporter. J Med Chem 40:1366-1372.
-
(1997)
J Med Chem
, vol.40
, pp. 1366-1372
-
-
Emond, P.1
Garreau, L.2
Chalon, S.3
Boazi, M.4
Caillet, M.5
Bricard, J.6
Frangin, Y.7
Mauclaire, L.8
Besnard, J.-C.9
Guilloteau, D.10
-
19
-
-
0030877835
-
Dopamine transporter is required for in vivo MPTP neurotoxicity: Evidence from mice lacking the transporter
-
Gainetdinov RR, Fumagalli F, Jones SR and Caron MG (1997) Dopamine transporter is required for in vivo MPTP neurotoxicity: Evidence from mice lacking the transporter. J Neurochem 69:1322-1325.
-
(1997)
J Neurochem
, vol.69
, pp. 1322-1325
-
-
Gainetdinov, R.R.1
Fumagalli, F.2
Jones, S.R.3
Caron, M.G.4
-
20
-
-
0030875425
-
N-(3-iodoprop-2E-enyl)-2β-carbomethoxy-3β-(3′,4′- dichlorophenyl) nortropane (β-CDIT), a tropane derivative: Pharmacological characterization as a specific ligand for the dopamine transporter in the rodent brain
-
Garreau L, Emond P, Chalon S, Belzung C, Guilloteau D, Frangin Y, Besnard JC and Guilloteau D (1997) N-(3-iodoprop-2E-enyl)-2β-Carbomethoxy-3β-(3′,4′- dichlorophenyl) nortropane (β-CDIT), a tropane derivative: Pharmacological characterization as a specific ligand for the dopamine transporter in the rodent brain. J Pharmacol Exp Ther 282:467-474.
-
(1997)
J Pharmacol Exp Ther
, vol.282
, pp. 467-474
-
-
Garreau, L.1
Emond, P.2
Chalon, S.3
Belzung, C.4
Guilloteau, D.5
Frangin, Y.6
Besnard, J.C.7
Guilloteau, D.8
-
21
-
-
0026335164
-
Cloning and functional characterization of a cocaine-sensitive dopamine transporter
-
Giros B, El Mestikawy S, Bertrand L and Caron MG (1991) Cloning and functional characterization of a cocaine-sensitive dopamine transporter. FEBS Lett 295:149-154.
-
(1991)
FEBS Lett
, vol.295
, pp. 149-154
-
-
Giros, B.1
El Mestikawy, S.2
Bertrand, L.3
Caron, M.G.4
-
22
-
-
0030071106
-
Hyperlocomotion and indifference to cocaine and amphetamine in mice lacking the dopamine transporter
-
Giros B, Jaber M, Jones SR, Wightman RM and Caron MG (1996) Hyperlocomotion and indifference to cocaine and amphetamine in mice lacking the dopamine transporter. Nature (Lond) 379:606-612.
-
(1996)
Nature (Lond)
, vol.379
, pp. 606-612
-
-
Giros, B.1
Jaber, M.2
Jones, S.R.3
Wightman, R.M.4
Caron, M.G.5
-
23
-
-
0028337480
-
Synthesis and characterization of radioiodinated N-(3-iodopropen-1-yl)-2β-carbomethoxy-3β-(4-chlorophenyl)tropanes: Potential dopamine reuptake site imaging agents
-
Goodman MM, Kong MP, Kabalka GW, Kung HF and Switzer R (1994) Synthesis and characterization of radioiodinated N-(3-iodopropen-1-yl)-2β-carbomethoxy-3β-(4-chlorophenyl)tropanes: Potential dopamine reuptake site imaging agents. J Med Chem 37:1535-1542.
-
(1994)
J Med Chem
, vol.37
, pp. 1535-1542
-
-
Goodman, M.M.1
Kong, M.P.2
Kabalka, G.W.3
Kung, H.F.4
Switzer, R.5
-
24
-
-
0031961325
-
Exploration of the dopamine transporter: In vitro and in vivo characterization of a high-affinity and high-specificity iodinated tropane derivative (E)-N-(3-iodoprop-2-enyl)-2β-carbomethoxy-3β-(4′-methylphenyl) nortropane (PE2I)
-
Guilloteau D, Emond P, Baulieu JL, Garreau L, Frangin Y, Pourcelot L, Mauclaire L, Besnard J-C and Chalon S (1998) Exploration of the dopamine transporter: In vitro and in vivo characterization of a high-affinity and high-specificity iodinated tropane derivative (E)-N-(3-iodoprop-2-enyl)-2β-carbomethoxy-3β-(4′-methylphenyl) nortropane (PE2I). Nucl Med Biol 25:331-337.
-
(1998)
Nucl Med Biol
, vol.25
, pp. 331-337
-
-
Guilloteau, D.1
Emond, P.2
Baulieu, J.L.3
Garreau, L.4
Frangin, Y.5
Pourcelot, L.6
Mauclaire, L.7
Besnard, J.-C.8
Chalon, S.9
-
25
-
-
0032799203
-
125I]PE2I
-
125I]PE2I. Neuroimage 9:108-116.
-
(1999)
Neuroimage
, vol.9
, pp. 108-116
-
-
Hall, H.1
Halldin, C.2
Guilloteau, D.3
Chalon, S.4
Emond, P.5
Besnard, J.C.6
Farde, L.7
Sedvall, G.8
-
27
-
-
0026560079
-
The low affinity binding sites for the cocaine analog, WIN 35,428, is an artifact of freezing caudate tissue
-
Kirifides AL, Harvey JA and Aloyo VJ (1992) The low affinity binding sites for the cocaine analog, WIN 35,428, is an artifact of freezing caudate tissue. Life Sci 50:139-142.
-
(1992)
Life Sci
, vol.50
, pp. 139-142
-
-
Kirifides, A.L.1
Harvey, J.A.2
Aloyo, V.J.3
-
28
-
-
15144360264
-
Pharmacokinetics and dosimetry of iodine-123 labelled PE2I in humans, a radioligand for dopamine transporter imaging
-
Kuikka JT, Baulieu JL, Hiltunen J, Halldin C, Bergström KA, Farde L, Emond P, Chalon S, Yu M, Nikula T, Laitinen T, Karhu J, Tupala E, Hallikainen T, Kolehmainen V, Mauclaire L, Mazière B, Tiihonen J and Guilloteau D (1998) Pharmacokinetics and dosimetry of iodine-123 labelled PE2I in humans, a radioligand for dopamine transporter imaging. Eur J Nucl Med 25:531-534.
-
(1998)
Eur J Nucl Med
, vol.25
, pp. 531-534
-
-
Kuikka, J.T.1
Baulieu, J.L.2
Hiltunen, J.3
Halldin, C.4
Bergström, K.A.5
Farde, L.6
Emond, P.7
Chalon, S.8
Yu, M.9
Nikula, T.10
Laitinen, T.11
Karhu, J.12
Tupala, E.13
Hallikainen, T.14
Kolehmainen, V.15
Mauclaire, L.16
Mazière, B.17
Tiihonen, J.18
Guilloteau, D.19
-
29
-
-
0029134955
-
IPT: A novel iodinated ligand for the CNS dopamine transporter
-
Kung MP, Essman WD, Frederick D, Meegala S, Goodman M, Mu M, Lucki I and Kung HF (1995) IPT: A novel iodinated ligand for the CNS dopamine transporter. Synapse 20:316-324.
-
(1995)
Synapse
, vol.20
, pp. 316-324
-
-
Kung, M.P.1
Essman, W.D.2
Frederick, D.3
Meegala, S.4
Goodman, M.5
Mu, M.6
Lucki, I.7
Kung, H.F.8
-
31
-
-
0027997873
-
123I]β-CIT binding to dopamine transporters in healthy human subjects
-
123I]β-CIT binding to dopamine transporters in healthy human subjects. J Cereb Blood Flow Metab 14:982-994.
-
(1994)
J Cereb Blood Flow Metab
, vol.14
, pp. 982-994
-
-
Laruelle, M.1
Wallace, E.2
Seibyl, J.P.3
Baldwin, R.M.4
Zea-Ponce, Y.5
Zoghbi, S.S.6
Neumeyer, J.L.7
Charney, D.S.8
Hoffer, P.B.9
Innis, R.B.10
-
33
-
-
0031945368
-
Altropane, a SPECT or PET imaging probe for dopamine neurons: I. Dopamine transporter binding in primate brain
-
Madras BK, Meltzer PC, Liang AY, Elmaleh DR, Babich J and Fishman AJ (1998) Altropane, a SPECT or PET imaging probe for dopamine neurons: I. Dopamine transporter binding in primate brain. Synapse 29:93-104.
-
(1998)
Synapse
, vol.29
, pp. 93-104
-
-
Madras, B.K.1
Meltzer, P.C.2
Liang, A.Y.3
Elmaleh, D.R.4
Babich, J.5
Fishman, A.J.6
-
36
-
-
0025195947
-
3H]WIN 35,065-2: A ligand for cocaine receptors in striatum
-
3H]WIN 35,065-2: A ligand for cocaine receptors in striatum. J Neurochem 55:1556-1562.
-
(1990)
J Neurochem
, vol.55
, pp. 1556-1562
-
-
Ritz, M.C.1
Boja, J.W.2
Grigoriadis, D.3
Zaczek, R.4
Carroll, F.I.5
Lewis, A.H.6
Kuhar, M.J.7
-
37
-
-
0025008955
-
Cocaine inhibition of ligand binding at dopamine, norepinephrine and serotonin transporters: A structure activity study
-
Ritz MC, Cone EJ and Kuhar MJ (1990a) Cocaine inhibition of ligand binding at dopamine, norepinephrine and serotonin transporters: A structure activity study. Life Sci 46:635-645.
-
(1990)
Life Sci
, vol.46
, pp. 635-645
-
-
Ritz, M.C.1
Cone, E.J.2
Kuhar, M.J.3
-
38
-
-
0028292625
-
125I]RTI-55
-
125I]RTI-55. J Pharmacol Exp Ther 270:296-309.
-
(1994)
J Pharmacol Exp Ther
, vol.270
, pp. 296-309
-
-
Rothman, R.B.1
Cadet, J.L.2
Akunne, H.C.3
Silverthorn, M.L.4
Baumann, M.H.5
Carroll, F.I.6
Rice, K.C.7
De Costa, B.R.8
Partilla, J.S.9
Wang, J.B.10
Uhl, G.11
Glowa, J.R.12
Dersch, C.M.13
-
39
-
-
0028215940
-
Dopamine transporter messenger RNA in Parkinson's disease and control substantia nigra neurons
-
Uhl GR, Walther D, Mash D, Faucheux B and Javoy-Agid F (1994) Dopamine transporter messenger RNA in Parkinson's disease and control substantia nigra neurons. Ann Neurol 35:494-498.
-
(1994)
Ann Neurol
, vol.35
, pp. 494-498
-
-
Uhl, G.R.1
Walther, D.2
Mash, D.3
Faucheux, B.4
Javoy-Agid, F.5
|