[3H]CGP 61594, the first photoaffinity ligand for the glycine site of NMDA receptors

Neuropharmacology

Volumn 38, Issue 2, 1999, Pages 233-242

  Benke, Dietmar ^a   Honer, Michael ^a   Heckendorn, Roland ^b   Pozza, Mario F ^b   Allgeier, Hans ^b   Angst, Christof ^b   Mohler, Hanns ^a  

^a UNIVERSITY OF ZURICH   (Switzerland)

^b NOVARTIS PHARMA AG   (Switzerland)

Author keywords

Glycine site antagonist; NMDA receptor; NR1 subunit; Photoaffinity labeling

Indexed keywords

CGP 61594; GLUTAMIC ACID; GLYCINE; LIGAND; N METHYL DEXTRO ASPARTIC ACID RECEPTOR; POLYAMINE; PROTEIN; UNCLASSIFIED DRUG; AMINO ACID RECEPTOR STIMULATING AGENT; AZIDE; N METHYLASPARTIC ACID; QUINOLINE DERIVATIVE; SERINE; TRITIUM;

ANIMAL CELL; ANIMAL TISSUE; ARTICLE; BINDING SITE; BRAIN MEMBRANE; BRAIN SLICE; CONTROLLED STUDY; ELECTROPHYSIOLOGY; IMMUNOAFFINITY CHROMATOGRAPHY; MALE; NEOCORTEX; NONHUMAN; PHOTOAFFINITY LABELING; PRIORITY JOURNAL; RAT; SCATCHARD PLOT; ULTRAVIOLET IRRADIATION; AFFINITY LABELING; ANIMAL; BINDING COMPETITION; BRAIN; BRAIN CORTEX; CELL MEMBRANE; DRUG EFFECT; EVOKED RESPONSE; HIPPOCAMPUS; IN VITRO STUDY; KINETICS; METABOLISM; PHYSIOLOGY; SPRAGUE DAWLEY RAT; SYNTHESIS;

AFFINITY LABELS; ANIMALS; AZIDES; BINDING SITES; BINDING, COMPETITIVE; BRAIN; CELL MEMBRANE; CEREBRAL CORTEX; ELECTROPHYSIOLOGY; EVOKED POTENTIALS; EXCITATORY AMINO ACID AGONISTS; GLYCINE; HIPPOCAMPUS; KINETICS; LIGANDS; MALE; N-METHYLASPARTATE; NEOCORTEX; QUINOLINES; RATS; RATS, SPRAGUE-DAWLEY; RECEPTORS, N-METHYL-D-ASPARTATE; SERINE; TRITIUM;

EID: 0032589226     PISSN: 00283908     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0028-3908(98)00191-9     Document Type: Article

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