Diinosine pentaphosphate (IP5I) is a potent antagonist at recombinant rat P2X1 receptors

British Journal of Pharmacology

Volumn 128, Issue 5, 1999, Pages 981-988

  King, B F ^a   Liu, M ^a   Pintor, J ^b   Gualix, J ^b   Miras Portugal, M T ^b   Burnstock, G ^a  

^a ROYAL FREE AND UNIVERSITY COLLEGE MEDICAL SCHOOL   (United Kingdom)

^b UNIVERSIDAD COMPLUTENSE DE MADRID   (Spain)

Author keywords

Antagonist; ATP; Diinosine polyphosphate; Dinucleotide; Ion channel; IP5I; P2X receptor; Xenopus oocyte

Indexed keywords

ADENOSINE MONOPHOSPHATE DEAMINASE; ADENOSINE TRIPHOSPHATE; DIADENOSINE POLYPHOSPHATE; DIINOSINE PENTAPHOSPHATE; INOSINE PHOSPHATE; INOSINE TRIPHOSPHATE; PURINE P2X RECEPTOR; RECOMBINANT RECEPTOR; UNCLASSIFIED DRUG; ADENOSINE DEAMINASE; DINUCLEOSIDE PHOSPHATE; PURINE P2 RECEPTOR; PURINE P2X1 RECEPTOR; RECOMBINANT PROTEIN;

ANIMAL CELL; ARTICLE; COMPETITIVE INHIBITION; CONCENTRATION RESPONSE; CONTROLLED STUDY; DRUG POTENCY; DRUG SELECTIVITY; FEMALE; MEMBRANE CURRENT; NONHUMAN; OOCYTE; PRIORITY JOURNAL; RAT; RECEPTOR BLOCKING; REVERSED PHASE LIQUID CHROMATOGRAPHY; VOLTAGE CLAMP; XENOPUS; ANIMAL; ASPERGILLUS; CELL MEMBRANE POTENTIAL; DRUG ANTAGONISM; DRUG EFFECT; ELECTROPHYSIOLOGY; ELECTROSTIMULATION; ENZYMOLOGY; HIGH PERFORMANCE LIQUID CHROMATOGRAPHY; PHYSIOLOGY; XENOPUS LAEVIS;

ADENOSINE DEAMINASE; ANIMALS; ASPERGILLUS; CHROMATOGRAPHY, HIGH PRESSURE LIQUID; DINUCLEOSIDE PHOSPHATES; ELECTRIC STIMULATION; ELECTROPHYSIOLOGY; MEMBRANE POTENTIALS; OOCYTES; RATS; RECEPTORS, PURINERGIC P2; RECOMBINANT PROTEINS; XENOPUS LAEVIS;

EID: 0032585938     PISSN: 00071188     EISSN: None     Source Type: Journal    
DOI: 10.1038/sj.bjp.0702876     Document Type: Article

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