Characterization of [125I]AR-M100613, a high-affinity radioligand for δ opioid receptors

Peptides

Volumn 20, Issue 11, 1999, Pages 1327-1335

  Fraser, Graeme L ^a,b   Labarre, Maryse ^a   Godbout, Claude ^a   Butterworth, Joanne ^a   Clarke, Paul B S ^b   Payza, Kemal ^a   Schmidt, Ralf ^a  

^a ASTRAZENECA   (United Kingdom)

^b MCGILL UNIVERSITY   (Canada)

Author keywords

Binding; Delta opioid receptor; Radioligand; Rat brain; 35S GTP S

Indexed keywords

AR M 100613; DELTA OPIATE RECEPTOR; ENKEPHALIN[2 DEXTRO ALANINE 4 METHYLPHENYLALANINE 5 GLYCINE]; ENKEPHALIN[2,5 DEXTRO PENICILLAMINE]; N METHYL N [7 (1 PYRROLIDINYL) 1 OXASPIRO[4.5]DEC 8 YL]BENZENEACETAMIDE; RADIOLIGAND; UNCLASSIFIED DRUG; DELTORPHIN II, ALA(2); DELTORPHIN II, ALA(2)-; DRUG DERIVATIVE; LIGAND; NALTREXONE; NALTRINDOLE; OLIGOPEPTIDE; RADIOACTIVE IODINE;

ANIMAL EXPERIMENT; ANIMAL TISSUE; ARTICLE; BRAIN MEMBRANE; CONTROLLED STUDY; DRUG RECEPTOR BINDING; DRUG SPECIFICITY; MALE; NONHUMAN; PRIORITY JOURNAL; RADIOASSAY; RAT; ANIMAL; BRAIN; KINETICS; METABOLISM; SPRAGUE DAWLEY RAT;

ANIMALS; BRAIN; IODINE RADIOISOTOPES; KINETICS; LIGANDS; MALE; NALTREXONE; OLIGOPEPTIDES; RADIOLIGAND ASSAY; RATS; RATS, SPRAGUE-DAWLEY; RECEPTORS, OPIOID, DELTA;

EID: 0032585776     PISSN: 01969781     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0196-9781(99)00138-2     Document Type: Article

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