Solution conformation of an ET(B) selective agonist, ET-1[Cys(Acm)1,15,Ala3,Leu7,Aib11], in CD3OH/H2O by 1H NMR and molecular modelling

FEBS Letters

Volumn 425, Issue 2, 1998, Pages 234-238

  Hewage, Chandralal M ^a   Jiang, Lu ^a   Parkinson, John A ^a   Ramage, Robert ^a   Sadler, Ian H ^a  

^a UNIVERSITY OF EDINBURGH   (United Kingdom)

Author keywords

Endothelin; Molecular modeling; Nuclear magnetic resonance; Peptide solution structure

Indexed keywords

ENDOTHELIN; ENDOTHELIN B RECEPTOR; ENDOTHELIN DERIVATIVE; ENDOTHELIN RECEPTOR; RECEPTOR SUBTYPE;

ARTICLE; DRUG ACTIVITY; HIGH PERFORMANCE LIQUID CHROMATOGRAPHY; IN VITRO STUDY; MASS SPECTROMETRY; MOLECULAR MODEL; NUCLEAR MAGNETIC RESONANCE SPECTROSCOPY; PEPTIDE SYNTHESIS; PRIORITY JOURNAL; PROTEIN STRUCTURE; RECEPTOR BINDING; STRUCTURE ACTIVITY RELATION;

AMINO ACID SEQUENCE; CADMIUM COMPOUNDS; ENDOTHELIN-1; MODELS, MOLECULAR; MOLECULAR SEQUENCE DATA; NUCLEAR MAGNETIC RESONANCE, BIOMOLECULAR; PROTEIN STRUCTURE, SECONDARY; RECEPTOR, ENDOTHELIN B; RECEPTORS, ENDOTHELIN; SOLUTIONS; TEMPERATURE; WATER;

EID: 0032571570     PISSN: 00145793     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0014-5793(98)00239-7     Document Type: Article

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