A novel deprotection/functionalisation sequence using 2,4- dinitrobenzenesulfonamide: Part 2

Tetrahedron Letters

Volumn 39, Issue 13, 1998, Pages 1673-1676

  Messeri, Tommaso ^a,b   Sternbach, Daniel D ^a   Tomkinson, Nicholas C O ^a  

^a GLAXOSMITHKLINE   (United States)

^b GSK   (Italy)

Author keywords

[No Author keywords available]

Indexed keywords

2,4 DINITROBENZENESULFONAMIDE; AMIDE; CARBONIC ACID DERIVATIVE; CESIUM; DITHIOCARBAMIC ACID; HYDROXAMIC ACID; SULFONAMIDE; THIOACID; THIOAMIDE; THIOUREA DERIVATIVE; UNCLASSIFIED DRUG;

ARTICLE; CHEMICAL REACTION; CHEMICAL STRUCTURE; METHODOLOGY; ORGANIC CHEMISTRY; REACTION ANALYSIS; SYNTHESIS;

EID: 0032568330     PISSN: 00404039     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0040-4039(98)00018-5     Document Type: Article

References (11)

1. 2. An entire issue of Chemical Reviews has dealt with recent advances in combinatorial chemistry; Chem. Rev. 1997, 97, 349-509.
2. 3. Messeri, T.; Sternbach, D. D.; Tomkinson, N. C. O. Tetrahedron Lett. 1998, 39, 1669.
3. 4. (a) Bauer, L.; Exner, O. Angew. Chem. Int. Ed. Engl. 1974, 13, 376;
4. (b) Yale, H. L. Chem. Rev. 1943, 33, 209.
5. 5. Ando, W.; Hidetoshi, T. Synth. Commun. 1983, 13, 1053.
6. 6. (a) Ozaki, S. Chem. Rev. 1972, 72, 457;
7. (b) Twitchett, H. J. Chem. Soc. Rev. 1974, 3, 209.
8. 7. Brown. P. J.; Hurley, K. P.; Stuart, L. W.; Willson, T. M. Synthesis 1997, 778.
9. 8. Similar strategies have been used before. For the synthesis of dithioacids see, Zupan, M.; Bregar, Z. Tetrahedron Lett. 1990, 31, 3357. For the synthesis of dithioamides see reference 10.
10. 9. Yamazaki, N.; Tomioka, T.; Higashi, F. Synthesis 1975, 384.
11. 10. Sugimoto, N.; Makino, I.; Hirai, K. J. Org. Chem. 1988, 53, 2263.