The first total synthesis of a bioxanthracene (-)-ES-242-4, an N- methyl-D-aspartate receptor antagonist

Tetrahedron Letters

Volumn 39, Issue 13, 1998, Pages 1771-1772

  Tatsuta, Kuniaki ^a   Yamazaki, Toru ^a   Mase, Takanobu ^a   Yoshimoto, Takuji ^a  

^a WASEDA UNIVERSITY   (Japan)

Author keywords

[No Author keywords available]

Indexed keywords

ANTHRACENE DERIVATIVE; BIOXANTHRACENE; N METHYL DEXTRO ASPARTIC ACID RECEPTOR BLOCKING AGENT; UNCLASSIFIED DRUG;

ARTICLE; DIMERIZATION; DRUG HYDROLYSIS; DRUG OXIDATION; DRUG PURIFICATION; DRUG SYNTHESIS; REACTION ANALYSIS;

EID: 0032568324     PISSN: 00404039     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0040-4039(98)00040-9     Document Type: Article

References (10)

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2. 2. Toki, S.; Ando, K.; Kawamoto, I.; Sano, H.; Yoshida, M.; Matsuda, Y. J. Antibiot., 45, 1047-1054 (1992).
3. 3. Toki, S.; Tsukuda, E.; Nazawa, M.; Nonaka, H.; Yoshida, M.; Matsuda, Y. J. Biolog. Chem., 267, 14884-14892 (1992).
4. 4. Tatsuta, K.; Akimoto, K.; Annaka, M.; Ohno, Y.; Kinoshita, M. Bull. Chem. Soc. Jpn., 58, 1699-1706 (1985).
5. 5. Tatsuta, K.; Yoshimoto, T.; Gunji, H. J. Antibiot., 50, 289-290 (1997).
6. 6. Noji, M.; Nakajima, M.; Koga, K. Tetrahedron Lett., 35, 7983-7984 (1994).
7. 7. Jarglis, P.; Lichtenthaler, F. W. Tetrahedron Lett., 23, 3781-3784 (1982).
8. 8. Solladié, G.; Rubio, A.; Carreño, M. C.; Ruano, J. L. G. Tetrahedron Assym., 1, 187-198 (1990).
9. 3): 7.20(1H, s), 9.25(1H, s).
10. 10. An authentic sample of (-)-ES-242-4 was kindly provided by Dr. S. Toki, Kyowa Hakko Kogyo Co., Ltd.