Synthesis of 4-arylaminoquinazolines via 2-amino-N-arylbenzamidines

Tetrahedron Letters

Volumn 39, Issue 13, 1998, Pages 1785-1786

  Szczepankiewicz, Wojciech ^a   Suwiński, Jerzy ^a  

^a SILESIAN UNIVERSITY OF TECHNOLOGY   (Poland)

Author keywords

[No Author keywords available]

Indexed keywords

4 (3 BROMOANILINO) 6,7 DIMETHOXYQUINAZOLINE; ALUMINUM CHLORIDE; ANTHRANILIC ACID DERIVATIVE; AROMATIC AMINE; BENZAMIDINE DERIVATIVE; FORMIC ACID; NITRILE; PROTEIN TYROSINE KINASE INHIBITOR; QUINAZOLINE DERIVATIVE;

ARTICLE; CHEMICAL REACTION; DRUG ACTIVITY; DRUG SYNTHESIS; HEATING;

EID: 0032568225     PISSN: 00404039     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0040-4039(97)10864-4     Document Type: Article

References (11)

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7. 6. Armarego, W.L.F. Heterocyclic Compounds, Fused Pyrimidines, Part I, Quinazolines; Interscience Publisher: New York, 1967; p. 222.
8. 7. Giris, N.S.; Møller, J.; Pedersen, E.B. Chemica Scripta 1986, 26, 617.
9. 8. Taylor, E.C.; Ravindranathan, R.V. J.Org.Chem. 1962, 27, 2622.
10. 9. Cooper, F.C.; Partridge, M.W. Organic Syntheses 1956, 36, 64.
11. 6): δ 7.31-7.41(m,2H,4′+5′), 7.65-7.71(m,1H,6′), 7.82-7.97(m,3H,6+7+8), 8.28-8.29(m,1H,2′), 8.57-8.59 (m,1H,5), 8.70(s,1H,2), 9.90(s,1H,NH).