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Life Sciences

Volumn 63, Issue 18, 1998, Pages 1599-1609

In vitro stability and intestinal absorption characteristics of hexapeptide endothelin receptor antagonists

(5) Han, Hyo Kyung a Stewart, Barbra H b Doherty, Annette M b Cody, Wayne L b Amidon, Gordon L a

a UNIVERSITY OF MICHIGAN (United States)

b PFIZER INC (United States)

Author keywords

Biliary excretion; Endothelin antagonist; Intestinal absorption; PD 156252; Protease

Indexed keywords

AMASTATIN; CHYMOSTATIN; ENDOTHELIN A RECEPTOR; ENDOTHELIN B RECEPTOR; ENDOTHELIN C RECEPTOR; ENDOTHELIN RECEPTOR; ENDOTHELIN RECEPTOR ANTAGONIST; HEXAPEPTIDE; N ACETYL 10,11 DIHYDRO 5H DIBENZO[A,D]CYCLOHEPTEN 5 YLGLYCYLLEUCYLASPARTYLISOLEUCYLISOLEUCYLTRYPTOPHAN; PD 156252; PROTEINASE INHIBITOR; THIORPHAN; UNCLASSIFIED DRUG;

ANIMAL TISSUE; ARTICLE; BILIARY EXCRETION; CONTROLLED STUDY; DRUG DEGRADATION; DRUG ELIMINATION; DRUG HALF LIFE; DRUG STABILITY; HIGH PERFORMANCE LIQUID CHROMATOGRAPHY; INTESTINE ABSORPTION; MALE; MOUSE; NONHUMAN; URINARY EXCRETION;

NON-PROGRAMMATIC;

ANIMALS; BILE; BIOTRANSFORMATION; CHROMATOGRAPHY, HIGH PRESSURE LIQUID; INJECTIONS, INTRAVENOUS; INTESTINAL ABSORPTION; LIVER; MALE; OLIGOPEPTIDES; PROTEASE INHIBITORS; RATS; RATS, SPRAGUE-DAWLEY; RECEPTORS, ENDOTHELIN;

EID: 0032566856 PISSN: 00243205 EISSN: None Source Type: Journal
DOI: 10.1016/S0024-3205(98)00429-9 Document Type: Article

Times cited : (5)

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