Regioselective N-alkylation of 2-aminobenzylamine via chelation to 9- BBN

Tetrahedron Letters

Volumn 39, Issue 17, 1998, Pages 2643-2644

  Bar Haim, Galia ^a   Kol, Moshe ^a  

^a TEL AVIV UNIVERSITY   (Israel)

Author keywords

[No Author keywords available]

Indexed keywords

2 AMINO N ALKYLBENZYLAMINE DERIVATIVE; AMINE; BENZYLAMINE DERIVATIVE; BORANE DERIVATIVE; BUTOXIDE; CHELATE; HALIDE; POTASSIUM DERIVATIVE; UNCLASSIFIED DRUG;

ALKYLATION; ARTICLE; CHELATION; DRUG STRUCTURE; DRUG SYNTHESIS;

EID: 0032560025     PISSN: 00404039     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0040-4039(98)00227-5     Document Type: Article

References (9)

1. 1. Bar-Haim, G.; Kol, M. J. Org. Chem, 1997, 62, 6682.
2. 2. Coyne, W. E.; Cusic, J. W. J. Med. Chem. 1968, 11, 1208.
3. 3. Ishikawa, F.; Watanabe, Y.; Saegusa, J. Chem. Pharm. Bull. 1980, 28, 1357.
4. 4. Kornet, M. J. J. Heterocyclic Chem. 1992, 29, 103.
5. 5. Orth, R. E.; Jones, J. W. J. Pharm. Sci. 1961, 50, 866.
6. 6, 115.5 MHz) δ -3.7.
7. 7. Bar-Haim, G.; Shach, R.; Kol, M. Chem Commun. 1997, 229.
8. +, 80%), 106 (100%).
9. 9. Brown, H. C.; Vara Prasad, J. V. N. J. Org. Chem. 1986, 51, 4526.