Concise and regiospecific syntheses of tri-substituted 1,2,4-triazoles

Tetrahedron Letters

Volumn 39, Issue 43, 1998, Pages 7983-7986

  Dunstan, Andrew R ^a   Weber, Hans Peter ^b   Rihs, Grety ^c   Widmer, Hans ^c   Dziadulewicz, Edward K ^a  

^a Novatis Inst for Medical Sciences   (United Kingdom)

^b Nova Research Services   (Switzerland)

^c NOVARTIS PHARMA AG   (Switzerland)

Author keywords

Isomers; Peptide mimetics; Regiochemistry; Triazoles

Indexed keywords

1,2,4 TRIAZOLE DERIVATIVE; 3 (2 METHOXYBENZYLAMINO) 2 PHENYLPIPERIDINE; 3 [3,5 BIS(TRIFLUOROMETHYL)BENZYLOXY] 2 PHENYLPIPERIDINE; GUANAZOLE; GUANIDINE DERIVATIVE; NEUROKININ 1 RECEPTOR ANTAGONIST; PHENYLHYDRAZINE;

ALKYLATION; ARTICLE; CYCLIZATION; DRUG SYNTHESIS; LIGAND BINDING; MOLECULAR RECOGNITION; PKA; PROTON NUCLEAR MAGNETIC RESONANCE; STEREOCHEMISTRY; X RAY CRYSTALLOGRAPHY;

EID: 0032558673     PISSN: 00404039     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0040-4039(98)01736-5     Document Type: Article

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