Direct preparation of peptide thioesters using an Fmoc solid-phase method

Tetrahedron Letters

Volumn 39, Issue 47, 1998, Pages 8669-8672

  Li, Xiangqun ^a   Kawakami, Toru ^a   Aimoto, Saburo ^a  

^a OSAKA UNIVERSITY   (Japan)

Author keywords

Deblocking; Peptides and polypeptides; Solid phase synthesis; Thioesters

Indexed keywords

DIMETHYL SULFOXIDE; HEXAMETHYLENEIMINE DERIVATIVE; METHYLPYRROLIDINE; THIOESTER; UNCLASSIFIED DRUG;

ARTICLE; CHEMICAL REACTION; HIGH PERFORMANCE LIQUID CHROMATOGRAPHY; MASS SPECTROMETRY; PEPTIDE SYNTHESIS; REACTION ANALYSIS;

EID: 0032548051     PISSN: 00404039     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0040-4039(98)01868-1     Document Type: Article

References (18)

1. [1] Hojo H, Aimoto S, Bull. Chem. Soc. Jpn. 1991;64:111-117.
2. [2] Hojo H, Yoshimura S, Go M, Aimoto S, Bull. Chem. Soc. Jpn. 1995;68:330-336.
3. [3] Kawakami T, Kogure S, Aimoto S, Bull. Chem. Soc. Jpn. 1996;69:3331-3338.
4. [4] Merrifield RB, J. Am. Chem. Soc. 1963;85:2149-2154.
5. [5] Kent SBH, Ann. Rev. Biochem. 1988;57:957-989.
6. [6] Atherton E, Fox H, Harkiss D, Logan CJ, Sheppard RC, Williams BJ, J. Chem. Soc., Chem. Commun. 1978:537-539.
7. [7] Chang CD, Meienhofer J, Int. J. Peptide Protein Res. 1978;11:246-249.
8. [8] Dawson PE, Muir TW, Clark-Lewis I, Kent SBH, Science 1994;266:776-779.
9. [9] Canne LE, Bark SJ, Kent SBH, J. Am. Chem. Soc. 1996;118:5891-5896.
10. [10] Hackeng TM, Mounier CM, Bon C, Dawson PE, Griffin JH, Kent SBH, Proc. Natl. Acad. Sci., USA 1997;94:7845-7850.
11. [11] Tam JP, Lu YA, Liu CF, Shao J, Proc. Natl. Acad. Sci., USA 1995;92:12485-12489.
12. [12] Kawakami T, Aimoto S, Chem. Lett. 1997:1157-1158.
13. [13] Fields GB, Fields CG, J. Am. Chem. Soc. 1991;113:4202-4207.
14. [14] Martinez J, Bodanszky M, Int. J. Peptide Protein Res. 1978;12:277-283.
15. [15] Lauer JL, Fields CG, Fields GB, Lett. Peptide Science 1995;1:197-205.
16. [16] Seidah NG, Donohue-Rolfe A, Lazure C, Auclair F, Keusch GT, Chretien M, J. Biol. Chem. 1986;261:13928-13931.
17. [17] Rink H, Tetrahedron Lett. 1987;28:3787-3790.
18. [18] King DS, Fields CG, Fields GB, Int. J. Peptide Protein Res. 1990;36:255-266.