Differential α1-adrenoceptor labeling by [3H]prazosin and [3H]tamsulosin

European Journal of Pharmacology

Volumn 342, Issue 1, 1998, Pages 85-92

  Michel, Martin C ^a   Goepel, Mark ^a  

^a UNIVERSITY OF DUISBURG ESSEN   (Germany)

Author keywords

1 Adrenoceptor; Prazosin; Radioligand binding; Tamsulosin

Indexed keywords

4 (2 HYDROXYETHYL) 1 PIPERAZINEETHANESULFONIC ACID; ALPHA 1 ADRENERGIC RECEPTOR; ALPHA 1A ADRENERGIC RECEPTOR; ALPHA 1B ADRENERGIC RECEPTOR; ALPHA 1D ADRENERGIC RECEPTOR; EDETIC ACID; GLYCYLGLYCINE; PRAZOSIN; RADIOLIGAND; TAMSULOSIN; TRITIUM; TROMETAMOL; ALPHA ADRENERGIC RECEPTOR BLOCKING AGENT; NORADRENALIN; RECOMBINANT PROTEIN; SULFONAMIDE;

ANIMAL CELL; ANIMAL TISSUE; ARTICLE; CONTROLLED STUDY; HUMAN; HUMAN CELL; HUMAN TISSUE; ISOTOPE LABELING; LIGAND BINDING; MALE; NONHUMAN; PRIORITY JOURNAL; PROSTATE; RAT; RECEPTOR AFFINITY; RECEPTOR DENSITY; ANIMAL; BINDING COMPETITION; COMPARATIVE STUDY; DRUG EFFECT; IN VITRO STUDY; KINETICS; LIVER; METABOLISM; RADIOASSAY; WISTAR RAT;

ADRENERGIC ALPHA-ANTAGONISTS; ANIMALS; BINDING, COMPETITIVE; HUMANS; KINETICS; LIVER; MALE; NOREPINEPHRINE; PRAZOSIN; PROSTATE; RADIOLIGAND ASSAY; RATS; RATS, WISTAR; RECEPTORS, ADRENERGIC, ALPHA-1; RECOMBINANT PROTEINS; SULFONAMIDES;

EID: 0032545532     PISSN: 00142999     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0014-2999(97)01419-2     Document Type: Article

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