Acid-catalysed rearrangement of the n-quinazolinonyl- and n- phthalimido-aziridines derived from 3-phenylcyclohex-2-enol

Tetrahedron Letters

Volumn 39, Issue 51, 1998, Pages 9571-9572

  Marples, Brian A ^a   Toon, Richard C ^a   Slawin, Alexandra M Z ^a  

^a LOUGHBOROUGH UNIVERSITY   (United Kingdom)

Author keywords

[No Author keywords available]

Indexed keywords

3 PHENYLCYCLOHEX 2 ENOL; AZIRIDINE DERIVATIVE; DIAZADIOXABICYCLO[2.2.2]OCTANE; N PHTHALIMIDOAZIRIDINE; N QUINAZOLINONYLAZIRIDINE; OCTANE; UNCLASSIFIED DRUG;

ARTICLE; CHEMICAL REACTION; REACTION ANALYSIS; STRUCTURE ANALYSIS; SYNTHESIS;

EID: 0032542134     PISSN: 00404039     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0040-4039(98)02127-3     Document Type: Article

References (9)

1. 1. Atkinson, R. S.; Kelly, B. J. J. Chem. Soc., Perkin Trans, 1, 1989, 1515-1519.
2. 2. Dickinson, J. M.; Murphy, J. A. Tetrahedron, 1992, 48, 1317-1326.
3. 3.
4. 4. Ganboa, I.; Palomo C. Synthesis, 1986, 52-54.
5. 5. Triethylamine at -30°C directs aziridination through a triethylammonium imide:-Atkinson, R.S.; Barker, E. J. Chem. Soc., Chem. Commun., 1995, 819-820.
6. 6. Also established by X-ray crystallography-unpublished results.
7. 7. Chilmonczyk Z.; Egli M.; Behringer C.; Dreiding A. Helv. Chim. Acta, 1989, 72, 1095-1106.
8. 1H-nmr analysis of the reaction mixtures.
9. 9. Atkinson, R. S.; Fawcett, J.; Russell, D. R.; Williams, P. J. Tetrahedron Lett., 1995, 18, 3241-3244.