Inhibition of elastase by N-sulfonylaryl β-lactams: Anatomy of a stable acyl-enzyme complex

Biochemistry

Volumn 37, Issue 50, 1998, Pages 17506-17513

  Wilmouth, Rupert C ^a  

^a UNIVERSITY OF OXFORD   (United Kingdom)

Author keywords

[No Author keywords available]

Indexed keywords

BETA LACTAM ANTIBIOTIC; ELASTASE;

ARTICLE; BACTERIAL CELL WALL; BACTERIAL INFECTION; COMPLEX FORMATION; DRUG PROTEIN BINDING; ENZYME ACTIVITY; ENZYME INHIBITION; ENZYME STABILITY; HYDROLYSIS; PRIORITY JOURNAL;

AMINO ACID SEQUENCE; ANIMALS; ANTI-BACTERIAL AGENTS; AZETIDINES; BETA-LACTAMS; CASEINS; CHROMATOGRAPHY, HIGH PRESSURE LIQUID; CRYSTALLIZATION; CRYSTALLOGRAPHY, X-RAY; ENDORPHINS; MACROMOLECULAR SUBSTANCES; MAGNETIC RESONANCE SPECTROSCOPY; MASS SPECTROMETRY; MOLECULAR SEQUENCE DATA; PANCREATIC ELASTASE; PEPTIDE FRAGMENTS; SERINE PROTEINASE INHIBITORS; SOLUTIONS; SWINE;

BACTERIA (MICROORGANISMS); SUIDAE;

EID: 0032535644     PISSN: 00062960     EISSN: None     Source Type: Journal    
DOI: 10.1021/bi9816249     Document Type: Article

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