Development of 2,2-dimethylchromanol cysteinyl LT1 receptor antagonists

Bioorganic and Medicinal Chemistry Letters

Volumn 8, Issue 24, 1998, Pages 3577-3582

  Chambers, R J ^a   Antognoli, G W ^a   Cheng, J B ^a   Kuperman, A V ^a   Liston, T C ^a   Marfat, A ^a   Owens, B S ^a   Pillar, J S ^a   Shirley, J T ^a   Watson, J W ^a  

^a PFIZER INC   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

CP 265298; CP 288886; LEUKOTRIENE RECEPTOR BLOCKING AGENT; PRANLUKAST; UNCLASSIFIED DRUG; ZAFIRLUKAST;

ANIMAL CELL; ANIMAL EXPERIMENT; ANIMAL TISSUE; ARTICLE; ASTHMA; DRUG POTENCY; DRUG RECEPTOR BINDING; DRUG SYNTHESIS; HUMAN; HUMAN CELL; LIVER CLEARANCE; NONHUMAN; RAT;

ANIMALS; ANTI-ASTHMATIC AGENTS; BIOLOGICAL AVAILABILITY; GUINEA PIGS; HUMANS; LEUKOTRIENE ANTAGONISTS; MAGNETIC RESONANCE SPECTROSCOPY; MEMBRANE PROTEINS; QUINOLINES; RATS; RECEPTORS, LEUKOTRIENE; STEREOISOMERISM; THIAZOLES; U937 CELLS;

ANIMALIA;

EID: 0032535161     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0960-894X(98)00654-4     Document Type: Article

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