Differential effects of thiocyanate on the binding thermodynamics of bicuculline methiodide versus SR95531 (gabazine) to the γ-aminobutyric acid receptor-ionophore complex

Biochemical Pharmacology

Volumn 56, Issue 6, 1998, Pages 729-731

  Maksay, Gábor ^a  

^a CTRL RES INSTITUTE FOR CHEMISTRY   (Hungary)

Author keywords

Bicuculline methiodide; Chaotropic effects of thiocyanate; GABA(A) antagonists; GABA(A) receptor binding; Gabazine (SR 95531); Thermodynamics of binding

Indexed keywords

3 AMINO 2 (3 CARBOXYPROPYL) 6 (4 METHOXYPHENYL)PYRIDAZINIUM BROMIDE; 4 AMINOBUTYRIC ACID A RECEPTOR; 4 AMINOBUTYRIC ACID A RECEPTOR BLOCKING AGENT; BICUCULLINE METHIODIDE; IONOPHORE; THIOCYANATE;

ANIMAL TISSUE; ARTICLE; BRAIN SYNAPTOSOME; CONTROLLED STUDY; DRUG RECEPTOR BINDING; MALE; NONHUMAN; PRIORITY JOURNAL; RAT; THERMODYNAMICS;

ANIMALS; BICUCULLINE; COLORING AGENTS; GABA ANTAGONISTS; IONOPHORES; KINETICS; MALE; PROTEIN BINDING; PYRIDAZINES; RATS; RATS, WISTAR; RECEPTORS, GABA; TEMPERATURE; THERMODYNAMICS; THIOCYANATES;

EID: 0032530858     PISSN: 00062952     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0006-2952(98)00064-1     Document Type: Article

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