Novel inhibitors of α4β1 integrin receptor interactions through library synthesis and screening

Bioorganic and Medicinal Chemistry Letters

Volumn 8, Issue 17, 1998, Pages 2297-2302

  Souers, Andrew J ^a   Virgilio, Alex A ^a   Schürer, Stephan S ^a   Ellman, Jonathan A ^a   Kogan, Timothy P ^b   West, Henry E ^b   Ankener, Wendy ^b   Vanderslice, Peter ^b  

^a UNIVERSITY OF CALIFORNIA   (United States)

^b TEXAS BIOTECHNOLOGY CORPORATION   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

INTEGRIN; INTEGRIN RECEPTOR;

ARTICLE; CELL ADHESION; PROTEIN DOMAIN; PROTEIN PROTEIN INTERACTION; PROTEIN SECONDARY STRUCTURE; SOLID PHASE EXTRACTION; STEREOCHEMISTRY; SYNTHESIS;

ALTERNATIVE SPLICING; AMINO ACIDS; BINDING SITES; CARBOXYLIC ACIDS; DATABASES; DRUG DESIGN; INTEGRIN ALPHA4BETA1; INTEGRINS; LIGANDS; MOLECULAR CONFORMATION; MOLECULAR STRUCTURE; RECEPTORS, LYMPHOCYTE HOMING; RECEPTORS, VERY LATE ANTIGEN; REPRODUCIBILITY OF RESULTS; STEREOISOMERISM; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 0032497423     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0960-894X(98)00416-8     Document Type: Article

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