An approach to use an unusual adenosine transporter to selectively deliver polyamine analogues to trypanosomes

Bioorganic and Medicinal Chemistry Letters

Volumn 8, Issue 7, 1998, Pages 811-816

  Tye, Ching Kim ^a   Kasinathan, Ganasan ^a   Barrett, Michael P ^b   Brun, Reto ^c   Doyle, Valerie E ^a   Fairlamb, Alan H ^d   Weaver, Richard ^a   Gilbert, Ian H ^a,d  

^a CARDIFF UNIVERSITY   (United Kingdom)

^b UNIVERSITY OF GLASGOW   (United Kingdom)

^c SWISS TROPICAL AND PUBLIC HEALTH INSTITUTE   (Switzerland)

^d UNIVERSITY OF DUNDEE   (United Kingdom)

Author keywords

[No Author keywords available]

Indexed keywords

ADENOSINE; CARRIER PROTEIN; POLYAMINE DERIVATIVE;

ARTICLE; DRUG ACTIVITY; DRUG SYNTHESIS; NONHUMAN; POLYAMINE METABOLISM; PROTEIN BINDING; TRYPANOSOMA; TRYPOMASTIGOTE;

ADENOSINE; ANIMALS; BIOLOGICAL TRANSPORT; CARRIER PROTEINS; INDICATORS AND REAGENTS; KINETICS; POLYAMINES; PROTOZOAN PROTEINS; STRUCTURE-ACTIVITY RELATIONSHIP; TRYPANOCIDAL AGENTS; TRYPANOSOMA BRUCEI BRUCEI;

TRYPANOSOMA;

EID: 0032492653     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0960-894X(98)00095-X     Document Type: Article

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