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5 DeMarsh, P. L.; Frey, C. L.; Sucoloski, S. K.; Henne, S. L.; Barney, S.; Bhatnagar, P. K.; Petteway, S. R. Abstract in Program and Abstracts of the 33rd Interscience Conference on Antimicrobial Agents and Chemotherapy, New Orleans, 1993, American Society of Microbiology, p. 395.
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7 Laerum, O. D.: Sletvold, O.; Bjerknes, R.; Eriksen, J. A.; Johansen, J. H.; Schanche, J. S.; Tverteraas, T.; Paukovits, W. R. Exp. Hematol. 1988, 16, 274-280.
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Hartmann, M.9
Heerding, D.10
Hiebl, J.11
Huffman, W.F.12
Hysben, M.13
King, A.G.14
Kremminger, P.15
Kwon, C.16
LoCastro, S.17
Løvhaug, D.18
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more..
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12
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c) Schäfer, H.-J. Angew. Chem. 1981, 93, 978-1000; Angew. Chem. Int. Ed. Engl. 1981, 20, 911.
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c) Schäfer, H.-J. Angew. Chem. 1981, 93, 978-1000; Angew. Chem. Int. Ed. Engl. 1981, 20, 911.
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17
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0010580050
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PCT Int. Appl. WO 93 24,523
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b) Undheim, K.; Kremminger, P. PCT Int. Appl. WO 93 24,523; Chem. Abstracts 1995, 122, 10682a.
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Undheim, K.1
Kremminger, P.2
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3743115370
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b) Undheim, K.; Kremminger, P. PCT Int. Appl. WO 93 24,523; Chem. Abstracts 1995, 122, 10682a.
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19
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0010618614
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note
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14 Di-Boc-L,L-DAS-di-OH (12) was obtained in 18% yield with the Kolbe electrolysis and with 20% yield using the procedure described in ref. 13a. trans-1,4-Dibromo-2-butene was used for the dialkylation step because of higher diastereoselectivity compared to cis 1,4-dibromo-2-butene, 1,4-dibromobutane or 1,4-dibromo-2-butyne. The isolated yield of the dialkylation product was 45% because repeated crystallization was necessary to reach a diastereoselectivity >95%.
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21
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0010579657
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as replacement for cystine: see ref. 1; ref. 2; ref. 9
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16 a) as replacement for cystine: see ref. 1; ref. 2; ref. 9;
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-
-
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22
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0030970263
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b) as replacement for bis-(homocysteine) to stabilize a helical conformation: Andrews, M. J. I.; Tabor, A. B. Tetrahedron Lett. 1997, 38, 3063-3066.
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(1997)
Tetrahedron Lett.
, vol.38
, pp. 3063-3066
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-
Andrews, M.J.I.1
Tabor, A.B.2
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23
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0010580359
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c) as precursors for the preparation of rigid dipeptide mimetics: (i) Mueller, R.; Revesz, L. Tetrahedron Lett. 1997, 38, 3063-3066. (ii) Lombart, H.-G.; Lubell, W. D. J. Org. Chem. 1996, 61, 9437-9446 and references therein.
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(1997)
Tetrahedron Lett.
, vol.38
, pp. 3063-3066
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Mueller, R.1
Revesz, L.2
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24
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0030446803
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-
and references therein
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c) as precursors for the preparation of rigid dipeptide mimetics: (i) Mueller, R.; Revesz, L. Tetrahedron Lett. 1997, 38, 3063-3066. (ii) Lombart, H.-G.; Lubell, W. D. J. Org. Chem. 1996, 61, 9437-9446 and references therein.
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(1996)
J. Org. Chem.
, vol.61
, pp. 9437-9446
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-
Lombart, H.-G.1
Lubell, W.D.2
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27
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0010611181
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note
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19 We also investigated the Kolbe electroysis of Fmoc-Glu-OtBu. Unfortunately, no desired product of di-Fmoc-DAS-di-OtBu could be isolated from the reaction mixture.
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28
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84987592446
-
-
footnote on page 868
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20 Bold, G.; Allmendinger, T.; Herald, P.; Moesch, L.; Schär, H.-P.; Duthaler, R. O. Helv. Chim. Acta 1992, 75, 865-882 (footnote on page 868).
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(1992)
Helv. Chim. Acta
, vol.75
, pp. 865-882
-
-
Bold, G.1
Allmendinger, T.2
Herald, P.3
Moesch, L.4
Schär, H.-P.5
Duthaler, R.O.6
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29
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0010616742
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Unfortunately, Boc-Asp-OMe is not commercially available at the moment
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21 Unfortunately, Boc-Asp-OMe is not commercially available at the moment.
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