A novel series of 6-methoxy-1H-benzotriazole-5-carboxamide derivatives with dual antiemetic and gastroprokinetic activities

Bioorganic and Medicinal Chemistry Letters

Volumn 8, Issue 15, 1998, Pages 1973-1978

  Hirokawa, Yoshimi ^a   Yamazaki, Hiroshi ^a   Yoshida, Naoyuki ^a   Kato, Shiro ^a  

^a DAINIPPON SUMITOMO PHARMA CO LTD   (Japan)

Author keywords

[No Author keywords available]

Indexed keywords

6 METHOXY 1H BENZOTRIAZOLE 5 CARBOXAMIDE; DOMPERIDONE; DOPAMINE 2 RECEPTOR; DRUG DERIVATIVE; METOCLOPRAMIDE; MOSAPRIDE CITRATE; N (1 ETHYLHEXAHYDROAZEPIN 3 YL)BENZAMIDE; PROKINETIC AGENT; SEROTONIN 3 RECEPTOR; UNCLASSIFIED DRUG;

ANTIEMETIC ACTIVITY; ARTICLE; DOG; DRUG ACTIVITY; DRUG POTENCY; NONHUMAN; RAT; STOMACH EMPTYING; STRUCTURE ACTIVITY RELATION; VOMITING;

ANIMALS; ANTIEMETICS; AZEPINES; AZOCINES; DIGESTIVE PHYSIOLOGY; DIGESTIVE SYSTEM; DOGS; GASTRIC EMPTYING; GASTROINTESTINAL AGENTS; RATS; STRUCTURE-ACTIVITY RELATIONSHIP; TRIAZOLES;

EID: 0032483109     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0960-894X(98)00341-2     Document Type: Article

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