Transdermal iontophoresis of sodium nonivamide acetate. IV. Effect of polymer formulations

International Journal of Pharmaceutics

Volumn 173, Issue 1-2, 1998, Pages 127-140

  Fang, Jia You ^a,c   Huang, Yaw Bin ^a   Lin, Hung Hong ^b   Tsai, Yi Hung ^a  

^a KAOHSIUNG MEDICAL UNIVERSITY   (Taiwan)

^b CHIA NAN UNIVERSITY OF PHARMACY AND SCIENCE   (Taiwan)

^c TAIPEI MEDICAL UNIVERSITY   (Taiwan)

Author keywords

Hydrogel; Polymer; Sodium nonivamide acetate; Transdermal iontophoresis

Indexed keywords

HYDROXYMETHYLCELLULOSE; HYDROXYPROPYLCELLULOSE; HYDROXYPROPYLMETHYLCELLULOSE; METHYLCELLULOSE; MYRISTIC ACID ISOPROPYL ESTER; NONIVAMIDE; POLYMER; POVIDONE;

ARTICLE; DRUG FORMULATION; HYDROGEL; IONTOPHORESIS; PRIORITY JOURNAL; TRANSDERMAL DRUG ADMINISTRATION;

EID: 0032444168     PISSN: 03785173     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0378-5173(98)00213-0     Document Type: Article

References (39)

1. Brand, R.M., Iversen, P.L., 1996. Iontophoretic delivery of a telomeric oligonucleotide. Pharm. Res. 13, 851-854.
2. Cascone, M.G., Sim, B., Downes, S., 1995. Blends of synthetic and natural polymers as drug systems for growth hormone. Biomaterials 16, 569-574.
3. Chen, I.J., Yang, J.M., Yeh, J.L., Wu, B.N., Lo, Y.C., Chen, S.J., 1992. Hypotensive and antinociceptive effects of ether-linked and relatively non-pungent analogues of N-nonanoyl vanillylamide. Eur. J. Med. Chem. 27, 187-192.
4. Chow, D.S., Kaka, I., Wang, T.I., 1984. Concentration-dependent enhancement of 1-dodecylazacycloheptan-2-one on the percutaneous penetration kinetic of triamcinolone acetonide. J. Pharm. Sci. 73, 1794-1799.
5. Chien, Y.W., Siddiqui, O., Shi, W.M., Lelawongs, P., Liu, J.C., 1989. Direct current iontophoretic transdermal delivery of peptide and protein drug. J. Pharm. Sci. 78, 376-383.
6. D'Emanuele, A., 1996. Responsive polymeric drug delivery systems. Clin. Pharmacokinet. 31, 241-245.
7. Dempski, R.E., De Marco, J.D., Markus, A.D., 1965. An in vitro study of the relative moisture occlusive properties of several topical vehicles and saran wrap. J. Invest. Dermatol. 44, 361-363.
8. Doelker, E., Water-swollen cellulose derivatives in pharmacy. In: Peppas, N.A. (Eds.), Hydrogels in Medicine and Pharmacy, vol. II: Polymers. CRC Press, Boca Raton, FL, 1987, pp. 115-160.
9. Fang, J.Y., Wu, P.C., Huang, Y.B., Tsai, Y.H., 1995. In vitro permeation study of capsaicin and its synthetic derivatives from ointment base using various skin types. Int. J. Pharm. 126, 119-128.
10. Fang, J.Y., Wu, P.C., Huang, Y.B., Tsai, Y.H., 1996a. In vivo percutaneous absorption of capsaicin, nonivamide and sodium nonivamide acetate from ointment bases: skin erythema test and non-invasive surface recovery technique in humans. Int. J. Pharm. 131, 143-151.
11. Fang, J.Y., Huang, Y.B., Wu, P.C., Tsai, Y.H., 1996b. Transdermal iontophoresis of sodium nonivamide acetate. Consideration of electrical and chemical factors. Int. J. Pharm. 143, 47-58.
12. Fang, J.Y., Huang, Y.B., Wu, P.C., Tsai, Y.H., 1996c. Transdermal iontophoresis of sodium nonivamide acetate. II. Optimization and evaluation on solutions and gels. Int. J. Pharm. 145, 175-186.
13. Fang, J.Y., Fang, C.L., Huang, Y.B., Tsai, Y.H., 1997a. Transdermal iontophoresis of sodium nonivamide acetate. III. Combined effect of pretreatment by penetration enhancers. Int. J. Pharm. 149, 183-193.
14. Fang, J.Y., Tsai, M.J., Huang, Y.B., Wu, P.C., Tsai, Y.H., 1997b. Percutaneous absorption and skin erythema: quantification of capsaicin and its synthetic derivatives from gels incorporated with benzalkonium chloride by using non-invasive bioengineering methods. Drug Dev. Res. 40, 56-67.
15. Hadgraft, J., 1996. Pharmaceutical aspects of transdermal nitroglycerin. Int. J. Pharm. 135, 1-11.
16. Ho, H.O., Huang, F.C., Sokoloski, T.D., Sheu, M.T., 1994. The influence of cosolvents on the in-vitro percutaneous penetration of diclofenac sodium from a gel system. J. Pharm. Pharmacol. 46, 636-642.
17. Inada, H., Ghanem, A.H., Higuchi, W.I., 1994. Studies on the effects of applied voltage and duration on human epidermal membranealteration/recovery and the resultant effects upon iontophoresis. Pharm. Res. 11, 687-695.
18. Inagi, T., Marumatsu, T., Nagai, H., Terada, H., 1981. Influence of vehicle composition on the penetration of indomethacin through guinea-pig skin. Chem. Pharm. Bull. 29, 1708-1714.
19. Jones, D.S., Woolfson, A.D., Brown, A.F., 1997. Textural, viscoelastic and mucoadhesive properties of pharmaceutical gels composed of cellulose polymers. Int. J. Pharm. 151, 223-233.
20. Kasting, G.B., Bowman, L.A., 1990. DC electrical properties of frozen, excised human skin. Pharm. Res. 7, 134-143.
21. Kim, H., Fassihi, R., 1997. Application of a binary polymer system in drug release modulation. 1. Characterization of release mechanism. J. Pharm. Sci. 86, 316-322.
22. Kondo, S., Sugimoto, I., 1987. Enhancement of transdermal delivery by superfluous thermodynamic potential. I. Thermodynamic analysis of nifedipine transport across the lipoidal barrier. J. Pharmacobio-Dyn. 10, 587-594.
23. Langer, R., Brown, L., Edelman, F., 1985. Controlled release and magnetically modulated release systems for macromolecules. Methods Enzymol. 112, 399-422.
24. Lashmar, U.T., Manger, J., 1994. Investigation into the potential for iontophoresis facilitated transdermal delivery of acyclovir. Int. J. Pharm. 111, 73-82.
25. Lelawongs, P., Liu, J.C., Chien, Y.W., 1990. Transdermal iontophoretic delivery of arginine-vasopressin (II): Evaluation of electrical and operational factors. Int. J. Pharm. 61, 179-188.
26. Martin, A., Swarbrick, J., Cammarata, A., Physical Pharmacy, ch. 22, Polymer Science, Lea and Febiger, 1983, pp. 592-638.
27. Megrab, N.A., Williams, A.C., Barry, B.W., 1995. Oestradiol permeation through human skin and silastic membrane: effects of propylene glycol and supersaturation. J. Control. Release 36, 277-294.
28. Mitchell, K., Ford, J.L., Armstrong, D.J., Elliot, P.N.C., Hogan, T.E., Rostron, C., 1993. The influence of drugs on the properties of gels and swelling characteristics of matrices containing methylcellulose or hydroxypropyl methylcellulose. Int. J. Pharm. 100, 165-173.
29. Munjeri, O., Collett, J.H., Fell, J.T., 1997. Hydrogel beads based on amidated pectins for colon-specific drug delivery: the role of chitosan in modifying drug release. J. Control. Release 46, 273-278.
30. Narasimhan, B., Peppas, N.A., 1997. Molecular analysis of drug delivery systems controlled by dissolution of the polymer carrier. J. Pharm. Sci. 86, 297-304.
31. Okabe, H., Takayama, K., Nagai, T., 1992. Percutaneous absorption of ketoprofen from acrylic gel patches containing d-limonene and ethanol as absorption enhancers. Chem. Pharm. Bull. 40, 1906-1910.
32. Rao, V.U., Misra, A.N., 1994. Enhancement of iontophoretic permeation of insulin across human cadaver skin. Pharmazie 49, 538-539.
33. Santi, P., Guy, R.H., 1996. Reverse iontophoresis - Parameters determining electroosmotic flow: I. pH and ionic strength. J. Control. Release 38, 159-165.
34. Srinivasan, V., Higuchi, W.I., Sims, S.M., Ghanem, A.H., Behl, C.R., 1989. Transdermal iontophoretic drug delivery: mechanistic analysis and application to polypeptide delivery. J. Pharm. Sci. 78, 370-375.
35. Srinivasan, V., Su, M.H., Higuchi, W.I., Behl, C.R., 1990. Iontophoresis of polypeptides: Effect of ethanol pretreatment of human skin. J. Pharm. Sci. 79, 588-591.
36. Takahashi, Y., Nambu, N., Nagai, T., 1978. Interaction of several nonsteroidal antiinflammatory drugs with pectin in aqueous solution and in solid state. Chem. Pharm. Bull. 26, 3836-3842.
37. Tsai, Y.H., Huang, Y.B., Fang, J.Y., Wu, P.C., 1994. Percutaneous absorption of capsaicin and its derivatives. Drug Dev. Ind. Pharm. 20, 719-730.
38. Wakerly, Z., Fell, J., Attwood, D., Parkins, D., 1997. Studies on amidated pectins as potential carriers in colonic drug delivery. J. Pharm. Pharmacol. 49, 622-625.
39. Williams, A.C., Barry, B.W., 1991. The enhancement index concept applied to terpene penetration enhancers for human skin and model lipophilic (oestradiol) and hydrophilic (5-fluorouracil) drugs. Int. J. Pharm. 74, 157-168.