Process development of 5-methoxy-1H-indole-2-carboxylic acid from ethyl 2-methylmalonate

Organic Process Research and Development

Volumn 2, Issue 4, 1998, Pages 214-220

  Bessard, Yves ^a  

^a LONZA AG   (Switzerland)

Author keywords

[No Author keywords available]

Indexed keywords

EID: 0032337066     PISSN: 10836160     EISSN: None     Source Type: Journal    
DOI: 10.1021/op980006x     Document Type: Article

References (6)

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3. (b) Caubere, P.; Jamart-Gregoire, B.; Caubere, C.; Bizot-Espiard, J. G.; Renard, P.; Adam, G. Eur. Pat. Appl. EP 624,575 (Chem. Abstr. 1995, 122, 81177f).
4. (c) Morales-Rios, M. S.; Joseph-Nathan, P. Rev. Soc. Quim. Méx. 1989, 33, 331.
5. (a) Romero, D. L.; Morge, R. A.; Biles, C.; Berrios-Pèna, N.; May, P. D.; Palmer, J. R.; Johnson, P. D.; Smith, H. W.; Busso, M.; Tan, C. K.; Voorman, R. L.; Reusser, F.; Althaus, I. W.; Downey, K. M.; So, A. G.; Resnick, L.; Tarpley, W. G.; Aristoff, P. A. J. Med. Chem. 1994, 37, 999.
6. (b) Livermore; D. G. H.; Bethell, R. C.; Cammack, N.; Hancock, A. P.; Hann, M. M.; Green, D. V. S.; Lamont, R. B.; Noble, S. A.; Orr, D. C.; Payne, J. J.; Ramsay, M. V. J.; Shingler, A. H.; Smith, C.; Storer, R.; Williamson, C.; Willson, T. J. Med. Chem. 1993, 36, 3784.