A novel synthesis of heterocyclic compounds containing coumarin moiety of potential antimicrobial activity

Archives of Pharmacal Research

Volumn 21, Issue 6, 1998, Pages 723-728

  Abd El Fattah, M E ^a  

^a Suez Canal University   (Egypt)

Author keywords

4 Methyl 2 oxo 2H benzopyran 7 yl oxoacetyl hydrazine; Acid azide; Antimicrobial activity; Coumarin; Heterocyclic compounds

Indexed keywords

ACID ANHYDRIDE; ANTIINFECTIVE AGENT; COUMARIN DERIVATIVE; HETEROCYCLIC COMPOUND; PHTHALAZINE DERIVATIVE;

ARTICLE; CHEMISTRY; DRUG SCREENING; IN VITRO STUDY; SYNTHESIS;

ANHYDRIDES; ANTI-INFECTIVE AGENTS; COUMARINS; DRUG EVALUATION; HETEROCYCLIC COMPOUNDS; PHTHALAZINES;

EID: 0032240187     PISSN: 02536269     EISSN: None     Source Type: Journal    
DOI: 10.1007/bf02976765     Document Type: Article

References (14)

1. Chakraborty, D. P., Dasgupta, A. and Bose, P. K., Antifungal action of some natural coumarins. Ann, Biochem. and Exptl. Med. (Calcutta), 17, 59-62 (1957)
2. [C. A. 52, 1352].
3. El-Deen, I. M., Synthesis and reaction of a 4-methyl-3-(3′-thioxo)-1′-2′-4′-triazol-5′- ylcoumarin. J. Indian. Chem. Soc., 69 (1992).
4. El-Deen, I. M., Abd El-Fattah, M. E. and El Tamany, S. H., Some reactions of 5-mercapto-3,4 (di-p-chlorophenyl)-2,3-dihydro-1,2,4-triazole. Arch. Pharm. Res., 17, 294-297 (1994).
5. El-Kerdawy, M. M., Eisa, M., Barghash, A. and Marouf, A., Development of some 1,3,4-oxadiazoles, a 1,3,4-thiadiazol as potential antimicrobial agents. Sulfur, Lett., 10, 57-70 (1989).
6. El-Tamany, S. H., El-Deen, I. M., and El-Fattah, M. E., Synthesis and biological activity of 1-(4-methyl-2-oxo-2H-1-benzopyran-7-yloxoacetyl)-4-alkylthiosemicarbazides; 1,3/4-thiadiazo!esand 1,2,4-triazoles. Pak. J. Sci. Ind. Res., 38, 115 (1995).
7. Hofmann, K., Johi, A., Furlemeier, A. E. and Kappeler, H., Polypeptides VIII. Synthesis of peptides related to corticotropin. J. Am. Chem. Soc., 79, 1636 (1957).
8. Hofmann, K., Thompson, T. A. and Yajima, H., Polypeptides XIV. Synthesis of peptides related to the N-terminal of α-MSH and of the corticotropins. J. Am. Chem., 82, 3715 (1960).
9. Muria, A. D., Cole, A. I. J. and Walker, J. R. L., Antibiotic compounds from New Zealand and antidermatiphyte agent from Schefflera digitate. Planta Medica, 44, 129-133 (1982).
10. Soliman, A. Y., El Assy, N. B., El-Shahed, F., El-Kady, M., El-Deen, I. M., Synthesis and reactions of a 2-(4-methyl-2-oxo-2H-1-benzopyran-7-yloxomethyl)-4H-3,1-benzoxazin-4-one. Indian J. Chem., 29B, 326 (1990)
11. [C. A. 113, 78293].
12. Toda, T., Tokunaga, T., Ouchida, T., Shiroya, K. and Nakamoto, T., Chemotherapeutic agents. 1. The antibacterial activity of pyrone derivatives in vitro. Chemotherapy (Tokyo), 6, 91-5 (1958)
13. [C. A. 52, 203888].
14. Yousif, M. Y., Ismaeil, A. M., El Emam, A. A. and El-Kerdawy, M. M., Synthesis of substituted mercapto-1, 2,4-triazoles and substituted 1,2,4-triazol-5-yl mercaptomethyl-1,3,4-oxadiazoles and antimicarbial agents. J. Chem. Soc. 8, 183 (1996) (Pakistan).