Histamine receptor-independent muscle relaxation elicited by a series of histamine H2-receptor agonists on the isolated guinea pig duodenum: A study into the mechanism of action

General Pharmacology

Volumn 31, Issue 4, 1998, Pages 643-651

  Coruzzi, Gabriella ^a   Poli, Enzo ^a   Pozzoli, Cristina ^a   Bertaccini, Giulio ^a   Timmerman, Henk ^b  

^a UNIVERSITY OF PARMA   (Italy)

^b VU UNIVERSITY AMSTERDAM   (Netherlands)

Author keywords

H2 Receptor agonists; Intestinal muscle; Receptor independent effect; Spasmolytic activity

Indexed keywords

1,4 DIHYDRO 2,6 DIMETHYL 5 NITRO 4 [2 (TRIFLUOROMETHYL)PHENYL] 3 PYRIDINECARBOXYLIC ACID METHYL ESTER; [[7 [[2 (3 CHLOROPHENYL) 2 HYDROXYETHYL]AMINO] 5,6,7,8 TETRAHYDRO 2 NAPHTHYL]OXY]ACETIC ACID ETHYL ESTER; ACETYLCHOLINE; ALPHA METHYLHISTAMINE; AMILORIDE; AMTHAMINE; ATROPINE; CHELERYTHRINE; CLOBENPROPIT; DIMAPRIT; FAMOTIDINE; FORSKOLIN; HISTAMINE H2 RECEPTOR; HISTAMINE H2 RECEPTOR ANTAGONIST; HISTIDINE DERIVATIVE; HOMODIMAPRIT; IMPROMIDINE; ISOBUTYLMETHYLXANTHINE; LIDOCAINE; MEPYRAMINE; MEPYRAMINE MALEATE; N(G) NITROARGININE METHYL ESTER; NIFEDIPINE; NITROPRUSSIDE SODIUM; ONDANSETRON; PINACIDIL; PROCAINE; RUTHENIUM RED; TETRODOTOXIN; TETRYLAMMONIUM; THIOPERAMIDE; TOLAZOLINE; TRIFLUOPERAZINE; UNINDEXED DRUG; ZAPRINAST;

ANIMAL TISSUE; ARTICLE; CONTROLLED STUDY; GUINEA PIG; INTESTINE CONTRACTION; INTESTINE MUSCLE; MALE; MUSCLE RELAXATION; NONHUMAN; PRIORITY JOURNAL; STRUCTURE ACTIVITY RELATION;

ANIMALS; DIMAPRIT; DUODENUM; ELECTRIC STIMULATION; GUINEA PIGS; HISTAMINE AGONISTS; IMPROMIDINE; MALE; MUSCLE CONTRACTION; MUSCLE, SMOOTH; PARASYMPATHOLYTICS; STRUCTURE-ACTIVITY RELATIONSHIP; THIAZOLES;

EID: 0032190453     PISSN: 03063623     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0306-3623(98)00077-9     Document Type: Article

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