Rapid x-ray diffraction analysis of HIV-1 protease-inhibitor complexes: Inhibitor exchange in single crystals of the bound enzyme

Acta Crystallographica Section D: Biological Crystallography

Volumn 54, Issue 5, 1998, Pages 1053-1060

  Munshi, Sanjeev ^a   Chen, Zhonguo ^a   Ying, L I ^a   Olsen, David B ^a   Fraley, Mark E ^a   Hungate, Randall W ^a   Kuo, Lawrence C ^a  

^a MERCK RESEARCH LABORATORIES   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

PROTEINASE; PROTEINASE INHIBITOR;

ARTICLE; BINDING SITE; CHEMICAL STRUCTURE; CHEMISTRY; COMPARATIVE STUDY; CRYSTALLIZATION; DRUG DESIGN; MACROMOLECULE; MOLECULAR GENETICS; PROTEIN BINDING; PROTEIN CONFORMATION; X RAY CRYSTALLOGRAPHY;

BINDING SITES; CRYSTALLIZATION; CRYSTALLOGRAPHY, X-RAY; DRUG DESIGN; HIV PROTEASE; HIV PROTEASE INHIBITORS; MACROMOLECULAR SUBSTANCES; MODELS, MOLECULAR; MOLECULAR SEQUENCE DATA; PROTEIN BINDING; PROTEIN CONFORMATION;

HUMAN IMMUNODEFICIENCY VIRUS 1;

EID: 0032169572     PISSN: 09074449     EISSN: None     Source Type: Journal    
DOI: 10.1107/S0907444998003588     Document Type: Article

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