Enzymatic synthesis of [4-methoxy-11C]daunorubicin for functional imaging of P-glycoprotein with PET

Applied Radiation and Isotopes

Volumn 49, Issue 7, 1998, Pages 811-813

  Eriks Fluks, E ^a   Elsinga, P H ^a   Hendrikse, N H ^a   Franssen, E J F ^a   Vaalburg, W ^a  

^a UNIVERSITY MEDICAL CENTER GRONINGEN   (Netherlands)

Author keywords

[No Author keywords available]

Indexed keywords

CATALYST ACTIVITY; DIAGNOSTIC RADIOGRAPHY; ENZYMES; POSITRON EMISSION TOMOGRAPHY; SYNTHESIS (CHEMICAL);

FUNCTIONAL IMAGING; P GLYCOPROTEINS;

RADIOACTIVE MATERIALS;

4 METHOXYDAUNORUBICIN; CARBON 11; CARUBICIN; DAUNORUBICIN DERIVATIVE; GLYCOPROTEIN P; METHYLTRANSFERASE; S METHYLMETHIONINE; UNCLASSIFIED DRUG;

ARTICLE; DRUG SYNTHESIS; ISOTOPE LABELING; METHYLATION; MULTIDRUG RESISTANCE; POSITRON EMISSION TOMOGRAPHY; PRIORITY JOURNAL;

CARBON RADIOISOTOPES; CARUBICIN; DAUNORUBICIN; ISOTOPE LABELING; METHYLATION; P-GLYCOPROTEIN; RADIOPHARMACEUTICALS; TOMOGRAPHY, EMISSION-COMPUTED;

EID: 0032128465     PISSN: 09698043     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0969-8043(97)00302-3     Document Type: Article

References (8)

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5. Elsinga, P. H., Franssen, E. J. F., Hendrikse, N. H., Fluks, L., Weemaes, A. M. A., van der Graaf, W. T. A., de Vries, E. G. E., Visser, G. M. and Vaalburg, W. (1996) Carbon-11-labeled daunorubicin and verapamil for probing P-glycoprotein in tumors with PET. J. Nucl. Med. 37, 1571-1575.
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