Synthesis and biological activity of branched enkephalin analogues

European Journal of Medicinal Chemistry

Volumn 33, Issue 4, 1998, Pages 255-266

  Bobrova, Irina ^a,b   Abissova, Natalia ^a   Mishlakova, Natalia ^a   Rozentals, Guntis ^a   Chipens, Gunar ^a  

^a LATVIAN INSTITUTE OF ORGANIC SYNTHESIS   (Latvia)

^b KAROLINSKA UNIVERSITY HOSPITAL   (Sweden)

Author keywords

Analgesic effect; Binding assay; Enkephalin analog; GPI and MVD bioassay; Peptide synthesis

Indexed keywords

ENKEPHALIN DERIVATIVE; TYROSYL (N DELTA PROLYL) DEXTRO ORNITHYL GLYCYL PHENYLALANINE AMIDE; UNCLASSIFIED DRUG;

AMIDATION; AMINO ACID COMPOSITION; ANALGESIA; ARTICLE; BINDING AFFINITY; CARBOXY TERMINAL SEQUENCE; CYCLIZATION; DRUG RECEPTOR BINDING; DRUG SYNTHESIS; NONHUMAN; PEPTIDE SYNTHESIS;

EID: 0032051819     PISSN: 02235234     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0223-5234(98)80060-3     Document Type: Article

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