Synthesis of 2-[18F]fluoro-3-[2(S)-2-azetidinylmethoxy]pyridine, a highly potent radioligand for in vivo imaging central nicotinic acetylcholine receptors

Journal of Labelled Compounds and Radiopharmaceuticals

Volumn 41, Issue 5, 1998, Pages 451-463

  Dolle, Frédéric ^a   Valette, Héric ^a   Bottlaender, Michel ^a   Hinnen, Françoise ^a   Vaufrey, Françoise ^a   Guenther, Ilonka ^a   Crouzel, Christian ^a  

^a SERVICE HOSPITALIER FRÉDÉRIC JOLIOT   (France)

Author keywords

A 85380; Fluorine 18; Nicotinic receptors; Positron emission tomography

Indexed keywords

CHELATION; FLUORINE; FLUORINE COMPOUNDS; IONS; LEAD COMPOUNDS; LIGANDS; POSITRON EMISSION TOMOGRAPHY; SYNTHESIS (CHEMICAL);

A-85380; ACETYLCHOLINE RECEPTOR; EPIBATIDINE; FLUORIDE ION; FLUORINE-18; IN-VIVO IMAGING; NICOTINIC ACETYLCHOLINE; NICOTINIC RECEPTOR; RADIOLABELLING; RADIOLIGANDS;

PYRIDINE;

2 FLUORO 3 (AZETIDINYLMETHOXY)PYRIDINE F 18; 3 [2 AZETIDINYLMETHOXY]PYRIDINE; DIMETHYL SULFOXIDE; EPIBATIDINE; FLUORINE 18; NICOTINIC RECEPTOR; RECEPTOR SUBTYPE; UNCLASSIFIED DRUG;

ARTICLE; HIGH PERFORMANCE LIQUID CHROMATOGRAPHY; ISOTOPE LABELING; MICROWAVE RADIATION; NONHUMAN; POSITRON EMISSION TOMOGRAPHY; RADIOACTIVITY; RADIOCHEMISTRY; RAT; SYNTHESIS; THALAMUS;

EID: 0031966027     PISSN: 03624803     EISSN: None     Source Type: Journal    
DOI: 10.1002/(SICI)1099-1344(199805)41:5<451::AID-JLCR111>3.0.CO;2-R     Document Type: Article

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