Comparison of the effects and disposition kinetics of articaine and lidocaine in 20 patients undergoing intravenous regional anaesthesia during day case surgery

Pharmacy World and Science

Volumn 20, Issue 2, 1998, Pages 88-92

  Simon, Marc A M ^a   Vree, Tom B ^b   Gielen, Mathieu J M ^b   Booij, Leo H D J ^b  

^a MEDISCH SPECTRUM TWENTE   (Netherlands)

^b RADBOUD UNIVERSITY MEDICAL CENTER   (Netherlands)

Author keywords

Articaine; Disposition; Elimination kinetics; Intravenous regional analgesia; Lidocaine

Indexed keywords

ARTICAINE; LIDOCAINE;

ADULT; AGED; ARTICLE; DRUG BLOOD LEVEL; DRUG CLEARANCE; DRUG DISPOSITION; DRUG ELIMINATION; DRUG HALF LIFE; DRUG HYDROLYSIS; FEMALE; HUMAN; HUMAN EXPERIMENT; INTRAVENOUS REGIONAL ANESTHESIA; MALE;

ADULT; ANESTHESIA, CONDUCTION; ANESTHESIA, INTRAVENOUS; ANESTHETICS, LOCAL; AREA UNDER CURVE; CARTICAINE; DOUBLE-BLIND METHOD; FEMALE; HALF-LIFE; HUMANS; LIDOCAINE; MALE; MIDDLE AGED;

EID: 0031959825     PISSN: 09281231     EISSN: None     Source Type: Journal    
DOI: 10.1023/A:1008622018161     Document Type: Article

References (37)

1. Bier A. Über einen neuen Weg Lokal anästhesie an der Gliedmaassen zu erzeugen. Arch Klin Chir 1908; 86: 1007-16.
2. Davies JAH, Gill SS, Weber JCP. Intravenous regional anaesthesia using bupivacaine. Anesthesia 1981; 36: 1059-60.
3. Albright GA. Cardiac arrest following regional anesthesia with etidocaine or bupivacaine. Anesthesiology 1979; 51: 285-6.
4. Heath ML. Bupivacaine toxicity and Bier blocks. Anesthesiology 1983; 59:481.
5. Heath ML. Deaths after intravenous regional anaesthesia. Br Med J 1982; 285: 913-4.
6. Van Oss GECJM, Vree TB, Baars AM, Termond EFS, Booij LHDJ. Pharmacokinetics, metabolism, and renal excretion of articaine and its metabolite articainic acid in patients after epidural administration. Eur J Anaesthesiol 1989; 6: 49-56.
7. Eerola R. A comparative study of carticaine and prilocaine in regional intravenous analgesia. Prakt Anästh 1974; 9: 171-5.
8. Adams JP, Dealy EJ, Kenmore PI. Intravenous regional anesthesia in hand surgery. J Bone Jt Surg 1964; 46A; 811-6.
9. Bell HM, Slater EM, Harris WH. Regional anesthesia with intravenous lidocaine. J Am Med Assoc 1963;186: 544-9.
10. Biscoping J. Die intravenöse Regionalanästhesie des Armes (IVRA). Wiener Medizinische Wochenschrift 1993; 143: 179-83.
11. Eriksson E, Persson A, Örtengren B. Intravenous regional anaesthesia - an attempt to determine the safety of the method and a comparsion between prilocaine and lidocaine. Acta Chirurg Scand 1966; Suppl 358:47-54.
12. Miles DW, James JL, Clark DE, Whitwam JG. Site of action of intravenous regional anaesthesia. J Neurol Neurosurg Psychiat 1964; 27: 574-6.
13. Moller RA, Covino BG. Cardiac electrophysiologic effects of articaine compared with bupivacaine and lidocaine. Anesth Analg 1993; 76: 1266-73.
14. Schüle H. Klinisch-experimentelle Untersuchungen über die Verkerhrstüchtigkeit nach zahnärztlichen Eingriffen. Dtsch Zahnarzt Z 1980; 35: 183-9.
15. Wörner H, Frank S, Stumpf H. Lokalanästhesie und Verkehrstüchtigkeit. Dtsch Zahnärztl Z 1980; 35: 377-84.
16. Tam YK, Tawfik SR, Ke J, Coutts RT, Gray MR, Wyse DG. Highperformance liquid chromatography of lidocaine and nine of its metabolites in human plasma and urine. J Chromatogr 1987; 423: 199-206.
17. Vree TB, Baars AM, van Oss GECJM, Booij LHDJ. High performance liquid chromatography and preliminary pharmacokinetics of articaine and its 2-carboxy metabolite in humans in serum and urine. J Chromatogr 1988; 424: 440-4.
18. Proost JH, Meijer DKW. MW/Pharm, an integrated software package for drug dosage regimen calculation and therapeutic drug monitoring. Comput Biol Med 1992; 22: 155-63.
19. Holmes CMcK. Intravenous regional analgesia. A useful method of producing analgesia of the limbs. Lancet 1963; A: 245-7.
20. Lofgren N, Tegner C. Studies on local anesthetics. XX. Synthesis of some α-monoalkylamino-2-methyl propionanilides. Acta Chem Scand 1960; 14: 486-9.
21. Bonica JJ. Regional anesthetica with tetracaine. Anesthesiology 1950; 11: 716-29.
22. Merrifield AJ, Carter SJ. Intravenous regional analgesia: lignocaine blood levels. Anaesthesia 1965; 20: 287-303
23. Hargrove RL, Hoyle JR, Parker JBR, Beckett AH, Boyes RN. Blood lignocaine levels following intravenous regional analgesia. Anaesthesia 1966; 21: 37-41.
24. Dickler DJ, Friedman PL, Susman IC. Intravenous regional anesthesia with chloroprocaine. Anesthesiology 1965; 26: 244-5.
25. Pitkänen MT, Suzuki N, Rosenberg PH. Intravenous regional anaesthesia with 0.5% prilocaine or 0.5% chloroprocaine. A double blind comparison in volunteers. Anaesthesia 1992; 47: 618-9.
26. Borchard U, Niesel HC. Grundlagen der Pharmakologie der Lokalanästhetika. In: Niesel HC, ed. Regionalanästhesie Lokalanästhesie Regionale Schmerztherapie. Stuttgart, New York: Georg Thieme Verlag, 1994: 35-68.
27. Niesel HC. Klinische Pharmakologie und Toxikologie. Anwendung der Lokalanästhetika. In: Niesel HC, ed. Regionalanästhesie Lokalanästhesie Regionale Schmerztherapie. Stuttgart, New York: Georg Thieme Verlag, 1994; 69-165.
28. Thorn-Alquist AM. Blood concentrations of local anaesthetics after intravenous regional anaesthesia. Acta Anaesth Scand 1969; 13: 229-40.
29. Covino BG. Pharmacokinetics of local anaesthetic drugs: In: Prys-Robert C, Hug CG, eds. Pharmacokinetics of Anaesthesia. Oxford: Blackwell Sci Publishers, 1984; 270-92.
30. Akerman B, Aström A, Ross S, Telc A. Studies on absorption, distribution and metabolism of labelled prilocaine and lidocaine in some animals. Acta Pharmacol Toxicol 1966; 24: 389-403.
31. Sorbie C, Chacha P. Regional anaesthesia by the intravenous route. Br Med J 1965; 1: 957-60.
32. Deacock ARC, Simpson WT. Fatal reactions to lignocaine. Anaesthesia 1964; 19: 217-21.
33. Pieper JA, Rodman JH. Lidocaine. In: Evans WE, Schentag JJ, Jusko WJ, Harrison H, eds. Applied Pharmacokinetics. Principles of Therapeutic Monitoring (Second Edition). Spokane, USA: Applied Therapeutics Inc, 1986: 639-81.
34. Van Oss GECJM, Vree TB, Baars AM, Termond EFS, Booij LHDJ. Clinical effects and pharmacokinetics of articainic acid in one volunteer after intravenous administration. Pharm Weekbl [Sci] 1988; 10: 284-7.
35. De Jong R. Biotransformation of local anesthetics: general concepts, Int Anesthesiol Clin 1975; 13: 1-20.
36. Boyes RN. A review of the metabolism of amide local anaesthetic agents. Br J Anaesth 1975; 47: 225-30.
37. Tucker GT, Mather LE. Clinical pharmacokinetics of local anaesthetics. Clin Pharmacokin 1979; 4: 241-78.