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Volumn 101, Issue 4 SUPPL., 1998, Pages

Development of fluticasone propionate and comparison with other inhaled corticosteroids

Author keywords

Asthma; Fluticasone propionate; Inhaled corticosteroids; Structure activity relationships

Indexed keywords

BECLOMETASONE DIPROPIONATE; BECLOMETHASONE 17 MONOPROPIONATE; BUDESONIDE; CD3 ANTIGEN; CD4 ANTIGEN; CD8 ANTIGEN; CORTICOSTEROID; CYTOKINE; DEXAMETHASONE; FLUNISOLIDE; FLUOCINOLONE ACETONIDE; FLUTICASONE PROPIONATE; GLUCOCORTICOID RECEPTOR; HISTAMINE; HLA DR ANTIGEN; IMMUNOGLOBULIN E; INTERLEUKIN 2 RECEPTOR; METHYLPREDNISOLONE; MOMETASONE FUROATE; T LYMPHOCYTE ANTIGEN; TRIAMCINOLONE ACETONIDE; UNCLASSIFIED DRUG;

EID: 0031957726     PISSN: 00916749     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0091-6749(98)70155-1     Document Type: Article
Times cited : (122)

References (29)
  • 1
    • 0027494730 scopus 로고
    • Anti-inflammatory actions of steroids: Molecular mechanism
    • Barnes PJ, Adcock IM. Anti-inflammatory actions of steroids: molecular mechanism. Trends Pharmacol Sci 1993;14:436-41.
    • (1993) Trends Pharmacol Sci , vol.14 , pp. 436-441
    • Barnes, P.J.1    Adcock, I.M.2
  • 2
    • 0002469339 scopus 로고
    • Locally active corticosteroids: Structure-activity relationships
    • Wilson L, Markes R, editor. London: Churchill Livingstone
    • Phillipps GH. Locally active corticosteroids: structure-activity relationships. In: Wilson L, Markes R, editor. Mechanisms of topical corticosteroid activity. London: Churchill Livingstone; 1976. p. 1-18.
    • (1976) Mechanisms of Topical Corticosteroid Activity , pp. 1-18
    • Phillipps, G.H.1
  • 3
    • 0028135124 scopus 로고
    • Synthesis and structure-activity relationships in a series of anti-inflammatory corticosteroid analogues, halomethyl androstane-17β-carbothiates and 17β-carboselenoates
    • Phillipps GH, Bailey EJ, Bain BM, Borella RA, Buckton JB, Clark JC, et al. Synthesis and structure-activity relationships in a series of anti-inflammatory corticosteroid analogues, halomethyl androstane-17β-carbothiates and 17β-carboselenoates. J Med Chem 1994;37:3717-29.
    • (1994) J Med Chem , vol.37 , pp. 3717-3729
    • Phillipps, G.H.1    Bailey, E.J.2    Bain, B.M.3    Borella, R.A.4    Buckton, J.B.5    Clark, J.C.6
  • 4
    • 0013806318 scopus 로고
    • A bio-assay for the concomitant assessment of the antiphlogistic and thymolytic activities of topically applied corticoids
    • Tonelli G, Thibault L, Ringler I. A bio-assay for the concomitant assessment of the antiphlogistic and thymolytic activities of topically applied corticoids. Endocrinology 1965;77:625-34.
    • (1965) Endocrinology , vol.77 , pp. 625-634
    • Tonelli, G.1    Thibault, L.2    Ringler, I.3
  • 5
    • 0000324473 scopus 로고
    • The estimation of small amounts of corticosterone in rat plasma
    • Zenker N, Bernstein DE. The estimation of small amounts of corticosterone in rat plasma. J Biol Chem 1958;231:695-701.
    • (1958) J Biol Chem , vol.231 , pp. 695-701
    • Zenker, N.1    Bernstein, D.E.2
  • 6
    • 84915066328 scopus 로고
    • Percutaneous absorption of steroids
    • McKenzie AW. Percutaneous absorption of steroids. Arch Dermatol 1962;86:611-4.
    • (1962) Arch Dermatol , vol.86 , pp. 611-614
    • McKenzie, A.W.1
  • 7
    • 0015912235 scopus 로고
    • A comparison of the molecular structures of six corticosteroids
    • Weeks CM, Duax WL, Wolff ME. A comparison of the molecular structures of six corticosteroids. J Am Chem Soc 1973;95:2865-8.
    • (1973) J Am Chem Soc , vol.95 , pp. 2865-2868
    • Weeks, C.M.1    Duax, W.L.2    Wolff, M.E.3
  • 8
    • 0025092716 scopus 로고
    • Structure-activity relationships of topically active steroids: The selection of fluticasone propionate
    • Phillipps GH. Structure-activity relationships of topically active steroids: the selection of fluticasone propionate. Respir Med 1990;84(suppl):19-23.
    • (1990) Respir Med , vol.84 , Issue.SUPPL. , pp. 19-23
    • Phillipps, G.H.1
  • 9
    • 0030048729 scopus 로고    scopus 로고
    • Pharmacodynamics and pharmacokinetics of inhaled glucocorticoids
    • Johnson M. Pharmacodynamics and pharmacokinetics of inhaled glucocorticoids. J Allergy Clin Immunol 1996;97:169-76.
    • (1996) J Allergy Clin Immunol , vol.97 , pp. 169-176
    • Johnson, M.1
  • 10
    • 0000419721 scopus 로고
    • Dissolution tissue binding and kinetics of receptor binding of inhaled glucocorticoids
    • Högger P, Rawert L, Rohdewald P. Dissolution tissue binding and kinetics of receptor binding of inhaled glucocorticoids. Eur Respir J 1993;6:584s.
    • (1993) Eur Respir J , vol.6
    • Högger, P.1    Rawert, L.2    Rohdewald, P.3
  • 11
    • 0003230473 scopus 로고
    • Efflux of glucocorticoids from human lung tissue to human plasma in vitro
    • Högger P, Bonsmann U, Rohdewald P. Efflux of glucocorticoids from human lung tissue to human plasma in vitro. Eur Respir J 1994;7:382s.
    • (1994) Eur Respir J , vol.7
    • Högger, P.1    Bonsmann, U.2    Rohdewald, P.3
  • 14
    • 0027959815 scopus 로고
    • Binding kinetics of fluticasone propionate to the human glucocorticoid receptor
    • Högger P, Rohdewald P. Binding kinetics of fluticasone propionate to the human glucocorticoid receptor. Steroids 1994;59:597-602.
    • (1994) Steroids , vol.59 , pp. 597-602
    • Högger, P.1    Rohdewald, P.2
  • 15
    • 0025132348 scopus 로고
    • The human pharmacology of fluticasone propionate
    • Harding SM. The human pharmacology of fluticasone propionate. Respir Med 1990;84(suppl):25-9.
    • (1990) Respir Med , vol.84 , Issue.SUPPL. , pp. 25-29
    • Harding, S.M.1
  • 16
    • 33646405380 scopus 로고    scopus 로고
    • Ligand-induced differentiation of glucocorticoid receptor transrepression and transactivation
    • International Respiratory Forum. Reading UK: Colwood Publications
    • Adcock IM, Barnes PJ. Ligand-induced differentiation of glucocorticoid receptor transrepression and transactivation. In: Acute and chronic inflammation in the respiratory tract, International Respiratory Forum. Reading UK: Colwood Publications; 1996. p. 25.
    • (1996) Acute and Chronic Inflammation in the Respiratory Tract , pp. 25
    • Adcock, I.M.1    Barnes, P.J.2
  • 17
    • 33646421876 scopus 로고    scopus 로고
    • Effects of fluticasone propionate on random and stimulated T cell migration
    • International Respiratory Forum. Reading UK: Colwood Publications
    • Cruikshank W, Masterson J, Center D. Effects of fluticasone propionate on random and stimulated T cell migration. In: Acute and chronic inflammation in the respiratory tract, International Respiratory Forum. Reading UK: Colwood Publications; 1996. p. 19.
    • (1996) Acute and Chronic Inflammation in the Respiratory Tract , pp. 19
    • Cruikshank, W.1    Masterson, J.2    Center, D.3
  • 19
    • 0013612688 scopus 로고    scopus 로고
    • Effects of mometasone furoate and other glucocorticoids on cytokine production from cultured peripheral blood CD4+ T cells
    • Umland SP, Nahrebne MS, Razac S, Billah MM, Egan RW. Effects of mometasone furoate and other glucocorticoids on cytokine production from cultured peripheral blood CD4+ T cells. J Allergy Clin Immunol 1996;97:423.
    • (1996) J Allergy Clin Immunol , vol.97 , pp. 423
    • Umland, S.P.1    Nahrebne, M.S.2    Razac, S.3    Billah, M.M.4    Egan, R.W.5
  • 20
    • 4243312989 scopus 로고    scopus 로고
    • Comparison of the effect of inhaled glucocorticoids on human basophil histamine release and eosinophil viability
    • Bickel CA, Stellato C, Schleimer RP. Comparison of the effect of inhaled glucocorticoids on human basophil histamine release and eosinophil viability. J Allergy Clin Immunol 1997;99:1632.
    • (1997) J Allergy Clin Immunol , vol.99 , pp. 1632
    • Bickel, C.A.1    Stellato, C.2    Schleimer, R.P.3
  • 21
    • 0342486917 scopus 로고    scopus 로고
    • Fluticasone propionate is the most potent glucocorticoid in the induction of apoptosis of eosinophils
    • International Respiratory Forum. Reading UK: Colwood Publications
    • Kita H, Hagen JB, Gleich GJ. Fluticasone propionate is the most potent glucocorticoid in the induction of apoptosis of eosinophils. In: Acute and chronic inflammation in the respiratory tract, International Respiratory Forum. Reading UK: Colwood Publications; 1996. p. 17.
    • (1996) Acute and Chronic Inflammation in the Respiratory Tract , pp. 17
    • Kita, H.1    Hagen, J.B.2    Gleich, G.J.3
  • 22
    • 0029015546 scopus 로고
    • Anti-inflammatory properties of fluticasone propionate
    • Johnson M. Anti-inflammatory properties of fluticasone propionate. Int Arch Allergy Immunol 1995;107:439-40.
    • (1995) Int Arch Allergy Immunol , vol.107 , pp. 439-440
    • Johnson, M.1
  • 23
    • 33646410351 scopus 로고    scopus 로고
    • Effects of tumour necrosis factor-alpha on airway epithelial cells in vitro
    • International Respiratory Forum. Reading UK: Colwood Publications
    • Adler KB, Krunkosky TA, Fischer BM. Effects of tumour necrosis factor-alpha on airway epithelial cells in vitro. In: Acute and chronic inflammation in the respiratory tract, International Respiratory Forum. Reading UK: Colwood Publications; 1996. p. 18.
    • (1996) Acute and Chronic Inflammation in the Respiratory Tract , pp. 18
    • Adler, K.B.1    Krunkosky, T.A.2    Fischer, B.M.3
  • 24
    • 9044244752 scopus 로고
    • Corticosteroids increase secretory leukocyte protease inhibitor transcript levels in airway epithelial cells
    • Abbinante-Nissen JM, Simpson LG, Leikauf GD. Corticosteroids increase secretory leukocyte protease inhibitor transcript levels in airway epithelial cells. Am J Respir Crit Care Med 1994;149:A869.
    • (1994) Am J Respir Crit Care Med , vol.149
    • Abbinante-Nissen, J.M.1    Simpson, L.G.2    Leikauf, G.D.3
  • 25
    • 0021350520 scopus 로고
    • Correlation between chemical structure, receptor binding, and biological activity of some novel, highly active, 16α, 17α-acetyl-substituted glucocorticoids
    • Dahlberg E, Thalén A, Brattsand R, Gustafsson JA, Johansson U, Römpke K. Correlation between chemical structure, receptor binding, and biological activity of some novel, highly active, 16α, 17α-acetyl-substituted glucocorticoids. Mol Pharmacol 1983;25:70-8.
    • (1983) Mol Pharmacol , vol.25 , pp. 70-78
    • Dahlberg, E.1    Thalén, A.2    Brattsand, R.3    Gustafsson, J.A.4    Johansson, U.5    Römpke, K.6
  • 26
    • 4244119871 scopus 로고
    • Effect of fluticasone on airway inflammation as assessed by bronchoalveolar lavage (BAL)
    • Booth H, Gardiner PV, Ward C, Walls A, Hendrick DJ, Walters EH. Effect of fluticasone on airway inflammation as assessed by bronchoalveolar lavage (BAL). Eur Respir J 1993;6(suppl 17):584S.
    • (1993) Eur Respir J , vol.6 , Issue.17 SUPPL.
    • Booth, H.1    Gardiner, P.V.2    Ward, C.3    Walls, A.4    Hendrick, D.J.5    Walters, E.H.6
  • 28
    • 33646393737 scopus 로고    scopus 로고
    • Effect of therapy on matrix metallo-proteinase (MMP) activity in the broncho-alveolar lavage (BAL) of patients with mild asthma
    • In press
    • Warner JA, Shute JK, Howarth PH. Effect of therapy on matrix metallo-proteinase (MMP) activity in the broncho-alveolar lavage (BAL) of patients with mild asthma. Am J Resp Crit Care Med In press.
    • Am J Resp Crit Care Med
    • Warner, J.A.1    Shute, J.K.2    Howarth, P.H.3


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.