메뉴 건너뛰기




Volumn 123, Issue 6, 1998, Pages 1253-1259

SB-205384: A GABA(A) receptor modulator with novel mechanism of action that shows subunit selectivity

Author keywords

aminobutyric acid; GABA(A); SB 205384; Subunit; Xenopus oocytes

Indexed keywords

4 AMINO 5,6,7,8 TETRAHYDRO 7 HYDROXY 2 METHYLBENZO[B]THIENO[2,3 B]PYRIDINE 3 CARBOXYLIC ACID; 4 AMINOBUTYRIC ACID A RECEPTOR; 4 AMINOBUTYRIC ACID A RECEPTOR BLOCKING AGENT; RECEPTOR SUBUNIT; UNCLASSIFIED DRUG; ZOLPIDEM;

EID: 0031934847     PISSN: 00071188     EISSN: None     Source Type: Journal    
DOI: 10.1038/sj.bjp.0701721     Document Type: Article
Times cited : (19)

References (28)
  • 2
    • 6844260008 scopus 로고    scopus 로고
    • (1994). BTP receptor modulator of the GABA-A/chloride channel complex for prolonging the duration of the GABA induced membrane current. Intn. Patent No. WO 94/25027
    • BENHAM, C.D., MEADOWS, H.J., THOMAS, D.R & WOOD, M.D. (1994). BTP receptor modulator of the GABA-A/chloride channel complex for prolonging the duration of the GABA induced membrane current. Intn. Patent No. WO 94/25027.
    • Benham, C.D.1    Meadows, H.J.2    Thomas, D.R.3    Wood, M.D.4
  • 3
    • 0030004039 scopus 로고    scopus 로고
    • A receptor subunit (α1, α2, α3, α5, and β2+3) immunoreactivity in the medial prefrontal cortex of the rat
    • A receptor subunit (α1, α2, α3, α5, and β2+3) immunoreactivity in the medial prefrontal cortex of the rat. Neurosci. Lett., 210, 213-217.
    • (1996) Neurosci. Lett. , vol.210 , pp. 213-217
    • Dunn, E.1    Fritschy, J.-M.2    Carter, D.B.3    Merchant, K.M.4
  • 4
    • 0026648083 scopus 로고
    • Five subtypes of type A-aminobutyric acid receptors identified in neurons by double and triple immunofluorescence staining with subunit-specific antibodies
    • FRITSCHY, J.-M., BENKE, D., MERTENS, S., OERTEL, W.H., BACHI, T. & MOHLER, H. (1992). Five subtypes of type A-aminobutyric acid receptors identified in neurons by double and triple immunofluorescence staining with subunit-specific antibodies. Proc. Natl. Acad. Sci. U.S.A., 89, 6726-6730.
    • (1992) Proc. Natl. Acad. Sci. U.S.A. , vol.89 , pp. 6726-6730
    • Fritschy, J.-M.1    Benke, D.2    Mertens, S.3    Oertel, W.H.4    Bachi, T.5    Mohler, H.6
  • 6
    • 0027180684 scopus 로고
    • A-receptor subtypes: Differential association of the α1- and α3-subunits with serotonergic and GABAergic neurons
    • A-receptor subtypes: Differential association of the α1- and α3-subunits with serotonergic and GABAergic neurons. Neuroscience, 54, 881-892.
    • (1993) Neuroscience , vol.54 , pp. 881-892
    • Gao, B.1    Fritschy, J.-M.2    Benke, D.3    Mohler, H.4
  • 7
    • 0028983166 scopus 로고
    • A-receptor subtypes in cholinergic and parvalbumin-positive neurons of the rat and marmoset medial septum-diagonal band complex
    • A-receptor subtypes in cholinergic and parvalbumin-positive neurons of the rat and marmoset medial septum-diagonal band complex. Neuroscience, 65, 101-117.
    • (1995) Neuroscience , vol.65 , pp. 101-117
    • Gao, B.1    Hornung, J.-P.2    Fritschy, J.-M.3
  • 8
    • 0029416984 scopus 로고
    • A receptor gating kinetics on the α-subunit isoform: Implications for structure-function relations and synaptic transmission
    • A receptor gating kinetics on the α-subunit isoform: implications for structure-function relations and synaptic transmission. J. Physiol., 489, 529-543.
    • (1995) J. Physiol. , vol.489 , pp. 529-543
    • Gingrich, K.J.1    Roberts, W.A.2    Kass, R.S.3
  • 12
    • 0030610069 scopus 로고    scopus 로고
    • Effect of SB-205384 on the decay of GABA-activated chloride currents in granule cells cultured from rat cerebellum
    • MEADOWS, H.J., HARRIES, M.H., THOMPSON, M. & BENHAM, C.D. (1997). Effect of SB-205384 on the decay of GABA-activated chloride currents in granule cells cultured from rat cerebellum. Br. J. Pharmacol., 121, 1334-1338.
    • (1997) Br. J. Pharmacol. , vol.121 , pp. 1334-1338
    • Meadows, H.J.1    Harries, M.H.2    Thompson, M.3    Benham, C.D.4
  • 13
  • 14
    • 0025193448 scopus 로고
    • 5-subunit creates novel type II benzodiazepine receptor pharmacology
    • 5-subunit creates novel type II benzodiazepine receptor pharmacology. J. Neurochem., 54, 1802-1804.
    • (1990) J. Neurochem. , vol.54 , pp. 1802-1804
    • Pritchett, D.B.1    Seeburg, P.H.2
  • 17
    • 0028031943 scopus 로고
    • Functional diversity of GABA-activated Cl currents in purkinje versus granule neurons in rat cerebellar slices
    • PUIA, G., COSTA, E. & VICINI, S. (1994). Functional diversity of GABA-activated Cl currents in purkinje versus granule neurons in rat cerebellar slices. Neuron, 12, 117-126.
    • (1994) Neuron , vol.12 , pp. 117-126
    • Puia, G.1    Costa, E.2    Vicini, S.3
  • 20
    • 0029417325 scopus 로고
    • β-Carboline γ-aminobutyric acidA receptor inverse agonists modulate γ-aminobutyric acid via the loreclezole binding site as well as the benzodiazepine site
    • STEVENSON, A., WINGROVE, P.B., WHITING, P.J. & WAFFORD, K.A. (1995). β-Carboline γ-aminobutyric acidA receptor inverse agonists modulate γ-aminobutyric acid via the loreclezole binding site as well as the benzodiazepine site. Mol. Pharmacol., 48, 965-969.
    • (1995) Mol. Pharmacol. , vol.48 , pp. 965-969
    • Stevenson, A.1    Wingrove, P.B.2    Whiting, P.J.3    Wafford, K.A.4
  • 23
    • 0027328861 scopus 로고
    • Functional comparison of the role of γ subunits in recombinant human γ-aminobutyric acid A/benzodiazepine receptors
    • WAFFORD, K.A., BAIN, C.J., WHITING, P.J. & KEMP, J.A. (1993a). Functional comparison of the role of γ subunits in recombinant human γ-aminobutyric acid A/benzodiazepine receptors. Mol. Pharmacol.,44, 437-442.
    • (1993) Mol. Pharmacol. , vol.44 , pp. 437-442
    • Wafford, K.A.1    Bain, C.J.2    Whiting, P.J.3    Kemp, J.A.4
  • 24
    • 0027530534 scopus 로고
    • Differences in affinity and efficacy of benzodiazepine receptor ligands at recombinant γ-aminobutyric acid a receptor subtypes
    • WAFFORD, K.A., WHITING, P.J. & KEMP, J.A. (1993b). Differences in affinity and efficacy of benzodiazepine receptor ligands at recombinant γ-aminobutyric acid A receptor subtypes. Mol. Pharmacol., 43, 240-244.
    • (1993) Mol. Pharmacol. , vol.43 , pp. 240-244
    • Wafford, K.A.1    Whiting, P.J.2    Kemp, J.A.3
  • 27
    • 0026612363 scopus 로고
    • A receptor subunit mRNAs in the rat brain. I. Telencephalon, Diencephalon, Mesencephalon
    • A receptor subunit mRNAs in the rat brain. I. Telencephalon, Diencephalon, Mesencephalon. J. Neurosci., 12, 1040-1062.
    • (1992) J. Neurosci. , vol.12 , pp. 1040-1062
    • Wisden, W.1    Laurie, D.J.2    Monyer, H.3    Seeburg, P.H.4


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.