Synthesis of cotinine and cotinine N-oxide: Evaluation of their interaction with nicotine in the insecticidal activity

Natural Product Letters

Volumn 11, Issue 1, 1997, Pages 37-45

  Riah, Omar ^a,b   Dousset, Jean Claude ^a   Courriere, Philippe ^a   Baziard Mouysset, Geneviève ^a   Ecalle, René ^a  

^a UNIVERSITÉ DE TOULOUSE   (France)

^b FACULTÉ DES SCIENCES   (Morocco)

Author keywords

Analysis of interactions; Flies; Insecticidal activity; Nicotine derivatives synthesis; Nicotinic acetylcholine receptors

Indexed keywords

COTININE; INSECTICIDE; NICOTINE DERIVATIVE; NORNICOTINE;

ARTICLE; FLY;

EID: 0031929445     PISSN: 10575634     EISSN: None     Source Type: Journal    
DOI: 10.1080/10575639708043755     Document Type: Article

References (19)

1. E. R. Bowman, H. McKennis, (1963) (-)cotinine. Biochem. Prep., 10, 36-39.
2. 3 in the mouse. J. Pharmacol. Exp. Ther., 143, 301-308.
3. 14C in tissues of the mouse. Drug Metab. Dispos., 4, 530-539.
4. J. Rosenberg, N. L. Benowitz, P. Jacob III, K. M. Wilson (1980) Disposition kinetics and effects of intravenous nicotine. Clin. Pharmacol. Ther., 28, 517-522.
5. D. Bruniquel, J. C. Dousset, R. Ecalle, Ph. Courrière, I. Fourasté (1992) Synergy between nicotine and cotinine in their insecticidal activity. Med. Sci. Res., 20, 869-870.
6. F. M. Wadley (1945) The evidence required to show synergistic action of insecticides and a short cut in analysis. U.S. Dept. Agric. E.T. p. 223.
7. G. G. Steel, M. J. Peckham (1979) Exploitable mechanisms in combined radiotherapy-chimiotherapy : The concept of additivity. Rad. Oncol. Biol. Phys., 15, 85-91.
8. E.D. Gundelfinger, N. Hess (1992) Nicotinic acetylcholine receptor of the central nervous system of Drosophila. B. B. A., 1137, 299-308.
9. E. L. M. Ochoa (1994) Nicotine-related brain disorders : The neurobiology basis of nicotine dependence. Cel. Mol. Neurobiol., 14, 195-225.
10. S. R. Goldberg, M. E. Risner, I. P. Stolerman, C. Reavill, H. S. Garcha (1989) Nicotine and some related compounds : effects on schedule-controlled behavior and discriminative properties in the rat. Psychopharmacology, 97, 295-302.
11. E. Dagne, N. Castangoli, (1972) J. Med. Chem., 15 (8), 840-841.
12. T. Stalhandske (1969) The metabolism of nicotine and cotinine by a mouse liver preparation. Acta Physiol. Scand., 78, 236-248.
13. M. Hariharan, T. VanNoord, J. Greden (1988) A high performance liquid chromatographic method for routine simultaneous determination of nicotine and cotinine in plasma. Clin. Chem., 34, 724-729.
14. R. Chahine (1989) Recherche toxicologique et pharmacologique sur les effets de la métabolisation de la nicotine. Ph. D. Thesis, Paul-Sabatier University, TOU III, France.
15. I. Yamamoto, G. Yabuta, M. Tomizawa, T. Saito, T. Miyamoto, S. Kagabu (1995) Molecular mechanism for selective toxicity of nicotinoids and neonicotinoids. Nippond Noyaku Gakkaishi, 20, 33-40.
16. M. E. Risner, E. J. Cone, N. L. Benowitz, P. Jacob III (1988) Effects of the stereoisomers of nicotine and nomicotine on schedule-controlled responding and physiological parameters of dogs. J. Pharmacol. Exp. Ther., 244, 3, 807-813.
17. M. E. Risner, S. R. Goldberg, J. A. Prada, E. J. Cone (1985) Effects of nicotine, cocaine and some of their metabolites on schedule-controlled responding by beagle dogs and squirrel monkeys. J. Pharmacol. Exp. Ther., 234, 113-119.
18. R. J. Leatherbarrow (1987) ENZFITTER : a non-linearly regression data analysis program for the IBM PC (and true compatibles). Elsevier Science Publishers BV PO Box 1527 1000 BM, Amsterdam.
19. D. Schwartz (1994) Statistique en Biologie et en Médecine. Médecine-Sciences Flammarion Eds. pp. 290-291. Paris.