Chemistry of α-fluoro-α-amino acids: The first synthesis of α- fluoroglycine-containing dipeptides

Chemical and Pharmaceutical Bulletin

Volumn 46, Issue 6, 1998, Pages 1062-1064

  Takeuchi, Yoshio ^a,b   Kamezaki, Makoto ^a,b   Kirihara, Kiyotoshi ^a,b   Haufe, Günter ^a,b   Laue, Klaus W ^a,b   Shibata, Norio ^a,b  

^a UNIVERSITY OF TOYAMA   (Japan)

^b UNIVERSITY OF MÜNSTER   (Germany)

Author keywords

Fluorinated peptide; Gabriel reaction; Ruthenium tetroxide oxidation; fluoro amino acid

Indexed keywords

ALPHA FLUORO ALPHA AMINO ACID; ALPHA FLUOROGLYCINE; AMINO ACID DERIVATIVE; DIPEPTIDE; FLUORINE DERIVATIVE; RUTHENIUM; UNCLASSIFIED DRUG;

ARTICLE; CHEMICAL REACTION; FLUORINATION; PEPTIDE SYNTHESIS; PROTEIN MODIFICATION; PROTEIN STABILITY;

EID: 0031928003     PISSN: 00092363     EISSN: None     Source Type: Journal    
DOI: 10.1248/cpb.46.1062     Document Type: Article

References (6)

1. Takeuchi Y., Asahina M., Murayama A., Hori K., Koizumi T., J. Org. Chem., 51, 955-956 (1986);
2. Takeuchi Y., Yuki Gousei Kagaku Kyokai-shi, 55, 886-896 (1997).
3. Kukhar' V.P., Soloshonok V.A. (Eds.), "Fluorine-containing Amino Acids," John Wiley & Sons Ltd., West Sussex, England, 1995.
4. German L., Zemskov S. (Eds.), "New Fluorinating Agents in Organic Synthesis," Springer-Verlag, Berlin, 1989.
5. Zoller U., Ben-Ishai D., Tetrahedron, 31, 863-866 (1975);
6. Easton C.J., Chem. Rev., 97, 53-82 (1997).