Human progesterone receptor A and B isoforms in CHO cells. II. Comparison of binding, transactivation and ED50 values of several synthetic (anti)progestagens in vitro in CHO and MCF-7 cells and in vivo in rabbits and rats

Journal of Steroid Biochemistry and Molecular Biology

Volumn 64, Issue 3-4, 1998, Pages 157-170

  Schoonen, W G E J ^a   Dijkema, R ^a   De Ries, R J H ^a   Wagenaars, J L ^a   Joosten, J W H ^a   De Gooyer, M E ^a   Deckers, G H ^a   Kloosterboer, H J ^a  

^a Sci Devmt Grp N V Organon P   (Netherlands)

Author keywords

[No Author keywords available]

Indexed keywords

11BETA (4 ACETYLPHENYL) 17BETA HYDROXY 17ALPHA (1 PROPYNYL)ESTRA 4,9 DIEN 3 ONE; 11BETA [4 (DIMETHYLAMINO)PHENYL] 4',5' DIHYDRO 6BETA METHYLSPIRO[ESTRA 4,9 DIENE 17BETA,2'(3'H) FURAN] 3 ONE; 16ALPHA ETHYL 21 HYDROXY 19 NORPREGN 4 ENE 3,20 DIONE; 17ALPHA HYDROXY 11 METHYLENE 19 NORPREGNA 4,15 DIEN 20 YN 3 ONE; ANTIGESTAGEN; ETONOGESTREL; GESTAGEN; GESTODENE; LEVONORGESTREL; MIFEPRISTONE; NORETHISTERONE; ONAPRISTONE; ORG 2761; ORG 30943; ORG 31042; ORG 31806; ORG 32704; ORG 32985; ORG 33245; ORG 33628; ORG 33766; PROGESTERONE; PROGESTERONE RECEPTOR; PROMEGESTONE; RECEPTOR SUBTYPE; UNCLASSIFIED DRUG; VIRUS VECTOR;

ANIMAL CELL; ANIMAL EXPERIMENT; ARTICLE; BINDING AFFINITY; BREAST TUMOR; CELL LINE; CHO CELL; CONTROLLED STUDY; FEMALE; GENETIC TRANSFECTION; HORMONE RECEPTOR INTERACTION; HUMAN; HUMAN CELL; IN VITRO STUDY; INDUCED ABORTION; NONHUMAN; OVULATION INHIBITION; PROTEIN EXPRESSION; RABBIT; RAT; REPORTER GENE; SUBCUTANEOUS DRUG ADMINISTRATION; TRANSACTIVATION;

ANIMALIA; CRICETINAE; CRICETULUS GRISEUS; EUKARYOTA; MINK CELL FOCUS-FORMING VIRUS; MOUSE MAMMARY TUMOR VIRUS; ORYCTOLAGUS CUNICULUS; TUMOR VIRUS;

EID: 0031916316     PISSN: 09600760     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0960-0760(97)00161-1     Document Type: Article

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