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Volumn 284, Issue 2, 1998, Pages 661-668

Stereoselective hepatobiliary transport of the quinolone antibiotic grepafloxacin and its glucuronide in the rat

Author keywords

[No Author keywords available]

Indexed keywords

GREPAFLOXACIN; QUINOLINE DERIVED ANTIINFECTIVE AGENT;

EID: 0031884441     PISSN: 00223565     EISSN: None     Source Type: Journal    
DOI: None     Document Type: Article
Times cited : (17)

References (39)
  • 1
    • 0029094613 scopus 로고
    • Pharmacokinetics of grepafloxacin (IV): Metabolism after oral administration of grepafloxacin in rats, monkeys and humans
    • Akiyama H, Koike M, Kyuushiki K, Suzuki T, Kusumoto N, Morita S and Odomi M (1995) Pharmacokinetics of grepafloxacin (IV): Metabolism after oral administration of grepafloxacin in rats, monkeys and humans. Chemotherapy 43(S-1): 131-149.
    • (1995) Chemotherapy , vol.43 , Issue.S-1 , pp. 131-149
    • Akiyama, H.1    Koike, M.2    Kyuushiki, K.3    Suzuki, T.4    Kusumoto, N.5    Morita, S.6    Odomi, M.7
  • 3
    • 0028284238 scopus 로고
    • Cholestasis caused by inhibition of the adenosine triphosphate-dependent bile salt transport in rat liver
    • Bohme M, Muller M, Leier I, Jedlitschky G and Keppler D (1994) Cholestasis caused by inhibition of the adenosine triphosphate-dependent bile salt transport in rat liver. Gastroenterology 107:255-265.
    • (1994) Gastroenterology , vol.107 , pp. 255-265
    • Bohme, M.1    Muller, M.2    Leier, I.3    Jedlitschky, G.4    Keppler, D.5
  • 4
    • 0017184389 scopus 로고
    • A rapid and sensitive method for the quantitation of microgram quantities of protein utilizing the principle of protein-dye binding
    • Bradford MM (1976) A rapid and sensitive method for the quantitation of microgram quantities of protein utilizing the principle of protein-dye binding. Anal Biochem 72:248-254.
    • (1976) Anal Biochem , vol.72 , pp. 248-254
    • Bradford, M.M.1
  • 5
    • 0030959378 scopus 로고    scopus 로고
    • Multi-specific organic anion transporter is responsible for the biliary excretion of the camptothecin derivative irinotecan and its metabolites in rats
    • Chu XY, Kato Y, Niinuma K, Sudo K, Hakusui H and Sugiyama Y (1997a) Multi-specific organic anion transporter is responsible for the biliary excretion of the camptothecin derivative irinotecan and its metabolites in rats. J Pharmacol Exp Ther 281:304-314.
    • (1997) J Pharmacol Exp Ther , vol.281 , pp. 304-314
    • Chu, X.Y.1    Kato, Y.2    Niinuma, K.3    Sudo, K.4    Hakusui, H.5    Sugiyama, Y.6
  • 6
    • 0030906434 scopus 로고    scopus 로고
    • Multiplicity of biliary excretion mechanisms for irinotechan, CPT-11 and its metabolites in rats
    • Chu XY, Kato Y and Sugiyama Y (1997b) Multiplicity of biliary excretion mechanisms for irinotechan, CPT-11 and its metabolites in rats. Cancer Res 57:1934-1938.
    • (1997) Cancer Res , vol.57 , pp. 1934-1938
    • Chu, X.Y.1    Kato, Y.2    Sugiyama, Y.3
  • 8
    • 0026511550 scopus 로고
    • Canalicular transport of reduced glutathione in normal and mutant eisai hyperbilirubinemic rats
    • Fernandez-Checa JC, Takikawa H, Horie T, Ookhtens M and Kaplowitz N (1992) Canalicular transport of reduced glutathione in normal and mutant eisai hyperbilirubinemic rats. J Biol Chem 267:1667-1673.
    • (1992) J Biol Chem , vol.267 , pp. 1667-1673
    • Fernandez-Checa, J.C.1    Takikawa, H.2    Horie, T.3    Ookhtens, M.4    Kaplowitz, N.5
  • 9
    • 0026749343 scopus 로고
    • Stereoselective disposition and tissue distribution of carvedilol enantiomers in rats
    • Fujimaki M (1992) Stereoselective disposition and tissue distribution of carvedilol enantiomers in rats. Chirality 4:148-154.
    • (1992) Chirality , vol.4 , pp. 148-154
    • Fujimaki, M.1
  • 10
    • 15444339505 scopus 로고    scopus 로고
    • Characterization of ATP-dependent organic anion transport system on rat canalicular membrane maintained in EHBR
    • Hirohashi T, Niinuma K, Ito K, Suzuki H, Kume K, Shimizu T and Sugiyama Y (1996) Characterization of ATP-dependent organic anion transport system on rat canalicular membrane maintained in EHBR. Hepatology 24:203A.
    • (1996) Hepatology , vol.24
    • Hirohashi, T.1    Niinuma, K.2    Ito, K.3    Suzuki, H.4    Kume, K.5    Shimizu, T.6    Sugiyama, Y.7
  • 11
    • 0025132673 scopus 로고
    • ATP-dependent primary active transport of cysteinyl leukotrienes across liver canalicular membrane
    • Ishikawa T, Müller M, Klünemann C, Schaub T and Keppler D (1990) ATP-dependent primary active transport of cysteinyl leukotrienes across liver canalicular membrane. J Biol Chem 265:19279-19286.
    • (1990) J Biol Chem , vol.265 , pp. 19279-19286
    • Ishikawa, T.1    Müller, M.2    Klünemann, C.3    Schaub, T.4    Keppler, D.5
  • 12
    • 0025320414 scopus 로고
    • Transport of leucine, isoleucine and valine by luminal membrane vesicles from rabbit proximal tubule
    • Jorgensen KE, Kragh-hansen U and Sheikh MI (1990) Transport of leucine, isoleucine and valine by luminal membrane vesicles from rabbit proximal tubule. J Physiol 422:41-54.
    • (1990) J Physiol , vol.422 , pp. 41-54
    • Jorgensen, K.E.1    Kragh-hansen, U.2    Sheikh, M.I.3
  • 13
    • 0030638506 scopus 로고    scopus 로고
    • Hepatic canalicular membrane. Introduction: Transport across the hepatocyte canalicular membrane
    • Keppler D and Arias IM (1997) Hepatic canalicular membrane. Introduction: Transport across the hepatocyte canalicular membrane. FASEB J 11:15-18.
    • (1997) FASEB J , vol.11 , pp. 15-18
    • Keppler, D.1    Arias, I.M.2
  • 14
    • 0025803058 scopus 로고
    • ATP-dependent transport for glucuronides in canalicular plasma membrane vesicles
    • Kobayashi K, Komatsu S, Nishii T, Hara H and Hayashi K (1991) ATP-dependent transport for glucuronides in canalicular plasma membrane vesicles. Biochem Biophys Res Com 176:622-626.
    • (1991) Biochem Biophys Res Com , vol.176 , pp. 622-626
    • Kobayashi, K.1    Komatsu, S.2    Nishii, T.3    Hara, H.4    Hayashi, K.5
  • 15
    • 0025343017 scopus 로고
    • Mechanism of glutathione S-conjugate transport in canalicular and basolateral rat liver plasma membranes
    • Kobayashi K, Sogame Y, Hara H and Hayashi K (1990) Mechanism of glutathione S-conjugate transport in canalicular and basolateral rat liver plasma membranes. J Biol Chem 263:7737-7741.
    • (1990) J Biol Chem , vol.263 , pp. 7737-7741
    • Kobayashi, K.1    Sogame, Y.2    Hara, H.3    Hayashi, K.4
  • 16
    • 0026601365 scopus 로고
    • Intestinal absorption of β-lactam antibiotics and ologopeptides: Functional and stereospecific reconstitution of the oligopeptide transport system from rabbit small intestine
    • Kramer W, Girbig F, Gutjahr U, Kowalewski S, Adam F and Schiebler W (1992) Intestinal absorption of β-lactam antibiotics and ologopeptides: Functional and stereospecific reconstitution of the oligopeptide transport system from rabbit small intestine. Eur J Biochem 204:923-930.
    • (1992) Eur J Biochem , vol.204 , pp. 923-930
    • Kramer, W.1    Girbig, F.2    Gutjahr, U.3    Kowalewski, S.4    Adam, F.5    Schiebler, W.6
  • 17
    • 0021349075 scopus 로고
    • Structural and functional polarity of canalicular and basolateral plasma membrane vesicles isolated in high yield from rat liver
    • Meier PJ, Sztul ES, Reuben A and Boyer JL (1984) Structural and functional polarity of canalicular and basolateral plasma membrane vesicles isolated in high yield from rat liver. J Cell Biology 98:991-1000.
    • (1984) J Cell Biology , vol.98 , pp. 991-1000
    • Meier, P.J.1    Sztul, E.S.2    Reuben, A.3    Boyer, J.L.4
  • 18
    • 0022330348 scopus 로고
    • Assay of mephenytoin metabolism in human liver microsomes by high-performance liquid chromatography
    • Meier UT, Kronbach T and Meyer UA (1985) Assay of mephenytoin metabolism in human liver microsomes by high-performance liquid chromatography. Anal Biolchem 151:286-291.
    • (1985) Anal Biolchem , vol.151 , pp. 286-291
    • Meier, U.T.1    Kronbach, T.2    Meyer, U.A.3
  • 20
    • 0030818770 scopus 로고    scopus 로고
    • Kinetic analysis of the primary active transport of conjugated metabolites across the bile canalicular membrane: Comparative study of S-(2,4-dinitrophenyl)-glutathione and 4-(3-pyridylmethyl) benzothiazole glucuronide
    • Niinuma K, Takenaka O, Horie T, Kobayashi K, Kato Y, Suzuki H and Sugiyama Y (1997) Kinetic analysis of the primary active transport of conjugated metabolites across the bile canalicular membrane: Comparative study of S-(2,4-dinitrophenyl)-glutathione and 4-(3-pyridylmethyl) benzothiazole glucuronide. J Pharmacol Exp Ther 282:866-872.
    • (1997) J Pharmacol Exp Ther , vol.282 , pp. 866-872
    • Niinuma, K.1    Takenaka, O.2    Horie, T.3    Kobayashi, K.4    Kato, Y.5    Suzuki, H.6    Sugiyama, Y.7
  • 21
    • 0030444801 scopus 로고    scopus 로고
    • Stereoselective and carrier-mediated transport of monocarboxylic acids across Caco-2 cells
    • Ogihara T, Tamai I, Takanaga H, Sai Y and Tsuji A (1996) Stereoselective and carrier-mediated transport of monocarboxylic acids across Caco-2 cells. Pharm Res 13:1828-1832.
    • (1996) Pharm Res , vol.13 , pp. 1828-1832
    • Ogihara, T.1    Tamai, I.2    Takanaga, H.3    Sai, Y.4    Tsuji, A.5
  • 22
    • 0025973006 scopus 로고
    • Stereoselective glucuronide of ofloxacin in rat liver microsomes
    • Okazaki O, Kurata T, Hakusui H and Tachizawa H (1991) Stereoselective glucuronide of ofloxacin in rat liver microsomes. Drug Metab Dispos 19:376-380.
    • (1991) Drug Metab Dispos , vol.19 , pp. 376-380
    • Okazaki, O.1    Kurata, T.2    Hakusui, H.3    Tachizawa, H.4
  • 23
    • 0024522834 scopus 로고
    • Stereoselective metabolic disposition of enantiomers of ofloxacin in rats
    • Okazaki O, Kurata T and Tachizawa H (1989) Stereoselective metabolic disposition of enantiomers of ofloxacin in rats. Xenobiotica 19:419-429.
    • (1989) Xenobiotica , vol.19 , pp. 419-429
    • Okazaki, O.1    Kurata, T.2    Tachizawa, H.3
  • 24
    • 0027138659 scopus 로고
    • Stereoselective sulfate conjugation of isoproterenol in humans: Comparison of hepatic, intestinal, and platelet activity
    • Pesola GR and Walle T (1993) Stereoselective sulfate conjugation of isoproterenol in humans: Comparison of hepatic, intestinal, and platelet activity. Chirality 5:602-609.
    • (1993) Chirality , vol.5 , pp. 602-609
    • Pesola, G.R.1    Walle, T.2
  • 25
    • 0030824648 scopus 로고    scopus 로고
    • Carrier-mediated hepatic uptake of quinolone antibiotics in the rat
    • Sasabe H, Terasaki T, Tsuji A and Sugiyama Y (1997) Carrier-mediated hepatic uptake of quinolone antibiotics in the rat. J Pharmacol Exp Ther 282:162-171.
    • (1997) J Pharmacol Exp Ther , vol.282 , pp. 162-171
    • Sasabe, H.1    Terasaki, T.2    Tsuji, A.3    Sugiyama, Y.4
  • 26
  • 28
    • 0018901053 scopus 로고
    • Transport systems of isolated hepatocytes: Studies on the transport of biliary compounds
    • Schwenk M (1980) Transport systems of isolated hepatocytes: Studies on the transport of biliary compounds. Arch Toxicol 44:113-126.
    • (1980) Arch Toxicol , vol.44 , pp. 113-126
    • Schwenk, M.1
  • 30
    • 0025158275 scopus 로고
    • Carrier-mediated uptake of nicotinic acid by rat intestinal brush-border membrane vesicles and relation to monocarboxylic acid transport
    • Simanjuntak MT, Tamai I, Terasaki T and Tsuji A (1990) Carrier-mediated uptake of nicotinic acid by rat intestinal brush-border membrane vesicles and relation to monocarboxylic acid transport. J Pharmacobio-Dyn 13:301-309.
    • (1990) J Pharmacobio-Dyn , vol.13 , pp. 301-309
    • Simanjuntak, M.T.1    Tamai, I.2    Terasaki, T.3    Tsuji, A.4
  • 31
    • 0029582975 scopus 로고
    • Kinetic analysis of hepatobiliary transport for conjugative metabolites in the perfused liver of mutant rats (EHBR) with hereditary conjugative hyperbilirubinemia
    • Takenaka O, Horie T, Suzuki H, Kobayashi K and Sugiyama Y (1995a) Kinetic analysis of hepatobiliary transport for conjugative metabolites in the perfused liver of mutant rats (EHBR) with hereditary conjugative hyperbilirubinemia. Pharm Res 12:1746-1755.
    • (1995) Pharm Res , vol.12 , pp. 1746-1755
    • Takenaka, O.1    Horie, T.2    Suzuki, H.3    Kobayashi, K.4    Sugiyama, Y.5
  • 32
    • 0029026940 scopus 로고
    • Different biliary excretion systems for glucuronide and sulfate of a model compound: Study using Eisai Hyperbilirubinemic rats
    • Takenaka O, Horie T, Suzuki H and Sugiyama Y (1995b) Different biliary excretion systems for glucuronide and sulfate of a model compound: Study using Eisai Hyperbilirubinemic rats. J Pharmacol Exp Ther 274:1362-1369.
    • (1995) J Pharmacol Exp Ther , vol.274 , pp. 1362-1369
    • Takenaka, O.1    Horie, T.2    Suzuki, H.3    Sugiyama, Y.4
  • 34
    • 0027416040 scopus 로고
    • Stereoselective sulfation of albuterol in humans: Biosynthesis of the sulfate conjugate by HEP G2 cells
    • Walle T, Walle UK, Thornburg KR and Schey KL (1993) Stereoselective sulfation of albuterol in humans: Biosynthesis of the sulfate conjugate by HEP G2 cells. Drug Metab and Dispos 21:76-80.
    • (1993) Drug Metab and Dispos , vol.21 , pp. 76-80
    • Walle, T.1    Walle, U.K.2    Thornburg, K.R.3    Schey, K.L.4
  • 36
    • 0024492557 scopus 로고
    • Characterization of rose Bengal binding to sinusoidal and bile canalicular plasma membrane from rat liver
    • Yachi K, Sugiyama Y, Sawada Y, Iga T, Ikeda Y, Toda G and Hanano M (1989) Characterization of rose Bengal binding to sinusoidal and bile canalicular plasma membrane from rat liver. Biochim Biophys Acta 978:1-7.
    • (1989) Biochim Biophys Acta , vol.978 , pp. 1-7
    • Yachi, K.1    Sugiyama, Y.2    Sawada, Y.3    Iga, T.4    Ikeda, Y.5    Toda, G.6    Hanano, M.7
  • 37
    • 0019854279 scopus 로고
    • A pharmacokinetic analysis program (MULTI) for microcomputer
    • Yamaoka K, Tanigawara Y, Nakagami Y and Uno T (1981) A pharmacokinetic analysis program (MULTI) for microcomputer. J Pharmacobio-Dyn 4:879-885.
    • (1981) J Pharmacobio-Dyn , vol.4 , pp. 879-885
    • Yamaoka, K.1    Tanigawara, Y.2    Nakagami, Y.3    Uno, T.4
  • 38
    • 0029926676 scopus 로고    scopus 로고
    • Recent advances in carrier-mediated hepatic uptake and biliary excretion of xenobiotics
    • Yamazaki M, Suzuki H, Hanano M, Tokui T, Komai T and Sugiyama Y (1996) Recent advances in carrier-mediated hepatic uptake and biliary excretion of xenobiotics. Pharm Res 13:497-513.
    • (1996) Pharm Res , vol.13 , pp. 497-513
    • Yamazaki, M.1    Suzuki, H.2    Hanano, M.3    Tokui, T.4    Komai, T.5    Sugiyama, Y.6
  • 39
    • 0024307467 scopus 로고
    • Transport characteristics of ceftibuten (7432-S), a new oral cephem, in rat intestinal brush-border membrane vesicle: Proton-coupled and Stereoselective transport of ceftibuten
    • Yoshikawa T, Muranishi N, Yoshida M, Oguma T, Hirano K and Yamada H (1989) Transport characteristics of ceftibuten (7432-S), a new oral cephem, in rat intestinal brush-border membrane vesicle: Proton-coupled and Stereoselective transport of ceftibuten. Pharm Res 6:302-307.
    • (1989) Pharm Res , vol.6 , pp. 302-307
    • Yoshikawa, T.1    Muranishi, N.2    Yoshida, M.3    Oguma, T.4    Hirano, K.5    Yamada, H.6


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