The relationship between the agonist-induced activation and desensitization of the human tachykinin NK2 receptor expressed in Xenopus oocytes

British Journal of Pharmacology

Volumn 124, Issue 4, 1998, Pages 675-684

  Maudsley, S ^a,b   Gent, J P ^a   Findlay, J B C ^a   Donnelly, D ^a  

^a UNIVERSITY OF LEEDS   (United Kingdom)

^b DUKE UNIVERSITY MEDICAL CENTER   (United States)

Author keywords

Agonist induced desensitization; Efficacy; Neurokinin; NKA; Tachykinin; Xenopus oocyte expression

Indexed keywords

9 (TETRAHYDRO 2 FURYL)ADENINE; NEUROKININ 2 RECEPTOR; NEUROKININ A; NEUROKININ A [3-10][3 LYSINE 8 GLYCINE GAMMA LACTAM 9 LEUCINE]; NEUROKININ A [4-10];

ANIMAL CELL; ARTICLE; CHLORIDE CURRENT; DESENSITIZATION; FEMALE; NONHUMAN; OOCYTE; PRIORITY JOURNAL; XENOPUS;

ADENYLATE CYCLASE; ANIMALS; CALCIUM; CHLORIDE CHANNELS; CYCLIC AMP-DEPENDENT PROTEIN KINASES; ENZYME INHIBITORS; FEMALE; HUMANS; NEUROKININ A; OOCYTES; PATCH-CLAMP TECHNIQUES; PEPTIDE FRAGMENTS; RECEPTORS, NEUROKININ-2; SIGNAL TRANSDUCTION; XENOPUS LAEVIS;

EID: 0031835335     PISSN: 00071188     EISSN: None     Source Type: Journal    
DOI: 10.1038/sj.bjp.0701889     Document Type: Article

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