Synthesis and biological evaluation of cyclopropyl analogs of the antiestrogen MER 25

Bioorganic Chemistry

Volumn 26, Issue 1, 1998, Pages 15-31

  Overacre, Lynette B ^a   Magarian, Robert A ^a  

^a UNIVERSITY OF OKLAHOMA HEALTH SCIENCES CENTER   (United States)

Author keywords

Antiestrogen; Biological evaluation; Breast cancer; Gem dichlorocyclopropanes; MCF 7E3; MDA MB 231; Synthesis

Indexed keywords

ANTIESTROGEN; ESTROGEN RECEPTOR; ETHAMOXYTRIPHETOL; ETHAMOXYTRIPHETOL DERIVATIVE; FULVESTRANT; TAMOXIFEN; UNCLASSIFIED DRUG;

ANTINEOPLASTIC ACTIVITY; ARTICLE; CANCER CELL CULTURE; CELL STRAIN MCF 7; CONCENTRATION RESPONSE; CONTROLLED STUDY; DRUG SYNTHESIS; HUMAN; HUMAN CELL; PRIORITY JOURNAL; STRUCTURE ACTIVITY RELATION;

EID: 0031831058     PISSN: 00452068     EISSN: None     Source Type: Journal    
DOI: 10.1006/bioo.1998.1081     Document Type: Article

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