Theophylline derivatives as potential histamine H3-receptor antagonists

Pharmazie

Volumn 53, Issue 8, 1998, Pages 518-521

  Kiec Kononowicz K ^a   CegLa M T ^a  

^a JAGIELLONIAN UNIVERSITY MEDICAL COLLEGE   (Poland)

Author keywords

[No Author keywords available]

Indexed keywords

AMIDE; AMINE; ESTER; HISTAMINE H3 RECEPTOR; HISTAMINE H3 RECEPTOR ANTAGONIST; RECEPTOR SUBTYPE; THEOPHYLLINE DERIVATIVE; THIOUREA;

ANIMAL TISSUE; ARTICLE; BINDING AFFINITY; DRUG ACTIVITY; DRUG POTENCY; DRUG RECEPTOR BINDING; GUINEA PIG; ILEUM; LIPOPHILICITY; NONHUMAN;

ANIMALS; GUINEA PIGS; HISTAMINE ANTAGONISTS; ILEUM; MUSCLE CONTRACTION; MUSCLE, SMOOTH; RECEPTORS, HISTAMINE H3; THEOPHYLLINE;

EID: 0031815195     PISSN: 00317144     EISSN: None     Source Type: Journal    
DOI: None     Document Type: Article

References (21)

1. Arrang, J.-M.; Garbarg, M.; Schwartz, J.-C.: Nature (London) 302, 832 (1983)
2. Schwartz, J.-C.; Arrang, J.-M.; Garbarg, M.; Pollard, H.: Agents Actions 30, 13 (1990)
3. Stark, H.; Schlicker, E.; Schunack, W.: Drugs Future 21, 507 (1996)
4. Leurs, P.; Voilinga, R. C.; Timmermann, H.: Prog. Drug Res. 45, 107 (1995)
5. Pascal, J.-C.; Beranger, S.; Pinhas, H.; Poizot, A.; Desiles, J. -P.: J. Med. Chem. 28, 647 (1985)
6. Poizot, A.; Dumez, D.; Ferrandon, P.; Lefournier, C.; Michel, A.; Armstrong, J. M.: Arzneim.-Forsch./Drug Res. 36, 695 (1986)
7. Abou-Gharbia, M.; Moyer, J. A.; Nielsen, S. T.; Webb, M.; Patel, U.: J. Med. Chem. 38, 4026 (1995)
8. Lipp, R.; Stark, H.; Schunack, W.; in: Schwartz, J.-C.; Haas, H. L. (Eds.): The Histamine Receptor, Ser.: Receptor Biochemistry and Methodology, Wiley-Liss, New York 16, 57 (1992)
9. Kamiński, Z.: Synthesis 917 (1987)
10. Ono, N.; Yamada, T.; Saito, T.; Tanaka, K.; Kaji, A.: Bull. Chem. Soc. Jpn. 51, 2401 (1978)
11. Hüls, A.; Purand, K.; Stark, H.; Reidemeister, S.; Ligneau, X.; Arrang, J.-M.; Schwartz, J.-C.; Schunack, W.: Arch. Pharm. Pharm. Med. Chem. 329, 379 (1996)
12. van Rossum, J. M.: Arch. Int. Pharmacodyn. Ther. 143, 299 (1963)
13. Schlicker, E.; Kathmann, M.; Reidemeister, S.; Stark, H.; Schunack, W.: Br. J Pharmacol. 112, 1043 (1994) - Erratum 113, 657 (1994)
14. Stark, H.; Lipp, R.; Arrang, J.-M.; Garbarg, M.; Schwartz, J.-C.; Schunack, W.: Eur. J. Med. Chem. 29, 695 (1994)
15. Stark, H.; Hüls, A.; Ligneau, X.; Arrang, J.-M.; Schwartz, J.-C.; Schunack, W.: Pharmazie 52, 495 (1997)
16. Zelnik, R.; Pesson, M.: Bull. Soc. Chim. 1667 (1959)
17. Eckstein, M.; Drabczyńska, A.: Przegl. Metodyczny 6, 41 (1971)
18. Eckstein, M.; Zajaczkowska, J.: Dissertationes Pharm. 14, 41 (1962)
19. Eckstein, M.; Jakubowski, K.: Dissertationes Pharm. 16, 35 (1964)
20. Ligneau, X.; Garbarg, M.; Vizuete, M. L.; Diaz, J.; Purand, K.; Stark, H.; Schunack, W.; Schwartz, J.-C.: J. Pharmacol. Exp. Ther. 271, 452 (1994)
21. Lennartz, H. G.; Hepp, M.; Schunack, W.: Eur. J. Med. Chem. Chim. Ther. 13, 229 (1978)