Quantitative structure-activity relationship studies on some nonbenzodiazepine series of compounds acting at the benzodiazepine receptor

Bioorganic and Medicinal Chemistry

Volumn 6, Issue 11, 1998, Pages 2213-2218

  Gupta, S P ^a   Paleti, Anitha ^a  

^a BIRLA INSTITUTE OF TECHNOLOGY AND SCIENCE   (India)

Author keywords

2 Arylquinolines; 3 Substituted imidazo 1,2 b pyridazines, 2 phenylimidazo 1,2 pyridines, 2 (alkoxycarbonyl)imidazo 2,1 b benzothiazoles; BZR; Non benzodiazepines; QSAR

Indexed keywords

2 (ALKOXYCARBONYL)IMIDAZO[2,1 B]BENZOTHIAZOLE DERIVATIVE; 2 ARYLQUINOLINE DERIVATIVE; 2 PHENYLIMIDAZO[1,2 A]PYRIDINE DERIVATIVE; BENZODIAZEPINE RECEPTOR; BENZODIAZEPINE RECEPTOR AFFECTING AGENT; DIAZEPAM; FLUNITRAZEPAM; IMIDAZO[1,2 B]PYRIDAZINE DERIVATIVE; UNCLASSIFIED DRUG;

ARTICLE; BINDING SITE; DRUG RECEPTOR BINDING; PHYSICAL CHEMISTRY; QUANTITATIVE STRUCTURE ACTIVITY RELATION; RECEPTOR AFFINITY;

ANIMALS; BINDING, COMPETITIVE; BRAIN; FLUNITRAZEPAM; IMIDAZOLES; KINETICS; MOLECULAR CONFORMATION; MOLECULAR STRUCTURE; PYRIDAZINES; PYRIDINES; QUINOLINES; RECEPTORS, GABA-A; STRUCTURE-ACTIVITY RELATIONSHIP; THIAZOLES;

EID: 0031796533     PISSN: 09680896     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0968-0896(98)00169-2     Document Type: Article

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