Quinolone nucleosides: 6,7-dihalo-N-β- and α-glycosyl-1,4-dihydro-4- oxo-quinoline-3-carboxylic acids and derivatives. Synthesis, antimicrobial and antiviral activity

Nucleosides and Nucleotides

Volumn 17, Issue 12, 1998, Pages 2255-2266

  Al Masoudi, Najim A ^a   Al Soud, Yaseen A ^b   Ehrmann, Micheal ^a   De Clercq, Erik ^c  

^a UNIVERSITY OF KONSTANZ   (Germany)

^b Katholieke Universiteit Leuven ^*  (Jordan)

^c REGA INSTITUTE FOR MEDICAL RESEARCH   (Belgium)

Author keywords

[No Author keywords available]

Indexed keywords

AMIDE; AMMONIA; AZIDE; CARBOXYLIC ACID DERIVATIVE; DEOXYRIBOSE; NUCLEOSIDE DERIVATIVE; QUINOLONE DERIVATIVE;

ANTIMICROBIAL ACTIVITY; ANTIVIRAL ACTIVITY; ARTICLE; CHEMICAL REACTION; CONTROLLED STUDY; CRYSTALLIZATION; CYTOPATHOGENIC EFFECT; DRUG SYNTHESIS; ESCHERICHIA COLI; HUMAN; HUMAN CELL; HUMAN IMMUNODEFICIENCY VIRUS 1; HUMAN IMMUNODEFICIENCY VIRUS 2; LYMPHOID CELL LINE;

ESCHERICHIA COLI; HUMAN IMMUNODEFICIENCY VIRUS; HUMAN IMMUNODEFICIENCY VIRUS 1; HUMAN IMMUNODEFICIENCY VIRUS 2;

EID: 0031758545     PISSN: 07328311     EISSN: None     Source Type: Journal    
DOI: 10.1080/07328319808004315     Document Type: Article

References (21)

1. J.T. Smith and C.S. Lewin in The Quinolones. ed. V. T. Andriole, Academic Press, London; 1988, ch. 2.
2. M. Nasr, J.C. Drach, S.H. Smith, C. Shipman and J.H. Burckhalter, J. Med. Chem., 31 1347 (1988).
3. B.R. Baker and R.R. Bramhall, J. Med. Chem., 15, 230 (1972).
4. D.C. Hooper, J.C. Wolfson, N. Eng. J. Med., 324, 384 (1991).
5. L.A. Mitscber, R.M. Zavod, P.V. Devasthale, D.T.W. Chu, L.L. Shen, P.N. Sharma and A.G. Pernet, Chemtech., 50 (1991).
6. G.Y. Lesher, E.J. Froelich, M.D. Gruett, J.H. Bailey and R.P. Brundage, J. Med. Chem., 5, 1063 (1962).
7. H. Koga, A. Itoh, S. Murayama, S. Suzue and T. Ivikura, J. Med. Chem., 23, 1358, (1980).
8. R. Wise, J.M. Andrews, L.J. Edwards, Antimicrob. Agents Chemother., 23, 559, (1983).
9. M.P. Wentland, D.M. Bailey, J.B. Cornett, R.A. Dobson, R.G. Powles, R.B. Wagner, J. Med. Chem., 27, 1103, (1984).
10. T. Miyamoto, J. Matsumoto, K. Chiba, H. Egawa, K. Shibamori, A. Minamida, Y. Nishimura, H. Okada, M. Kataoka, M. Fuzita, T. Hirose, J. Nakano, J. Med. Chem., 33, 1645 (1990).
11. T. Yoshida, Y. Yamamoto, H. Ovito, M. Kakiuchi, Y. Takahashi, M. Itakura, N. Kado, K. Mitani, Sh. Yasuda, H. Kato and Y. Itoh, Chem. Pharm. Bull., 44 (5), 1074 (1996).
12. M. Fujita, H. Egawa, T. Miyamoto, J. Nakano and J-I Matsumoto, Chem. Pharm. Bull., 44(5), 978 (1996).
13. V. Cecchetti, A. Fravolini, M. Palumbo, C. Sissi, O. Tabarrini, P. Terni and T. Xin, J. Med. Chem., 39, 4952-5957 (1996).
14. I. Mozek and B. Sket, J. Heterocyclic Chem., 31, 1293 (1994).
15. M.Q. Zhang, A. Haemers, D.V. Berghe, S.R. Pattyn and W. Bollaert, J. Heterocyclic Chem., 28, 673 (1991).
16. C. Perigaud, G. Gosslin and J.L. Imbach, Nucleosides & Nucleotides, 11, 903 (1992).
17. A. de la Cruz, J. Elguero, P. Goya, A. Martinez and E. de Clercq, J. Chem. Soc. Perkin Trans. 1, 845 (1993).
18. A.D. da Matta, A.M.R. Bernardino, G.A. Romeiro, M:R.P. de Oliveira, M.C.B.V. de Souza and V.E. Ferreia, Nucleosides & Nucleotides, 15 (49), 889 (1996).
19. D. Kaminsky, Chem. Abst., 72, 90322v (1970).
20. L. Birkofer and A. Ritter, Angew. Chem., 77, 414 (1965).
21. N.A. Al-Masoudi, Y.A. Al-Soud and A. Geyer, Spectroscopy Lett., in press.